MXPA04001807A - Uso de pregnano dionas o dioles como agentes analgesicos neuropaticos. - Google Patents
Uso de pregnano dionas o dioles como agentes analgesicos neuropaticos.Info
- Publication number
- MXPA04001807A MXPA04001807A MXPA04001807A MXPA04001807A MXPA04001807A MX PA04001807 A MXPA04001807 A MX PA04001807A MX PA04001807 A MXPA04001807 A MX PA04001807A MX PA04001807 A MXPA04001807 A MX PA04001807A MX PA04001807 A MXPA04001807 A MX PA04001807A
- Authority
- MX
- Mexico
- Prior art keywords
- alkyl
- alkanoyl
- alkenyl
- compound
- formula
- Prior art date
Links
- 150000002009 diols Chemical class 0.000 title claims description 4
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- 239000000730 antalgic agent Substances 0.000 title description 5
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- RMRJXGBAOAMLHD-IHFGGWKQSA-N buprenorphine Chemical compound C([C@]12[C@H]3OC=4C(O)=CC=C(C2=4)C[C@@H]2[C@]11CC[C@]3([C@H](C1)[C@](C)(O)C(C)(C)C)OC)CN2CC1CC1 RMRJXGBAOAMLHD-IHFGGWKQSA-N 0.000 claims description 3
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- 230000000007 visual effect Effects 0.000 description 1
- 230000001755 vocal effect Effects 0.000 description 1
- 239000007762 w/o emulsion Substances 0.000 description 1
- 239000008215 water for injection Substances 0.000 description 1
- 239000001993 wax Substances 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AUPR7319A AUPR731901A0 (en) | 2001-08-28 | 2001-08-28 | Method of treatment |
| PCT/AU2002/001144 WO2003018027A1 (en) | 2001-08-28 | 2002-08-28 | Use of pregnane-diones or diols as neuropathic analgesic agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MXPA04001807A true MXPA04001807A (es) | 2005-03-07 |
Family
ID=3831271
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MXPA04001807A MXPA04001807A (es) | 2001-08-28 | 2002-08-28 | Uso de pregnano dionas o dioles como agentes analgesicos neuropaticos. |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US20050009796A1 (enExample) |
| EP (1) | EP1450817A4 (enExample) |
| JP (1) | JP2005504776A (enExample) |
| CN (2) | CN1549719A (enExample) |
| AU (2) | AUPR731901A0 (enExample) |
| BR (1) | BR0212205A (enExample) |
| CA (1) | CA2468466A1 (enExample) |
| MX (1) | MXPA04001807A (enExample) |
| RU (1) | RU2346690C2 (enExample) |
| WO (1) | WO2003018027A1 (enExample) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10141650C1 (de) | 2001-08-24 | 2002-11-28 | Lohmann Therapie Syst Lts | Transdermales Therapeutisches System mit Fentanyl bzw. verwandten Substanzen |
| GB0324423D0 (en) * | 2003-10-18 | 2003-11-19 | Vernalis Cambridge Ltd | Analgesia method |
| US20060009432A1 (en) * | 2004-07-09 | 2006-01-12 | Roger Whiting | Use of neurosteroids to treat neuropathic pain |
| RU2306929C1 (ru) * | 2005-12-28 | 2007-09-27 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией индапамида и l-аргинина при l-name-индуцированном дефиците оксида азота |
| RU2306924C1 (ru) * | 2005-12-28 | 2007-09-27 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией лозартана и резвератрола при l-name-индуцированном дефиците оксида азота |
| RU2296566C1 (ru) * | 2005-12-28 | 2007-04-10 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией амлодипина и l-аргинина при l-name-индуцированном дефиците оксида азота |
| RU2306930C1 (ru) * | 2005-12-28 | 2007-09-27 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией лозартана и l-аргинина при l-name-индуцированном дефиците оксида азота |
| RU2302241C1 (ru) * | 2005-12-28 | 2007-07-10 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции комбинацией индапамида и резвератрола при l-name-индуцированном дефиците оксида азота |
| JPWO2008120562A1 (ja) * | 2007-04-02 | 2010-07-15 | 東洋紡績株式会社 | 帯状疱疹後神経痛治療用錠剤および帯状疱疹後神経痛の治療方法 |
| RU2364393C1 (ru) * | 2008-03-19 | 2009-08-20 | Михаил Владимирович Покровский | Способ коррекции эндотелиальной дисфункции пикамилоном при l-name индуцированном дефиците оксида азота |
| WO2010025316A1 (en) * | 2008-08-29 | 2010-03-04 | Jeffrey Comanor | Composition and methods for relief of neuropathological pain |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1317184A (en) * | 1969-06-20 | 1973-05-16 | Glaxo Lab Ltd | Steroid-containing pharmaceutical preparations |
| GB1373913A (en) * | 1970-12-17 | 1974-11-13 | Glaxo Lab Ltd | Pharmaceutical compositions |
| US5888996A (en) * | 1995-07-26 | 1999-03-30 | Trustees Of Boston University | Inhibition of NMDA receptor activity and modulation of glutamate-mediated synaptic activity |
| JP4313435B2 (ja) * | 1995-07-24 | 2009-08-12 | トラスティーズ オブ ボストン ユニバーシティー | プレグネノロンサルフェート誘導体によるｎｍｄａレセプター活性の抑制 |
| AUPN498095A0 (en) * | 1995-08-23 | 1995-09-14 | Goodchild, Colin Stanley | Compounds and compositions |
| GB9607034D0 (en) * | 1996-04-03 | 1996-06-05 | Leo Pharm Prod Ltd | Chemical compounds |
| US6048848A (en) * | 1996-08-23 | 2000-04-11 | Monash University | Use of pregnane-diones as analgesic agents |
| US6787530B1 (en) * | 1996-08-23 | 2004-09-07 | Monash University | Use of pregnane-diones as analgesic agents |
| AU782250B2 (en) * | 1999-08-31 | 2005-07-14 | Trustees Of Boston University | Effect of steroids on NMDA receptors depends on subunit composition |
| US20030027833A1 (en) * | 2001-05-07 | 2003-02-06 | Cleary Gary W. | Compositions and delivery systems for administration of a local anesthetic agent |
-
2001
- 2001-08-28 AU AUPR7319A patent/AUPR731901A0/en not_active Abandoned
-
2002
- 2002-08-28 RU RU2004109517/14A patent/RU2346690C2/ru not_active IP Right Cessation
- 2002-08-28 CN CNA02817027XA patent/CN1549719A/zh active Pending
- 2002-08-28 US US10/487,922 patent/US20050009796A1/en not_active Abandoned
- 2002-08-28 EP EP02759883A patent/EP1450817A4/en not_active Withdrawn
- 2002-08-28 BR BR0212205-7A patent/BR0212205A/pt not_active IP Right Cessation
- 2002-08-28 CN CNA2009101264152A patent/CN101590062A/zh active Pending
- 2002-08-28 JP JP2003522545A patent/JP2005504776A/ja active Pending
- 2002-08-28 MX MXPA04001807A patent/MXPA04001807A/es not_active Application Discontinuation
- 2002-08-28 CA CA002468466A patent/CA2468466A1/en not_active Abandoned
- 2002-08-28 WO PCT/AU2002/001144 patent/WO2003018027A1/en not_active Ceased
-
2008
- 2008-03-03 US US12/041,593 patent/US20080227764A1/en not_active Abandoned
- 2008-06-20 AU AU2008202729A patent/AU2008202729A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CN1549719A (zh) | 2004-11-24 |
| RU2004109517A (ru) | 2005-06-27 |
| US20050009796A1 (en) | 2005-01-13 |
| CA2468466A1 (en) | 2003-03-06 |
| EP1450817A1 (en) | 2004-09-01 |
| US20080227764A1 (en) | 2008-09-18 |
| BR0212205A (pt) | 2004-09-21 |
| AUPR731901A0 (en) | 2001-09-20 |
| WO2003018027A1 (en) | 2003-03-06 |
| AU2008202729A1 (en) | 2008-07-17 |
| RU2346690C2 (ru) | 2009-02-20 |
| CN101590062A (zh) | 2009-12-02 |
| EP1450817A4 (en) | 2009-02-25 |
| JP2005504776A (ja) | 2005-02-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |