JP2005504776A5 - - Google Patents
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- Publication number
- JP2005504776A5 JP2005504776A5 JP2003522545A JP2003522545A JP2005504776A5 JP 2005504776 A5 JP2005504776 A5 JP 2005504776A5 JP 2003522545 A JP2003522545 A JP 2003522545A JP 2003522545 A JP2003522545 A JP 2003522545A JP 2005504776 A5 JP2005504776 A5 JP 2005504776A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- pharmaceutical composition
- composition according
- alkanoyl
- alkenyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
- 239000008194 pharmaceutical composition Substances 0.000 claims 7
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 claims 4
- 150000001875 compounds Chemical class 0.000 claims 4
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 4
- 241000725303 Human immunodeficiency virus Species 0.000 claims 2
- 241000124008 Mammalia Species 0.000 claims 2
- 208000004296 neuralgia Diseases 0.000 claims 2
- 208000021722 neuropathic pain Diseases 0.000 claims 2
- 150000003839 salts Chemical class 0.000 claims 2
- 208000030507 AIDS Diseases 0.000 claims 1
- 208000023890 Complex Regional Pain Syndromes Diseases 0.000 claims 1
- 208000032131 Diabetic Neuropathies Diseases 0.000 claims 1
- 208000002193 Pain Diseases 0.000 claims 1
- 208000004983 Phantom Limb Diseases 0.000 claims 1
- 206010056238 Phantom pain Diseases 0.000 claims 1
- 206010036376 Postherpetic Neuralgia Diseases 0.000 claims 1
- QRJOQYLXZPQQMX-FWROMSNXSA-N acetic acid [2-[(3R,5S,8S,9S,10S,13S,14S,17S)-3-hydroxy-10,13-dimethyl-11-oxo-1,2,3,4,5,6,7,8,9,12,14,15,16,17-tetradecahydrocyclopenta[a]phenanthren-17-yl]-2-oxoethyl] ester Chemical compound C([C@@H]1CC2)[C@H](O)CC[C@]1(C)[C@@H]1[C@@H]2[C@@H]2CC[C@H](C(=O)COC(=O)C)[C@@]2(C)CC1=O QRJOQYLXZPQQMX-FWROMSNXSA-N 0.000 claims 1
- 239000000654 additive Substances 0.000 claims 1
- 230000000996 additive effect Effects 0.000 claims 1
- 229910052794 bromium Inorganic materials 0.000 claims 1
- 229910052801 chlorine Inorganic materials 0.000 claims 1
- 239000003814 drug Substances 0.000 claims 1
- 229940079593 drug Drugs 0.000 claims 1
- 229910052731 fluorine Inorganic materials 0.000 claims 1
- 229910052736 halogen Inorganic materials 0.000 claims 1
- 150000002367 halogens Chemical class 0.000 claims 1
- 208000015181 infectious disease Diseases 0.000 claims 1
- 239000002207 metabolite Substances 0.000 claims 1
- 201000001119 neuropathy Diseases 0.000 claims 1
- 230000007823 neuropathy Effects 0.000 claims 1
- 208000033808 peripheral neuropathy Diseases 0.000 claims 1
- 206010044652 trigeminal neuralgia Diseases 0.000 claims 1
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AUPR7319A AUPR731901A0 (en) | 2001-08-28 | 2001-08-28 | Method of treatment |
| PCT/AU2002/001144 WO2003018027A1 (en) | 2001-08-28 | 2002-08-28 | Use of pregnane-diones or diols as neuropathic analgesic agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2005504776A JP2005504776A (ja) | 2005-02-17 |
| JP2005504776A5 true JP2005504776A5 (enExample) | 2006-01-05 |
Family
ID=3831271
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2003522545A Pending JP2005504776A (ja) | 2001-08-28 | 2002-08-28 | 神経因性鎮痛薬としてのプレグナン−ジオンまたはジオールの使用 |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US20050009796A1 (enExample) |
| EP (1) | EP1450817A4 (enExample) |
| JP (1) | JP2005504776A (enExample) |
| CN (2) | CN101590062A (enExample) |
| AU (2) | AUPR731901A0 (enExample) |
| BR (1) | BR0212205A (enExample) |
| CA (1) | CA2468466A1 (enExample) |
| MX (1) | MXPA04001807A (enExample) |
| RU (1) | RU2346690C2 (enExample) |
| WO (1) | WO2003018027A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10141650C1 (de) * | 2001-08-24 | 2002-11-28 | Lohmann Therapie Syst Lts | Transdermales Therapeutisches System mit Fentanyl bzw. verwandten Substanzen |
| GB0324423D0 (en) * | 2003-10-18 | 2003-11-19 | Vernalis Cambridge Ltd | Analgesia method |
| WO2006010085A1 (en) * | 2004-07-09 | 2006-01-26 | Roxro Pharma, Inc. | Use of neurosteroids to treat neuropathic pain |
| RU2306930C1 (ru) * | 2005-12-28 | 2007-09-27 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией лозартана и l-аргинина при l-name-индуцированном дефиците оксида азота |
| RU2306924C1 (ru) * | 2005-12-28 | 2007-09-27 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией лозартана и резвератрола при l-name-индуцированном дефиците оксида азота |
| RU2302241C1 (ru) * | 2005-12-28 | 2007-07-10 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией индапамида и резвератрола при l-name-индуцированном дефиците оксида азота |
| RU2296566C1 (ru) * | 2005-12-28 | 2007-04-10 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией амлодипина и l-аргинина при l-name-индуцированном дефиците оксида азота |
| RU2306929C1 (ru) * | 2005-12-28 | 2007-09-27 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией индапамида и l-аргинина при l-name-индуцированном дефиците оксида азота |
| KR20090125748A (ko) * | 2007-04-02 | 2009-12-07 | 토요 보세키 가부시기가이샤 | 대상포진 후 신경통 치료용 정제 및 대상포진 후 신경통의 치료 방법 |
| RU2364393C1 (ru) * | 2008-03-19 | 2009-08-20 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции пикамилоном при l-name индуцированном дефиците оксида азота |
| US8815300B2 (en) | 2008-08-29 | 2014-08-26 | Coastal Biologic Solutions | Composition and methods for relief of neuropathological pain |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1317184A (en) * | 1969-06-20 | 1973-05-16 | Glaxo Lab Ltd | Steroid-containing pharmaceutical preparations |
| GB1373913A (en) * | 1970-12-17 | 1974-11-13 | Glaxo Lab Ltd | Pharmaceutical compositions |
| US5888996A (en) * | 1995-07-26 | 1999-03-30 | Trustees Of Boston University | Inhibition of NMDA receptor activity and modulation of glutamate-mediated synaptic activity |
| EP0840612A1 (en) * | 1995-07-24 | 1998-05-13 | Trustees Of Boston University | Inhibition of nmda receptor activity by pregnenolone sulfate derivatives |
| AUPN498095A0 (en) * | 1995-08-23 | 1995-09-14 | Goodchild, Colin Stanley | Compounds and compositions |
| GB9607034D0 (en) * | 1996-04-03 | 1996-06-05 | Leo Pharm Prod Ltd | Chemical compounds |
| US6048848A (en) * | 1996-08-23 | 2000-04-11 | Monash University | Use of pregnane-diones as analgesic agents |
| US6787530B1 (en) * | 1996-08-23 | 2004-09-07 | Monash University | Use of pregnane-diones as analgesic agents |
| ATE425459T1 (de) * | 1999-08-31 | 2009-03-15 | Univ Boston | Der effekt von steroiden auf ndma-rezeptoren beruht auf der zusammensetzung der untereinheiten |
| US20030027833A1 (en) * | 2001-05-07 | 2003-02-06 | Cleary Gary W. | Compositions and delivery systems for administration of a local anesthetic agent |
-
2001
- 2001-08-28 AU AUPR7319A patent/AUPR731901A0/en not_active Abandoned
-
2002
- 2002-08-28 JP JP2003522545A patent/JP2005504776A/ja active Pending
- 2002-08-28 MX MXPA04001807A patent/MXPA04001807A/es not_active Application Discontinuation
- 2002-08-28 BR BR0212205-7A patent/BR0212205A/pt not_active IP Right Cessation
- 2002-08-28 CN CNA2009101264152A patent/CN101590062A/zh active Pending
- 2002-08-28 WO PCT/AU2002/001144 patent/WO2003018027A1/en not_active Ceased
- 2002-08-28 EP EP02759883A patent/EP1450817A4/en not_active Withdrawn
- 2002-08-28 CA CA002468466A patent/CA2468466A1/en not_active Abandoned
- 2002-08-28 CN CNA02817027XA patent/CN1549719A/zh active Pending
- 2002-08-28 RU RU2004109517/14A patent/RU2346690C2/ru not_active IP Right Cessation
- 2002-08-28 US US10/487,922 patent/US20050009796A1/en not_active Abandoned
-
2008
- 2008-03-03 US US12/041,593 patent/US20080227764A1/en not_active Abandoned
- 2008-06-20 AU AU2008202729A patent/AU2008202729A1/en not_active Abandoned
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