JP2005503416A - ６−ｏ−カルバメート−１１，１２−ラクト−ケトライド抗菌剤 - Google Patents

６−ｏ−カルバメート−１１，１２−ラクト−ケトライド抗菌剤 Download PDF

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Publication number
JP2005503416A
JP2005503416A JP2003528832A JP2003528832A JP2005503416A JP 2005503416 A JP2005503416 A JP 2005503416A JP 2003528832 A JP2003528832 A JP 2003528832A JP 2003528832 A JP2003528832 A JP 2003528832A JP 2005503416 A JP2005503416 A JP 2005503416A
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substituted
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JP2003528832A
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Japanese (ja)
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JP2005503416A5 (enExample
Inventor
グラント，ユージーン・ビー，ザサード
ヘニンガー，トツド・シー
ミシーラグ，マーク・ジエイ
ガイアデイーン，デオデイアルシング
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オーソ−マクニール・フアーマシユーチカル・インコーポレーテツド
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Publication of JP2005503416A publication Critical patent/JP2005503416A/ja
Publication of JP2005503416A5 publication Critical patent/JP2005503416A5/ja
Pending legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
JP2003528832A 2001-09-17 2002-09-16 ６−ｏ−カルバメート−１１，１２−ラクト−ケトライド抗菌剤 Pending JP2005503416A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32276201P 2001-09-17 2001-09-17
PCT/US2002/029314 WO2003024986A1 (en) 2001-09-17 2002-09-16 6-o-carbamate-11,12-lacto-ketolide antimicrobials

Publications (2)

Publication Number Publication Date
JP2005503416A true JP2005503416A (ja) 2005-02-03
JP2005503416A5 JP2005503416A5 (enExample) 2006-01-05

Family

ID=23256294

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003528832A Pending JP2005503416A (ja) 2001-09-17 2002-09-16 ６−ｏ−カルバメート−１１，１２−ラクト−ケトライド抗菌剤

Country Status (6)

Country Link
US (1) US6713455B2 (enExample)
EP (1) EP1430068A1 (enExample)
JP (1) JP2005503416A (enExample)
CN (1) CN1589277A (enExample)
CA (1) CA2460947A1 (enExample)
WO (1) WO2003024986A1 (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005526050A (ja) * 2002-02-28 2005-09-02 バジリア　ファルマスーチカ　アーゲー 抗菌活性を有するマクロライド
JP2010500329A (ja) * 2006-08-09 2010-01-07 バジリア ファルマスーチカ アーゲー 炎症性及びアレルギー性疾患に対して有用な新規マクロライド

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2002217277B2 (en) * 2000-12-21 2005-06-16 Glaxo Group Limited Macrolide antibiotics
US6727229B2 (en) 2002-08-19 2004-04-27 Enanta Pharmaceuticals, Inc. 11,12-substituted lactone ketolide derivatives having antibacterial activity
US6720308B1 (en) 2002-11-07 2004-04-13 Enanta Pharmaceuticals, Inc. Anhydrolide derivatives having antibacterial activity
US6790835B1 (en) 2003-06-05 2004-09-14 Enanta Pharmaceuticals, Inc. Bicyclic macrolide derivatives
US6716820B1 (en) 2003-06-05 2004-04-06 Enanta Pharmaceuticals, Inc. 6-O-substituted bicyclic macrolides
US6765016B1 (en) 2003-06-05 2004-07-20 Enanta Pharmaceuticals, Inc. Bicyclic ketolide derivatives
US6774115B1 (en) 2003-06-05 2004-08-10 Enanta Pharmaceuticals, Inc. 6-O-substituted bicyclic ketolides
WO2008014221A2 (en) * 2006-07-24 2008-01-31 Enanta Pharmaceuticals, Inc. Bridged carbamate macrolides
KR101617897B1 (ko) 2008-02-08 2016-05-03 바실리어 파마슈티카 아게 신규 마크로라이드 및 그의 용도
MY177250A (en) 2010-06-30 2020-09-10 Fujifilm Corp Novel nicotinamide derivative or salt thereof
EP2630133A1 (de) 2010-10-22 2013-08-28 Bayer Intellectual Property GmbH Neue heterocylische verbindungen als schädlingsbekämpfungsmittel

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8521402D0 (en) 1985-08-28 1985-10-02 Beecham Group Plc Chemical compounds
IL114589A (en) 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
US5559256A (en) 1992-07-20 1996-09-24 E. R. Squibb & Sons, Inc. Aminediol protease inhibitors
BR9507220A (pt) 1994-03-28 1997-09-09 Japat Ltd Antagonistas de receptores de endotelina
DE69631609T2 (de) 1995-11-08 2005-01-05 Abbott Laboratories, Abbott Park Tricyclische erythromycinderivate
CA2249650A1 (en) 1996-04-03 1997-10-09 Merck & Co., Inc. Inhibitors of farnesyl-protein transferase
ES2242983T3 (es) 1996-09-04 2005-11-16 Abbott Laboratories Cetolidos 6-0-sustituidos que tienen una actividad antibacteriana.
UA51730C2 (uk) 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
UA56197C2 (uk) 1996-11-08 2003-05-15 Зенека Лімітед Гетероциклічні похідні
UA59384C2 (uk) 1996-12-20 2003-09-15 Пфайзер, Інк. Похідні сульфонамідів та амідів як агоністи простагландину, фармацевтична композиція та способи лікування на їх основі
AU7937998A (en) 1997-07-08 1999-02-08 Sankyo Company Limited Antifungal triazole compounds
CO4990960A1 (es) 1997-10-29 2000-12-26 Abbott Lab Derivados de cetolidos 2-halo-6-o sustituidos
AR015986A1 (es) 1997-10-29 2001-05-30 Abbott Lab Derivados de eritromicina puenteados en 6,11, composiciones farmaceuticas que los contienen, su uso para la manufactura de un medicamento y procedimientospara su preparacion
AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
AU775637B2 (en) 1999-04-16 2004-08-12 Kosan Biosciences, Inc. Macrolide antiinfective agents
CA2370743A1 (en) 1999-04-16 2000-10-26 Dennis Hlasta Ketolide antibacterials
WO2000075156A1 (en) * 1999-06-07 2000-12-14 Abbott Laboratories 6-o-carbamate ketolide derivatives
EP1114826A3 (en) 1999-12-29 2001-10-31 Pfizer Products Inc. Novel antibacterial and prokinetic macrolides
EP1313751B1 (en) 2000-08-22 2008-09-17 Basilea Pharmaceutica AG New macrolides with antibacterial activity
GB0031312D0 (en) 2000-12-21 2001-02-07 Glaxo Group Ltd Macrolides

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005526050A (ja) * 2002-02-28 2005-09-02 バジリア　ファルマスーチカ　アーゲー 抗菌活性を有するマクロライド
JP2010500329A (ja) * 2006-08-09 2010-01-07 バジリア ファルマスーチカ アーゲー 炎症性及びアレルギー性疾患に対して有用な新規マクロライド

Also Published As

Publication number Publication date
CA2460947A1 (en) 2003-03-27
EP1430068A1 (en) 2004-06-23
WO2003024986A1 (en) 2003-03-27
CN1589277A (zh) 2005-03-02
US20030125267A1 (en) 2003-07-03
US6713455B2 (en) 2004-03-30

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