JP2005508955A - ヘルペスウイルス感染の治療で使用されるためのイミダゾ−ピリジン誘導体 - Google Patents

ヘルペスウイルス感染の治療で使用されるためのイミダゾ−ピリジン誘導体 Download PDF

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JP2005508955A
JP2005508955A JP2003534429A JP2003534429A JP2005508955A JP 2005508955 A JP2005508955 A JP 2005508955A JP 2003534429 A JP2003534429 A JP 2003534429A JP 2003534429 A JP2003534429 A JP 2003534429A JP 2005508955 A JP2005508955 A JP 2005508955A
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formula
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cycloalkyl
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JP2005508955A5 (cg-RX-API-DMAC7.html
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グドムンドソン,クリスティアン
ジョーンズ,ブライアン,エー.
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スミスクライン ビーチャム コーポレーション
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Publication of JP2005508955A5 publication Critical patent/JP2005508955A5/ja
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP2003534429A 2001-10-05 2002-09-23 ヘルペスウイルス感染の治療で使用されるためのイミダゾ−ピリジン誘導体 Pending JP2005508955A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32770501P 2001-10-05 2001-10-05
PCT/US2002/030056 WO2003031446A1 (en) 2001-10-05 2002-09-23 Imidazo-pyridine derivatives for use in the treatment of herpes viral infection

Publications (2)

Publication Number Publication Date
JP2005508955A true JP2005508955A (ja) 2005-04-07
JP2005508955A5 JP2005508955A5 (cg-RX-API-DMAC7.html) 2005-12-22

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JP2003534429A Pending JP2005508955A (ja) 2001-10-05 2002-09-23 ヘルペスウイルス感染の治療で使用されるためのイミダゾ−ピリジン誘導体

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US (2) US7244740B2 (cg-RX-API-DMAC7.html)
EP (1) EP1432712B1 (cg-RX-API-DMAC7.html)
JP (1) JP2005508955A (cg-RX-API-DMAC7.html)
AT (1) ATE326466T1 (cg-RX-API-DMAC7.html)
DE (1) DE60211539T2 (cg-RX-API-DMAC7.html)
ES (1) ES2262893T3 (cg-RX-API-DMAC7.html)
WO (1) WO2003031446A1 (cg-RX-API-DMAC7.html)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008059714A1 (en) * 2006-11-17 2008-05-22 Nihon Medi-Physics Co., Ltd. Novel compounds with affinity for amyloid
WO2009057577A1 (ja) * 2007-10-30 2009-05-07 Nihon Medi-Physics Co., Ltd. 新規アミロイド親和性化合物の使用及び製造方法
JP2020505419A (ja) * 2017-02-01 2020-02-20 オーセントラ セラピュティクス ピーティーワイ エルティーディーAucentra Therapeutics Pty Ltd 治療薬としてのN−シクロアルキル/ヘテロシクロアルキル−4−(イミダゾ[1,2−a]ピリジン)ピリミジン−2−アミン誘導体

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DE60214179T2 (de) * 2001-06-21 2007-01-04 Smithkline Beecham Corp. Imidazo-1,2-A/Pyriden-Derivate zur Prophylaxe und Behandlung von Herpes-Infektionen
JP2005525382A (ja) 2002-03-07 2005-08-25 スミスクライン ビーチャム コーポレーション ピラゾロピリミジンおよびピラゾロトリアジン誘導体ならびにそれを含む医薬組成物
GB0205693D0 (en) 2002-03-09 2002-04-24 Astrazeneca Ab Chemical compounds
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GB0205688D0 (en) 2002-03-09 2002-04-24 Astrazeneca Ab Chemical compounds
JP2006520819A (ja) * 2003-03-06 2006-09-14 メルク エンド カムパニー インコーポレーテッド 抗原虫薬イミダゾピリジン化合物
GB0311274D0 (en) 2003-05-16 2003-06-18 Astrazeneca Ab Chemical compounds
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TW200528101A (en) 2004-02-03 2005-09-01 Astrazeneca Ab Chemical compounds
UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
EP2303881A2 (en) 2008-07-14 2011-04-06 Gilead Sciences, Inc. Fused heterocyclyc inhibitors of histone deacetylase and/or cyclin-dependent kinases
NZ590283A (en) 2008-07-14 2012-11-30 Gilead Sciences Inc Imidazolylpyrimidine compounds as hdac and / or cdk inhibitors
US8344018B2 (en) 2008-07-14 2013-01-01 Gilead Sciences, Inc. Oxindolyl inhibitor compounds
EP2326622A1 (en) 2008-07-28 2011-06-01 Gilead Sciences, Inc. Cycloalkylidene and heterocycloalkylidene histone deacetylase inhibitor compounds
EP2440517B1 (en) 2009-06-08 2014-03-26 Gilead Sciences, Inc. Cycloalkylcarbamate benzamide aniline hdac inhibitor compounds
CA2763786C (en) 2009-06-08 2014-09-30 Gilead Sciences, Inc. Alkanoylamino benzamide aniline hdac inihibitor compounds
KR101774035B1 (ko) 2009-10-30 2017-09-01 얀센 파마슈티카 엔.브이. 이미다조[1,2―b]피리다진 유도체 및 PDE10 저해제로서의 그의 용도
AR080754A1 (es) 2010-03-09 2012-05-09 Janssen Pharmaceutica Nv Derivados de imidazo (1,2-a) pirazina y su uso como inhibidores de pde10
EA027418B1 (ru) 2011-06-27 2017-07-31 Янссен Фармацевтика Нв ПРОИЗВОДНЫЕ 1-АРИЛ-4-МЕТИЛ[1,2,4]ТРИАЗОЛО[4,3-a]ХИНОКСАЛИНА, ФАРМАЦЕВТИЧЕСКАЯ КОМПОЗИЦИЯ НА ИХ ОСНОВЕ, СПОСОБЫ ПОЛУЧЕНИЯ И ПРИМЕНЕНИЯ ИХ, ПРОМЕЖУТОЧНЫЕ СОЕДИНЕНИЯ
ES2855575T3 (es) 2012-06-26 2021-09-23 Janssen Pharmaceutica Nv Combinaciones que comprenden compuestos de 4-metil-[1,2,4]triazolo[4,3-a]quinoxalina como inhibidores de PDE2 e inhibidores de PDE10 para su uso en el tratamiento de trastornos neurológicos o metabólicos
KR102171706B1 (ko) 2012-07-09 2020-10-30 얀센 파마슈티카 엔.브이. 포스포디에스테라아제 10 효소의 억제제
CN120829428A (zh) * 2024-04-18 2025-10-24 中国医学科学院药物研究所 咪唑并吡啶衍生物及其用途

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Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2008059714A1 (en) * 2006-11-17 2008-05-22 Nihon Medi-Physics Co., Ltd. Novel compounds with affinity for amyloid
JPWO2008059714A1 (ja) * 2006-11-17 2010-03-04 日本メジフィジックス株式会社 新規アミロイド親和性化合物
WO2009057577A1 (ja) * 2007-10-30 2009-05-07 Nihon Medi-Physics Co., Ltd. 新規アミロイド親和性化合物の使用及び製造方法
JP2020505419A (ja) * 2017-02-01 2020-02-20 オーセントラ セラピュティクス ピーティーワイ エルティーディーAucentra Therapeutics Pty Ltd 治療薬としてのN−シクロアルキル/ヘテロシクロアルキル−4−(イミダゾ[1,2−a]ピリジン)ピリミジン−2−アミン誘導体
JP7113528B2 (ja) 2017-02-01 2022-08-05 オーセントラ セラピュティクス ピーティーワイ エルティーディー 治療薬としてのN-シクロアルキル/ヘテロシクロアルキル-4-(イミダゾ[1,2-a]ピリジン)ピリミジン-2-アミン誘導体

Also Published As

Publication number Publication date
US20080139594A1 (en) 2008-06-12
US7244740B2 (en) 2007-07-17
DE60211539D1 (de) 2006-06-22
DE60211539T2 (de) 2006-09-21
ATE326466T1 (de) 2006-06-15
ES2262893T3 (es) 2006-12-01
EP1432712B1 (en) 2006-05-17
EP1432712A1 (en) 2004-06-30
WO2003031446A1 (en) 2003-04-17
US20040248917A1 (en) 2004-12-09

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