JP2005519052A - プラバスタチン医薬製剤及びその使用方法 - Google Patents
プラバスタチン医薬製剤及びその使用方法 Download PDFInfo
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- JP2005519052A JP2005519052A JP2003557553A JP2003557553A JP2005519052A JP 2005519052 A JP2005519052 A JP 2005519052A JP 2003557553 A JP2003557553 A JP 2003557553A JP 2003557553 A JP2003557553 A JP 2003557553A JP 2005519052 A JP2005519052 A JP 2005519052A
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- pravastatin
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- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
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- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/22—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acyclic acids, e.g. pravastatin
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- A61K9/2833—Organic macromolecular compounds
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- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
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- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
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- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
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- Chemical & Material Sciences (AREA)
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- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US34777502P | 2002-01-11 | 2002-01-11 | |
| US40726902P | 2002-09-03 | 2002-09-03 | |
| PCT/IB2003/000336 WO2003057195A1 (en) | 2002-01-11 | 2003-01-10 | Pravastatin pharmaceutical formulations and methods of their use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005519052A true JP2005519052A (ja) | 2005-06-30 |
| JP2005519052A5 JP2005519052A5 (enExample) | 2006-01-05 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| JP2003557553A Pending JP2005519052A (ja) | 2002-01-11 | 2003-01-10 | プラバスタチン医薬製剤及びその使用方法 |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US6967218B2 (enExample) |
| EP (1) | EP1465605A1 (enExample) |
| JP (1) | JP2005519052A (enExample) |
| AU (1) | AU2003201735B2 (enExample) |
| CA (1) | CA2473106A1 (enExample) |
| IL (1) | IL162937A0 (enExample) |
| MX (1) | MXPA04006780A (enExample) |
| NO (1) | NO20043333L (enExample) |
| WO (1) | WO2003057195A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021517141A (ja) * | 2018-03-09 | 2021-07-15 | ザ・ブリガーム・アンド・ウーメンズ・ホスピタル・インコーポレーテッド | 心血管疾患のための組み合わせ治療 |
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| EP1465605A1 (en) * | 2002-01-11 | 2004-10-13 | Athpharma Limited | Pravastatin pharmaceutical formulations and methods of their use |
| US20050089572A1 (en) * | 2002-03-22 | 2005-04-28 | Manoj Kumar | Controlled release drug delivery system of pravastatin |
| SI21400A (sl) * | 2003-02-12 | 2004-08-31 | LEK farmacevtska družba d.d. | Stabilna farmacevtska oblika z inhibitorjem HMG-CoA reduktaze |
| US8987322B2 (en) | 2003-11-04 | 2015-03-24 | Circ Pharma Research And Development Limited | Pharmaceutical formulations for carrier-mediated transport statins and uses thereof |
| ES2684325T5 (es) * | 2004-01-20 | 2024-06-10 | Novartis Ag | Formulación y proceso de compresión directa |
| CN101618216B (zh) * | 2004-01-20 | 2012-01-04 | 诺瓦提斯公司 | 直接压片配方和方法 |
| EP1563837A1 (en) * | 2004-02-03 | 2005-08-17 | Ferrer Internacional, S.A. | Hypocholesterolemic compositions comprising a statin and an antiflatulent agent |
| AU2005305459A1 (en) * | 2004-11-22 | 2006-05-26 | Dexcel Pharma Technologies Ltd. | Controlled absorption of statins in the intestine |
| GR1006879B (el) * | 2005-09-14 | 2010-07-13 | "Φαρματεν" Φαρμακευτικη Βιομηχανικη Εμπορικη Α.Ε., | Βελτιωμενες φαρμακευτικες συνθεσεις που περιεχουν αναστολεις της αναγωγασης του 3-υδροξυ-3-μεθυλογλουταρυλοσυνενζυμου α (hmg-coa) και μεθοδος παρασκευης αυτων |
| US20100055173A1 (en) * | 2006-10-10 | 2010-03-04 | Adel Penhasi | Release of statins in the intestine |
| GB0713707D0 (en) * | 2007-07-13 | 2007-08-22 | Generics Uk Ltd | Stable compositions |
| US20090226516A1 (en) * | 2008-03-04 | 2009-09-10 | Pharma Pass Ii Llc | Sartan compositions |
| US20090226515A1 (en) * | 2008-03-04 | 2009-09-10 | Pharma Pass Ii Llc | Statin compositions |
| JP2013535516A (ja) * | 2010-08-17 | 2013-09-12 | ルピン・リミテッド | ドロネダロンの制御放出製剤 |
| EP2692354A1 (en) * | 2012-08-03 | 2014-02-05 | Max-Delbrück-Centrum für Molekulare Medizin (MDC) | Means for treating heart disease |
| CN111803462A (zh) * | 2020-07-15 | 2020-10-23 | 浙江诺得药业有限公司 | 一种普伐他汀钠肠溶片及其制备方法 |
Family Cites Families (17)
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| US4904474A (en) * | 1988-01-25 | 1990-02-27 | Alza Corporation | Delivery of drug to colon by oral disage form |
| US5180589A (en) * | 1988-03-31 | 1993-01-19 | E. R. Squibb & Sons, Inc. | Pravastatin pharmaceuatical compositions having good stability |
| US5030447A (en) * | 1988-03-31 | 1991-07-09 | E. R. Squibb & Sons, Inc. | Pharmaceutical compositions having good stability |
| US4997658A (en) * | 1988-11-21 | 1991-03-05 | Merck & Co., Inc. | Method for enhancing the lowering of plasma cholesterol levels |
| US5376383A (en) * | 1988-11-21 | 1994-12-27 | Merck & Co., Inc. | Method for enhancing the lowering of plasma-cholesterol levels |
| EP0465096A1 (en) | 1990-06-26 | 1992-01-08 | Merck & Co. Inc. | Plasma cholesterol level lowering composition |
| US5916595A (en) * | 1997-12-12 | 1999-06-29 | Andrx Pharmaceutials, Inc. | HMG co-reductase inhibitor |
| UA69413C2 (uk) * | 1998-05-22 | 2004-09-15 | Брістол-Майерс Сквібб Компані | Фармацевтична композиція, яка містить серцевину та ентеросолюбільну оболонку, фармацевтична композиція у вигляді сфероїдальних гранул, спосіб одержання сфероїдальних гранул та спосіб одержання фармацевтичної композиції |
| UA73092C2 (uk) * | 1998-07-17 | 2005-06-15 | Брістол-Майерс Сквібб Компані | Таблетка з ентеросолюбільним покриттям і спосіб її приготування |
| AU2161000A (en) | 1998-12-07 | 2000-06-26 | Bristol-Myers Squibb Company | Enteric coated pravastatin bead formulation |
| SI20109A (sl) * | 1998-12-16 | 2000-06-30 | LEK, tovarna farmacevtskih in kemi�nih izdelkov, d.d. | Stabilna farmacevtska formulacija |
| NZ513037A (en) * | 1999-01-29 | 2003-05-30 | Disphar Internat B | Coated sustained release pharmaceutical composition for the release of an agent in the gastrointestinal tract |
| US6569461B1 (en) * | 1999-03-08 | 2003-05-27 | Merck & Co., Inc. | Dihydroxy open-acid and salts of HMG-CoA reductase inhibitors |
| CA2404044A1 (en) * | 2000-04-11 | 2001-10-18 | Atherogenics, Inc. | Compounds and methods to increase plasma hdl cholesterol levels and improve hdl functionality |
| US6936731B2 (en) * | 2000-10-05 | 2005-08-30 | TEVA Gyógyszergyár Részvénytársaság | Pravastatin sodium substantially free of pravastatin lactone and epi-pravastatin, and compositions containing same |
| US20030091630A1 (en) * | 2001-10-25 | 2003-05-15 | Jenny Louie-Helm | Formulation of an erodible, gastric retentive oral dosage form using in vitro disintegration test data |
| EP1465605A1 (en) * | 2002-01-11 | 2004-10-13 | Athpharma Limited | Pravastatin pharmaceutical formulations and methods of their use |
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- 2003-01-10 AU AU2003201735A patent/AU2003201735B2/en not_active Ceased
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- 2003-01-10 MX MXPA04006780A patent/MXPA04006780A/es unknown
- 2003-01-10 WO PCT/IB2003/000336 patent/WO2003057195A1/en not_active Ceased
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- 2003-01-10 US US10/339,487 patent/US6967218B2/en not_active Expired - Fee Related
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2021517141A (ja) * | 2018-03-09 | 2021-07-15 | ザ・ブリガーム・アンド・ウーメンズ・ホスピタル・インコーポレーテッド | 心血管疾患のための組み合わせ治療 |
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| US20030176502A1 (en) | 2003-09-18 |
| CA2473106A1 (en) | 2003-07-17 |
| IL162937A0 (en) | 2005-11-20 |
| WO2003057195A1 (en) | 2003-07-17 |
| NO20043333L (no) | 2004-09-13 |
| EP1465605A1 (en) | 2004-10-13 |
| AU2003201735A1 (en) | 2003-07-24 |
| US20050277691A1 (en) | 2005-12-15 |
| MXPA04006780A (es) | 2005-06-08 |
| AU2003201735B2 (en) | 2008-11-13 |
| US6967218B2 (en) | 2005-11-22 |
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