JP2005523326A - プロテインキナーゼｃのペプチドインヒビター - Google Patents
プロテインキナーゼｃのペプチドインヒビター Download PDFInfo
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
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Landscapes
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US37453002P | 2002-04-22 | 2002-04-22 | |
| PCT/US2003/012541 WO2003089456A2 (en) | 2002-04-22 | 2003-04-22 | Peptide inhibitors of protein kinase c |
Related Child Applications (2)
| Application Number | Title | Priority Date | Filing Date |
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| JP2009011456A Division JP2009102392A (ja) | 2002-04-22 | 2009-01-21 | プロテインキナーゼｃのペプチドインヒビター |
| JP2012128849A Division JP2012176978A (ja) | 2002-04-22 | 2012-06-06 | プロテインキナーゼｃのペプチドインヒビター |
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| JP2005523326A true JP2005523326A (ja) | 2005-08-04 |
| JP2005523326A5 JP2005523326A5 (OSRAM) | 2006-05-25 |
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| JP2003586176A Withdrawn JP2005523326A (ja) | 2002-04-22 | 2003-04-22 | プロテインキナーゼｃのペプチドインヒビター |
| JP2003586177A Pending JP2005527209A (ja) | 2002-04-22 | 2003-04-22 | 疼痛管理のためのプロテインキナーゼＣγのペプチドインヒビター |
| JP2009010402A Pending JP2009091372A (ja) | 2002-04-22 | 2009-01-20 | 疼痛管理のためのプロテインキナーゼＣγのペプチドインヒビター |
| JP2009011456A Pending JP2009102392A (ja) | 2002-04-22 | 2009-01-21 | プロテインキナーゼｃのペプチドインヒビター |
| JP2012128849A Pending JP2012176978A (ja) | 2002-04-22 | 2012-06-06 | プロテインキナーゼｃのペプチドインヒビター |
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| JP2009010402A Pending JP2009091372A (ja) | 2002-04-22 | 2009-01-20 | 疼痛管理のためのプロテインキナーゼＣγのペプチドインヒビター |
| JP2009011456A Pending JP2009102392A (ja) | 2002-04-22 | 2009-01-21 | プロテインキナーゼｃのペプチドインヒビター |
| JP2012128849A Pending JP2012176978A (ja) | 2002-04-22 | 2012-06-06 | プロテインキナーゼｃのペプチドインヒビター |
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| EP (3) | EP1501533A4 (OSRAM) |
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| CA (3) | CA2785889A1 (OSRAM) |
| WO (2) | WO2003089457A2 (OSRAM) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005527209A (ja) * | 2002-04-22 | 2005-09-15 | ザ ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティー | 疼痛管理のためのプロテインキナーゼＣγのペプチドインヒビター |
| JP2009508879A (ja) * | 2005-09-19 | 2009-03-05 | カイ ファーマシューティカルズ インコーポレーティッド | 血管新生のプロテインキナーゼｃペプチドモジュレーター |
| JP2010516707A (ja) * | 2007-01-19 | 2010-05-20 | カイ ファーマシューティカルズ インコーポレーティッド | ペプチド組成物の安定性および送達効率を上昇させるための修飾方法 |
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| US6933275B2 (en) | 2002-05-01 | 2005-08-23 | The Board Of Trustees Of The Leland Stanford Junior University | Protein kinase C peptides for use in withdrawal |
| WO2004084889A1 (en) * | 2003-03-28 | 2004-10-07 | Pfizer Inc. | Use of protein kinase c inhibitor for suppressing sustained slow postsynaptic excitation (sspe) of enteric neurons |
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| AU2003264918A1 (en) * | 2003-10-02 | 2005-04-21 | The Board Of Trustees Of The Leland Stanford Junior University | Protein kinase c peptides for use in withdrawal |
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| EP1877424A4 (en) * | 2005-04-11 | 2010-09-29 | Pharmagap Inc | INHIBITORS OF PROTEIN KINASES AND USES THEREOF |
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-
2003
- 2003-04-22 CA CA2785889A patent/CA2785889A1/en not_active Abandoned
- 2003-04-22 EP EP03728495A patent/EP1501533A4/en not_active Withdrawn
- 2003-04-22 WO PCT/US2003/012542 patent/WO2003089457A2/en not_active Ceased
- 2003-04-22 AU AU2003234185A patent/AU2003234185C1/en not_active Ceased
- 2003-04-22 WO PCT/US2003/012541 patent/WO2003089456A2/en not_active Ceased
- 2003-04-22 EP EP10178878A patent/EP2332559A1/en not_active Withdrawn
- 2003-04-22 JP JP2003586176A patent/JP2005523326A/ja not_active Withdrawn
- 2003-04-22 US US10/513,003 patent/US7393835B2/en not_active Expired - Fee Related
- 2003-04-22 US US10/421,548 patent/US7459424B2/en not_active Expired - Fee Related
- 2003-04-22 CA CA2481512A patent/CA2481512C/en not_active Expired - Fee Related
- 2003-04-22 AU AU2003234186A patent/AU2003234186B2/en not_active Ceased
- 2003-04-22 US US10/421,503 patent/US7507711B2/en not_active Expired - Fee Related
- 2003-04-22 JP JP2003586177A patent/JP2005527209A/ja active Pending
- 2003-04-22 CA CA2482598A patent/CA2482598C/en not_active Expired - Fee Related
- 2003-04-22 EP EP03728494A patent/EP1501532A4/en not_active Withdrawn
-
2007
- 2007-07-16 US US11/879,414 patent/US7833984B2/en not_active Expired - Fee Related
-
2008
- 2008-06-16 US US12/214,104 patent/US7939493B2/en not_active Expired - Fee Related
- 2008-08-27 US US12/229,992 patent/US20090143293A1/en not_active Abandoned
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2009
- 2009-01-20 JP JP2009010402A patent/JP2009091372A/ja active Pending
- 2009-01-21 JP JP2009011456A patent/JP2009102392A/ja active Pending
- 2009-04-22 AU AU2009201593A patent/AU2009201593B2/en not_active Ceased
- 2009-05-04 AU AU2009201760A patent/AU2009201760B2/en not_active Ceased
-
2011
- 2011-05-05 US US13/101,540 patent/US8658594B2/en not_active Expired - Fee Related
-
2012
- 2012-06-06 JP JP2012128849A patent/JP2012176978A/ja active Pending
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2014
- 2014-02-21 US US14/187,070 patent/US9365837B2/en not_active Expired - Fee Related
Cited By (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005527209A (ja) * | 2002-04-22 | 2005-09-15 | ザ ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティー | 疼痛管理のためのプロテインキナーゼＣγのペプチドインヒビター |
| JP2009091372A (ja) * | 2002-04-22 | 2009-04-30 | Board Of Trustees Of The Leland Stanford Junior Univ | 疼痛管理のためのプロテインキナーゼＣγのペプチドインヒビター |
| US8658594B2 (en) | 2002-04-22 | 2014-02-25 | Board of Trustees of the Leland Stanford Junior Universit | Peptide inhibitors of protein kinase C |
| US9365837B2 (en) | 2002-04-22 | 2016-06-14 | The Board Of Trustees Of The Leland Stanford Junior University | Peptide inhibitors of protein kinase C |
| JP2009508879A (ja) * | 2005-09-19 | 2009-03-05 | カイ ファーマシューティカルズ インコーポレーティッド | 血管新生のプロテインキナーゼｃペプチドモジュレーター |
| JP2010516707A (ja) * | 2007-01-19 | 2010-05-20 | カイ ファーマシューティカルズ インコーポレーティッド | ペプチド組成物の安定性および送達効率を上昇させるための修飾方法 |
| JP2014224126A (ja) * | 2007-01-19 | 2014-12-04 | カイ ファーマシューティカルズ インコーポレーティッド | ペプチド組成物の安定性および送達効率を上昇させるための修飾方法 |
| JP2016147905A (ja) * | 2007-01-19 | 2016-08-18 | カイ ファーマシューティカルズ インコーポレーティッド | ペプチド組成物の安定性および送達効率を上昇させるための修飾方法 |
| JP2018111717A (ja) * | 2007-01-19 | 2018-07-19 | カイ ファーマシューティカルズ インコーポレーティッド | ペプチド組成物の安定性および送達効率を上昇させるための修飾方法 |
| JP2021098725A (ja) * | 2007-01-19 | 2021-07-01 | カイ ファーマシューティカルズ インコーポレーティッド | ペプチド組成物の安定性および送達効率を上昇させるための修飾方法 |
| JP2023078424A (ja) * | 2007-01-19 | 2023-06-06 | カイ ファーマシューティカルズ インコーポレーティッド | ペプチド組成物の安定性および送達効率を上昇させるための修飾方法 |
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