JP2005529915A - 男性及び女性のインポテンスの治療において有用な製剤 - Google Patents
男性及び女性のインポテンスの治療において有用な製剤 Download PDFInfo
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- JP2005529915A JP2005529915A JP2004503026A JP2004503026A JP2005529915A JP 2005529915 A JP2005529915 A JP 2005529915A JP 2004503026 A JP2004503026 A JP 2004503026A JP 2004503026 A JP2004503026 A JP 2004503026A JP 2005529915 A JP2005529915 A JP 2005529915A
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- extract
- diffuser
- tunella
- arginine
- ginkgo biloba
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- A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
- A61K36/16—Ginkgophyta, e.g. Ginkgoaceae (Ginkgo family)
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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Abstract
Description
本発明は、男性及び女性の性機能障害の処置において有用な製剤に関するものである。
・それぞれ1.5〜3.5:1〜2:0.1〜0.4の重量比のトリブルス・テレストリス(Tribulus terrestris)、ツルネラ・ディフューサ(Turnera diffusa)及びシナモン・カッシア(Cinnamon cassia)の抽出物、
・ギンコ・ビローバ(Ginkgo biloba)抽出物、及び場合により
・アルギニン又はその生理学的に等価なエステル、塩もしくは前駆物質、を含有している医薬組成物に関するものである。
各700mgコーティング錠は、以下のものを含有する。
トリブルス・テレストリス 250.00mg
ツルネラ・ディフューサ 150.00mg
シナモン・カッシア 20.00mg
ギンコ・ビローバ 50.00mg
L−アルギニン 100.00mg
ダイズ多糖 55.00mg
二酸化ケイ素 14.00mg
けい化微晶質セルロース 42.00mg
ステアリン酸マグネシウム 4.00mg
ヒドロキシプロピルメチルセルロース 6.40mg
タルク 5.20mg
二酸化チタン 2.00mg
グリセリン 0.12mg
ポリソルベート80 0.80mg
キノリン 0.43mg
インジゴチン 0.05mg
各340mgカプセル剤は、以下のものを含有する。
トリブルス・テレストリス 125.00mg
ツルネラ・ディフューサ 75.00mg
シナモン・カッシア 10.00mg
ギンコ・ビローバ 25.00mg
L−アルギニン 50.00mg
ダイズ多糖 25.00mg
二酸化ケイ素 7.00mg
けい化微晶質セルロース 20.00mg
ステアリン酸マグネシウム 1.50mg
タルク 1.50mg
各700mg軟ゼラチンカプセル剤は、以下のものを含有する。
トリブルス・テレストリス 125.00mg
ツルネラ・ディフューサ 75.00mg
シナモン・カッシア 10.00mg
ギンコ・ビローバ 25.00mg
L−アルギニン 50.00mg
ダイズ多糖 20.00mg
中鎖トリグリセリド 100.00mg
ポリソルベート80 10.00mg
ダイズ油 275.00mg
コロイド状二酸化ケイ素 10.00mg
各10mLバイアルは、以下のものを含有する。
トリブルス・テレストリス 250.00mg
ツルネラ・ディフューサ 150.00mg
シナモン・カッシア 20.00mg
ギンコ・ビローバ 50.00mg
L−アルギニン塩酸塩 100.00mg
グリセリン 30000.00mg
ポリソルベート20 800.00mg
プロピレングリコール 1000.00mg
アセスルファムK 175.00mg
サッカリンナトリウム 40.00mg
ネオヘスペリジンDC 2.50mg
風味剤 300.00mg
ソルビン酸カリウム 11.70mg
メチルパラベン 8.30mg
精製水 10.00mLにするのに十分な量
各5000mg包装袋(sachet)は、以下のものを含有する。
トリブルス・テレストリス 250.00mg
ツルネラ・ディフューサ 150.00mg
シナモン・カッシア 20.00mg
ギンコ・ビローバ 50.00mg
L−アルギニン塩酸塩 100.00mg
ポリソルベート20 500.00mg
アセスルファムK 175.00mg
サッカリンナトリウム 40.00mg
ネオヘスペリジンDC 2.50mg
風味剤 300.00mg
イヌリン 1000.00mg
マンニトール 2412.50mg
Claims (10)
- 適当な担体又は賦形剤と混和された、
・それぞれ1.5〜3.5:1〜2:0.1〜0.4の重量比のトリブルス・テレストリス、ツルネラ・ディフューサ及びシナモン・カッシアの抽出物、
・ギンコ・ビローバの抽出物、及び場合により
・アルギニン又はその生理学的に等価なエステル、塩もしくは前駆物質、を含有している医薬組成物。 - トリブルス・テレストリス、ツルネラ・ディフューサ及びシナモン・カッシアの抽出物の重量比が、2.5:1.5:0.2である、請求項1に記載の組成物。
- ギンコ・ビローバ抽出物が、アピゲニン二量体フラボノイドの画分により構成されている、請求項1又は2に記載の組成物。
- アピゲニン二量体フラボノイドの画分50mgを含有している、請求項3に記載の組成物。
- それぞれ1.5〜3.5:1〜2:0.1〜0.4:0.5〜1.5の重量比のトリブルス・テレストリス、ツルネラ・ディフューサ及びシナモン・カッシアの抽出物、並びにL−アルギニン又はL−アルギニン塩酸塩を含有している、請求項1〜4のいずれかに記載の組成物。
- トリブルス・テレストリス、ツルネラ・ディフューサ及びシナモン・カッシアの抽出物、並びにL−アルギニン又はL−アルギニン塩酸塩の重量比が、2.5:1.5:0.2:1である、請求項5に記載の組成物。
- 男性及び女性の性機能障害の処置のための医薬品の調製のための、ギンコ・ビローバ抽出物、及び場合によりアルギニン又はその生理学的に等価なエステル、塩もしくは前駆物質と組み合わせられた、それぞれ1.5〜3.5:1〜2:0.1〜0.4の重量比のトリブルス・テレストリス、ツルネラ・ディフューサ及びシナモン・カッシアの抽出物の使用。
- インポテンス、勃起機能障害、性欲障害、不感症及び無オルガズム症を処置するための、請求項7に記載の使用。
- ジオスシン、ツルネラ・ディフューサの親油性抽出物、ギンコ・ビローバの二量体フラボン及びケイ皮アルデヒドを含む医薬組成物。
- 男性及び女性の性機能障害の処置のための医薬品の調製のための、ジオスシン、ツルネラ・ディフューサの親油性抽出物、ギンコ・ビローバの二量体フラボン及びケイ皮アルデヒドの使用。
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
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IT2002MI000990A ITMI20020990A1 (it) | 2002-05-10 | 2002-05-10 | Formulazioni utili nel trattamento dell'impotenza maschile e femminile |
PCT/EP2003/004528 WO2003094943A1 (en) | 2002-05-10 | 2003-04-30 | Formulations useful in the treatment of male and female impotence |
Publications (2)
Publication Number | Publication Date |
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JP2005529915A true JP2005529915A (ja) | 2005-10-06 |
JP4603351B2 JP4603351B2 (ja) | 2010-12-22 |
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JP2004503026A Expired - Fee Related JP4603351B2 (ja) | 2002-05-10 | 2003-04-30 | 男性及び女性のインポテンスの治療において有用な製剤 |
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US (1) | US7128932B2 (ja) |
EP (2) | EP1658854B1 (ja) |
JP (1) | JP4603351B2 (ja) |
KR (1) | KR20040102212A (ja) |
CN (2) | CN101164559A (ja) |
AT (2) | ATE319466T1 (ja) |
AU (1) | AU2003240478B8 (ja) |
CA (1) | CA2485264A1 (ja) |
DE (2) | DE60303925T2 (ja) |
DK (2) | DK1503775T3 (ja) |
ES (2) | ES2259139T3 (ja) |
HK (1) | HK1085374A1 (ja) |
IL (2) | IL165081A (ja) |
IT (1) | ITMI20020990A1 (ja) |
NO (2) | NO332805B1 (ja) |
PT (2) | PT1658854E (ja) |
RU (2) | RU2313357C2 (ja) |
SI (2) | SI1658854T1 (ja) |
WO (1) | WO2003094943A1 (ja) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2007508292A (ja) * | 2003-10-10 | 2007-04-05 | エティファルム | イチョウ・エキスを含む放出持続性の微小顆粒およびそのような顆粒の製造方法 |
JP2020536590A (ja) * | 2017-10-13 | 2020-12-17 | クリスタルファルマ・ソチエタ・ア・レスポンサビリタ・リミタータ | 老化によって引き起こされる女性の障害を緩和するためのサプリメント |
Families Citing this family (19)
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US6952691B2 (en) * | 2002-02-01 | 2005-10-04 | International Business Machines Corporation | Method and system for searching a multi-lingual database |
WO2006021930A2 (en) * | 2004-08-25 | 2006-03-02 | Femi-X A/S | Aphrodisiac herbal composition for a female comprising epimedium grandiflorum, turnera diffusa var. aphrodisiaca, ilex paraguariensis and smilax spp |
KR100660116B1 (ko) * | 2005-01-26 | 2006-12-20 | (주)포메디 | 홍삼 및 대두를 주성분으로 포함하는 복합 한방 제제를유효성분으로 함유하는 성기능 개선용 조성물 |
US20070042054A1 (en) * | 2005-04-20 | 2007-02-22 | Council Of Scientific And Industrial Research | Functional aphrodisiac rolled herbal bidis and cigarettes |
EP1932531A1 (de) | 2006-12-11 | 2008-06-18 | Finzelberg GmbH & Co. KG | Spezialextrakt und seine Verwendung zur Hemmung des Abbaus von cyclischem Guanosinmonophosphat (cGMP) |
US8362088B2 (en) * | 2006-12-14 | 2013-01-29 | Warnock W Matthew | Method and article of manufacture for encapsulating a homeopathic ingredient with a second ingredient |
US20100178413A1 (en) * | 2008-12-17 | 2010-07-15 | Mark Gorris | Food-based Supplement Delivery System |
US9918489B2 (en) * | 2008-12-17 | 2018-03-20 | Mark Gorris | Food-based supplement delivery system |
CN102612370B (zh) * | 2009-09-17 | 2014-10-29 | 特拉达药物有限公司 | 刺激男性性功能的膳食补充剂 |
ES2386859B1 (es) * | 2011-02-07 | 2013-03-22 | Eduardo Antonio Gómez De Diego | Composición natural para aumentar el vigor. |
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ITLI20110007A1 (it) * | 2011-09-10 | 2013-03-11 | Lloyds Internat Credit Llc | Una innovativa composizione naturale efficace per la cura dell'impotenza |
TW201420745A (zh) * | 2012-11-26 | 2014-06-01 | Tian-De Li | 擴充男性海綿體的複方精油 |
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EP3560488A1 (en) * | 2018-04-24 | 2019-10-30 | Procare Health Iberia, S.L. | Compositions for treating female sexual dysfunction |
WO2022027122A1 (en) * | 2020-08-06 | 2022-02-10 | Ramade & Cia Holding Corp. | Compositions with cannabinoids of cannabis sativa for treating erectile and sexual dysfunction |
IT202100031175A1 (it) * | 2021-12-13 | 2023-06-13 | Anvest Group S R L | Composizione per il trattamento della disfunzione erettile |
GR1010519B (el) * | 2022-07-04 | 2023-08-10 | Νικολαος Τυμπανιδης | Καταπινομενο σκευασμα για τονωση της ζωτικοτητας, της αντοχης και της γενικοτερης ευεξιας των ανδρων |
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