JP2005507372A5 - - Google Patents

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Publication number
JP2005507372A5
JP2005507372A5 JP2002591483A JP2002591483A JP2005507372A5 JP 2005507372 A5 JP2005507372 A5 JP 2005507372A5 JP 2002591483 A JP2002591483 A JP 2002591483A JP 2002591483 A JP2002591483 A JP 2002591483A JP 2005507372 A5 JP2005507372 A5 JP 2005507372A5
Authority
JP
Japan
Prior art keywords
phenyl
methyl
ylidene
benzamide
diisopropyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002591483A
Other languages
English (en)
Japanese (ja)
Other versions
JP2005507372A (ja
Filing date
Publication date
Priority claimed from SE0101767A external-priority patent/SE0101767D0/xx
Application filed filed Critical
Publication of JP2005507372A publication Critical patent/JP2005507372A/ja
Publication of JP2005507372A5 publication Critical patent/JP2005507372A5/ja
Pending legal-status Critical Current

Links

JP2002591483A 2001-05-18 2002-05-16 ４−（フェニル−ピペリジン−４−イリデン−メチル）−ベンズアミド誘導体及び疼痛、不安症又は胃腸障害の治療のためのその使用 Pending JP2005507372A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0101767A SE0101767D0 (sv) 2001-05-18 2001-05-18 Novel compounds
PCT/SE2002/000946 WO2002094810A1 (en) 2001-05-18 2002-05-16 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders

Publications (2)

Publication Number Publication Date
JP2005507372A JP2005507372A (ja) 2005-03-17
JP2005507372A5 true JP2005507372A5 (OSRAM) 2005-12-22

Family

ID=20284170

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002591483A Pending JP2005507372A (ja) 2001-05-18 2002-05-16 ４−（フェニル−ピペリジン−４−イリデン−メチル）−ベンズアミド誘導体及び疼痛、不安症又は胃腸障害の治療のためのその使用

Country Status (25)

Country Link
US (1) US20040138259A1 (OSRAM)
EP (1) EP1395574B1 (OSRAM)
JP (1) JP2005507372A (OSRAM)
KR (1) KR20030094423A (OSRAM)
CN (1) CN1547579A (OSRAM)
AR (1) AR033756A1 (OSRAM)
AT (1) ATE287400T1 (OSRAM)
BG (1) BG108328A (OSRAM)
BR (1) BR0209667A (OSRAM)
CA (1) CA2446331A1 (OSRAM)
CO (1) CO5540304A2 (OSRAM)
CZ (1) CZ20033087A3 (OSRAM)
DE (1) DE60202679T2 (OSRAM)
EE (1) EE200300543A (OSRAM)
HU (1) HUP0401285A2 (OSRAM)
IL (1) IL158695A0 (OSRAM)
IS (1) IS7024A (OSRAM)
MX (1) MXPA03010438A (OSRAM)
NO (1) NO20035118D0 (OSRAM)
PL (1) PL366389A1 (OSRAM)
RU (1) RU2003131968A (OSRAM)
SE (1) SE0101767D0 (OSRAM)
SK (1) SK13932003A3 (OSRAM)
WO (1) WO2002094810A1 (OSRAM)
ZA (1) ZA200308635B (OSRAM)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CL2004000754A1 (es) * 2003-04-11 2005-02-25 Janssen Pharmaceutica Nv Uso de compuestos derivados de 4-fenil-4-(1h-imidazol-2-il)piperidina, como agonistas delta-opioides no peptidicos, para preparar un medicamento util en prevenir o tratar trastornos del sistema nervioso central.
SE0301443D0 (sv) * 2003-05-16 2003-05-16 Astrazeneca Ab Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
EP1641757A1 (en) * 2003-05-16 2006-04-05 AstraZeneca AB Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
WO2005005478A2 (en) * 2003-07-02 2005-01-20 Bayer Healthcare Ag Diagnostics and therapeutics for diseases associated with g protein-coupled opioid receptor; delta 1 (oprd1)
BRPI0415165A (pt) 2003-10-01 2007-01-09 Adolor Corp composto heterocìclico espirocìclico, composição farmacêutica, método para ligar receptores opióides, métodos para prevenir ou tratar dor, disfunção gastrointestinal, um distúrbio do trato urogenital, um distúrbio imunomodulatório, um distúrbio inflamatório, um distúrbio de função respiratória, ansiedade, distúrbio do humor, um distúrbio relacionado a estresse, distúrbio do sistema nervoso simpático, tosse, e um distúrbio motor, método para tratar uma lesão traumática ao sistema nervoso central, métodos para prevenir ou tratar acidente vascular, arritmia cardìaca, glaucoma, e disfunção sexual, métodos para tratar uma condição selecionada do grupo consistindo de choque, edema cerebral, isquemia cerebral, déficit cerebral após cirurgia cardìaca (bypass) e enxerto, lupus eritematoso sistêmico, doença de hodgkin, doença de sjogren, epilepsia, e rejeição em transplantes de órgão e enxertos de pele, e para tratar dependência de substáncias, métodos para melhorar a sobrevivência de órgãos e células, e cardioproteção após infarto do miocárdio, métodos para reduzir a necessidade de anestesia, para produzir ou manter um estado anestésico, derivado radiomarcado de um composto, derivado isotopicamente marcado de um composto, composto e método de diagnóstico por imagem
US7598261B2 (en) 2005-03-31 2009-10-06 Adolor Corporation Spirocyclic heterocyclic derivatives and methods of their use
US7576207B2 (en) 2006-04-06 2009-08-18 Adolor Corporation Spirocyclic heterocyclic derivatives and methods of their use
AU2007294968A1 (en) 2006-09-12 2008-03-20 Adolor Corporation Use of N-containing spirocompounds for the enhancement of cognitive function

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2898339A (en) * 1957-07-29 1959-08-04 Wm S Merrell Co N-substituted benzhydrol, benzhydryl, and benzhydrylidene piperidine
US4581171A (en) * 1983-07-27 1986-04-08 Janssen Pharmaceutica, N.V. [[Bis(aryl)methylene]-1-piperidinyl]alkyl-pyrimidinones useful for treating psychotropic disorders
US4816586A (en) * 1987-07-29 1989-03-28 Regents Of The University Of Minnesota Delta opioid receptor antagonists
US5140029A (en) * 1989-01-09 1992-08-18 Janssen Pharmaceutica N.V. 2-aminopyrimidinone derivatives
US4939137A (en) * 1989-06-28 1990-07-03 Ortho Pharmaceutical Corporation Ring-fused thienopyrimidinedione derivatives
US5683998A (en) * 1991-04-23 1997-11-04 Toray Industries, Inc. Tricyclic triazolo derivatives, processes for producing the same and the uses of the same
US5574159A (en) * 1992-02-03 1996-11-12 Delta Pharmaceuticals, Inc. Opioid compounds and methods for making therefor
TW548271B (en) * 1996-12-20 2003-08-21 Astra Pharma Inc Novel piperidine derivatives having an exocyclic double bond with analgesic effects
US6436959B1 (en) * 1998-12-23 2002-08-20 Ortho-Mcneil Pharmaceutical, Inc. 4-[aryl(piperidin-4-yl)]aminobenzamides
SE0001207D0 (sv) * 2000-04-04 2000-04-04 Astrazeneca Canada Inc Novel compounds

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