JP2004530705A5 - - Google Patents

Download PDF

Info

Publication number
JP2004530705A5
JP2004530705A5 JP2002592933A JP2002592933A JP2004530705A5 JP 2004530705 A5 JP2004530705 A5 JP 2004530705A5 JP 2002592933 A JP2002592933 A JP 2002592933A JP 2002592933 A JP2002592933 A JP 2002592933A JP 2004530705 A5 JP2004530705 A5 JP 2004530705A5
Authority
JP
Japan
Prior art keywords
triazolo
pyrazolo
dihydro
pyridine
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2002592933A
Other languages
English (en)
Japanese (ja)
Other versions
JP2004530705A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2002/005643 external-priority patent/WO2002096423A2/en
Publication of JP2004530705A publication Critical patent/JP2004530705A/ja
Publication of JP2004530705A5 publication Critical patent/JP2004530705A5/ja
Pending legal-status Critical Current

Links

JP2002592933A 2001-05-25 2002-05-23 閉塞性気道疾患及びその他の炎症性疾患を治療するためのpde4インヒビター及びチオトロピウム又はその誘導体の組み合わせ Pending JP2004530705A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29355501P 2001-05-25 2001-05-25
US30384501P 2001-07-09 2001-07-09
PCT/EP2002/005643 WO2002096423A2 (en) 2001-05-25 2002-05-23 Combination of a pde4 inhibitor and tiotropium or derivate thereof for treating obstructive airways

Publications (2)

Publication Number Publication Date
JP2004530705A JP2004530705A (ja) 2004-10-07
JP2004530705A5 true JP2004530705A5 (enExample) 2006-01-05

Family

ID=26968011

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2002592933A Pending JP2004530705A (ja) 2001-05-25 2002-05-23 閉塞性気道疾患及びその他の炎症性疾患を治療するためのpde4インヒビター及びチオトロピウム又はその誘導体の組み合わせ

Country Status (9)

Country Link
EP (1) EP1397135B1 (enExample)
JP (1) JP2004530705A (enExample)
AT (1) ATE347361T1 (enExample)
AU (1) AU2002314102A1 (enExample)
CA (1) CA2448363A1 (enExample)
DE (1) DE60216588T2 (enExample)
ES (1) ES2276942T3 (enExample)
MX (1) MXPA03010791A (enExample)
WO (1) WO2002096423A2 (enExample)

Families Citing this family (33)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2165768B1 (es) 1999-07-14 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de quinuclidina y composiciones farmaceuticas que los contienen.
MY140561A (en) 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
DK1610787T3 (da) * 2003-03-28 2008-06-02 Nycomed Gmbh Synergistisk kombination der omfatter roflumilast og et antikolinergt middel der er valgt blandt tiotropiumsalte til behandling af respiratoriske sygdomme
CA2522666A1 (en) * 2003-04-18 2004-10-28 Pharmacia & Upjohn Company Llc Combination therapies for chronic obstructive pulmonary disease (copd)
UA83041C2 (ru) * 2003-05-22 2008-06-10 Нікомед Гмбх Композиция, которая включает ингибитор pde4 и ингибитор pde5
WO2005013993A1 (en) * 2003-07-29 2005-02-17 Boehringer Ingelheim International Gmbh Medicaments comprising pde iv inhibitors and an anticholinergic for treating respiratory disorders
EP1504756A1 (en) * 2003-08-06 2005-02-09 Kyowa Hakko Kogyo Co., Ltd Medicament compositions comprising a heterocyclic compound and an anticholinergic
ES2381116T3 (es) * 2004-02-06 2012-05-23 Meda Pharma Gmbh & Co. Kg Combinación de anticolinérgicos e inhibidores de fosfodiesterasa tipo 4 para el tratamiento de enfermedades respiratorias
WO2005074983A2 (en) * 2004-02-06 2005-08-18 Meda Pharma Gmbh & Co. Kg Treatment of rhinitis with anticholinergics alone in combination with antihistamines phosphodiesterase 4 inhibitors, or corticosteroids
ES2413011T3 (es) 2004-02-06 2013-07-15 Meda Pharma Gmbh & Co. Kg Combinación de anticolinérgicos y glucocorticoides para el tratamiento a largo plazo de asma y EPOC
CA2553369A1 (en) * 2004-02-20 2005-09-01 Boehringer Ingelheim International Gmbh Pharmaceutical compositions based on anticholinergics and pegsunercept
US7507745B2 (en) 2004-02-20 2009-03-24 Boehringer Ingelheim International Gmbh Pharmaceutical compositions based on fluorenecarboxylic acid esters and soluble TNF receptor fusion proteins
ES2257152B1 (es) * 2004-05-31 2007-07-01 Laboratorios Almirall S.A. Combinaciones que comprenden agentes antimuscarinicos y agonistas beta-adrenergicos.
AU2005247104B2 (en) * 2004-05-31 2010-11-11 Laboratorios Almirall, S.A. Combinations comprising antimuscarinic agents and beta-adrenergic agonists
US20060079544A1 (en) * 2004-08-13 2006-04-13 Boehringer Ingelheim International Gmbh Medicaments for the prevention or treatment of alveolar pneumonia comprising an anticholinergic
RU2420285C2 (ru) 2005-03-16 2011-06-10 Меда Фарма Гмбх Унд Ко.Кг Комбинация r,r-гликопирролата и монтелукаста для лечения респираторных заболеваний и фармацевтическая композиция на ее основе
US8012971B2 (en) * 2005-04-28 2011-09-06 Dainippon Sumitomo Pharma Co., Ltd. Therapeutic agent for chronic obstructive pulmonary disease
DE102005035112A1 (de) * 2005-07-27 2007-02-15 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neues Verfahren zur Herstellung von Tiotropiumsalzen unter Anwendung von in organischen Lösungsmitteln löslichen N-Methylscopiniumsalzen
EP2258359A3 (en) 2005-08-26 2011-04-06 Braincells, Inc. Neurogenesis by muscarinic receptor modulation with sabcomelin
JP2009506069A (ja) 2005-08-26 2009-02-12 ブレインセルス,インコーポレイティド ムスカリン性受容体調節による神経発生
EP1940389A2 (en) 2005-10-21 2008-07-09 Braincells, Inc. Modulation of neurogenesis by pde inhibition
AU2006308889A1 (en) 2005-10-31 2007-05-10 Braincells, Inc. GABA receptor mediated modulation of neurogenesis
DK2098248T3 (da) 2005-12-21 2012-09-17 Meda Pharma Gmbh & Co Kg Kombination af anticholinergika, glucocorticoider og beta2-agonister til behandling af inflammatoriske sygdomme
US20100216734A1 (en) 2006-03-08 2010-08-26 Braincells, Inc. Modulation of neurogenesis by nootropic agents
WO2007134136A2 (en) 2006-05-09 2007-11-22 Braincells, Inc. Neurogenesis by modulating angiotensin
EP1905440A1 (de) * 2006-09-06 2008-04-02 Boehringer Ingelheim Pharma GmbH & Co. KG Verwendung einer pharmazeutischen Zusammensetzung enthaltend ein Anticholinergikum zur Abtötung von Mikroorganismen und zur Behandlung von Atemwegsinfektionen
US20100184806A1 (en) 2006-09-19 2010-07-22 Braincells, Inc. Modulation of neurogenesis by ppar agents
EP2100598A1 (en) 2008-03-13 2009-09-16 Laboratorios Almirall, S.A. Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease
EP2100599A1 (en) 2008-03-13 2009-09-16 Laboratorios Almirall, S.A. Inhalation composition containing aclidinium for treatment of asthma and chronic obstructive pulmonary disease
US20100216805A1 (en) 2009-02-25 2010-08-26 Braincells, Inc. Modulation of neurogenesis using d-cycloserine combinations
EP3090999A1 (en) * 2009-06-18 2016-11-09 Concert Pharmaceuticals Inc. Deuterated isoindoline-1, 3-dione derivatives as pde4 and tnf-alpha inhibitors
EP2510928A1 (en) 2011-04-15 2012-10-17 Almirall, S.A. Aclidinium for use in improving the quality of sleep in respiratory patients
WO2013106547A1 (en) 2012-01-10 2013-07-18 President And Fellows Of Harvard College Beta-cell replication promoting compounds and methods of their use

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2223624C (en) * 1995-06-06 2001-02-20 Pfizer Inc. Tricyclic 5,6-dihydro-9h-pyrazolo[3,4-c]-1,2,4-triazolo[4,3-.alpha.]pyridines
DE10110772A1 (de) * 2001-03-07 2002-09-12 Boehringer Ingelheim Pharma Neue Arzneimittelkompositionen auf der Basis von Anticholinergika und PDE-IV-Inhibitoren

Similar Documents

Publication Publication Date Title
JP2004530705A5 (enExample)
CN103402515B (zh) sGC刺激剂
JP5841531B2 (ja) フラビウイルス科ウイルスの阻害剤
JP2012515787A5 (enExample)
RU2001132632A (ru) Производные пиперазина, применимые в качестве антагонистов CCR5
JP2014526501A5 (enExample)
ES2651162T3 (es) Antagonistas fluorados de integrina
WO2002094273A3 (en) Combination of an adenosine a2a-receptor agonist and tiotropium or a derivative thereof for treating obstructive airways
JP2009507896A5 (enExample)
JP2007519649A5 (enExample)
JP2013517286A (ja) フラビウイルス科ウイルスのインヒビター
JP2013504576A (ja) Flaviviridaeウイルスの阻害剤
JP2006517939A5 (enExample)
JP2006515339A5 (enExample)
TWI778052B (zh) 流感病毒複製之抑制劑
JP2007522162A5 (enExample)
RU2015121037A (ru) Производные фенилэтилпиридина в качестве ингибиторов pde-4
JP2009501775A5 (enExample)
RU2012146874A (ru) Производные пиразолопиридина
CA2457717A1 (en) Use of compounds in a dry powder inhaler
RU2007101238A (ru) Пептидные агонисты вазопрессинового рецептора
JP2003513075A5 (enExample)
RU2008124836A (ru) Органические соединения, включающие соль гликопиррония
RU2016121852A (ru) Производные бензгидрила для лечения респираторных заболеваний
JP2003516994A5 (enExample)