JP2003522192A5 - - Google Patents

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Publication number
JP2003522192A5
JP2003522192A5 JP2001558056A JP2001558056A JP2003522192A5 JP 2003522192 A5 JP2003522192 A5 JP 2003522192A5 JP 2001558056 A JP2001558056 A JP 2001558056A JP 2001558056 A JP2001558056 A JP 2001558056A JP 2003522192 A5 JP2003522192 A5 JP 2003522192A5
Authority
JP
Japan
Prior art keywords
amino
formula
methyl
pyrimidin
thiazolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2001558056A
Other languages
English (en)
Japanese (ja)
Other versions
JP2003522192A (ja
Filing date
Publication date
Priority claimed from GB0003025A external-priority patent/GB2359081A/en
Application filed filed Critical
Publication of JP2003522192A publication Critical patent/JP2003522192A/ja
Publication of JP2003522192A5 publication Critical patent/JP2003522192A5/ja
Pending legal-status Critical Current

Links

JP2001558056A 2000-02-11 2001-02-07 ケモカインレセプター活性のモジュレーターとしてのチアゾロピリミジンおよびそれらの使用 Pending JP2003522192A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0003025A GB2359081A (en) 2000-02-11 2000-02-11 Pharmaceutically active thiazolopyrimidines
GB0003025.4 2000-11-02
PCT/SE2001/000247 WO2001058907A1 (en) 2000-02-11 2001-02-07 Thiazolopyrimidines and their use as modulators of chemokine receptor activity

Publications (2)

Publication Number Publication Date
JP2003522192A JP2003522192A (ja) 2003-07-22
JP2003522192A5 true JP2003522192A5 (enExample) 2008-03-27

Family

ID=9885290

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001558056A Pending JP2003522192A (ja) 2000-02-11 2001-02-07 ケモカインレセプター活性のモジュレーターとしてのチアゾロピリミジンおよびそれらの使用

Country Status (8)

Country Link
US (1) US6958343B2 (enExample)
EP (1) EP1257556B1 (enExample)
JP (1) JP2003522192A (enExample)
AT (1) ATE269340T1 (enExample)
AU (1) AU2001234273A1 (enExample)
DE (1) DE60103856T2 (enExample)
GB (1) GB2359081A (enExample)
WO (1) WO2001058907A1 (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9903544D0 (sv) * 1999-10-01 1999-10-01 Astra Pharma Prod Novel compounds
GB2359078A (en) 2000-02-11 2001-08-15 Astrazeneca Uk Ltd Pharmaceutically active pyrimidine derivatives
WO2001058906A1 (en) * 2000-02-11 2001-08-16 Astrazeneca Ab Pyrimidine compounds and their use as modulators of chemokine receptor activity
GB2359551A (en) * 2000-02-23 2001-08-29 Astrazeneca Uk Ltd Pharmaceutically active pyrimidine derivatives
SE0003828D0 (sv) * 2000-10-20 2000-10-20 Astrazeneca Ab Novel compounds
SE0101082D0 (sv) 2001-03-27 2001-03-27 Astrazeneca Ab Novel use
SE0101322D0 (sv) * 2001-04-12 2001-04-12 Astrazeneca Ab Novel compounds
SE0102716D0 (sv) * 2001-08-14 2001-08-14 Astrazeneca Ab Novel compounds
ATE323702T1 (de) 2002-08-06 2006-05-15 Astrazeneca Ab Kondensierte pyridine und pyrimidine mit tie2 (tek) aktivität
GB0221828D0 (en) * 2002-09-20 2002-10-30 Astrazeneca Ab Novel compound
GB0221829D0 (en) * 2002-09-20 2002-10-30 Astrazeneca Ab Novel compound
GB0328243D0 (en) * 2003-12-05 2004-01-07 Astrazeneca Ab Methods
AR053347A1 (es) 2005-04-06 2007-05-02 Astrazeneca Ab Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
UA90707C2 (en) * 2005-04-06 2010-05-25 Астразенека Аб Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
TW200820973A (en) 2006-09-29 2008-05-16 Astrazeneca Ab Novel compounds 480
AU2007300749B2 (en) 2006-09-29 2011-08-25 Astrazeneca Ab Novel 5,7-disubstituted [1, 3] thiazolo [4, 5] pyrimidin-2 (3H)-amine derivatives and their use in therapy
US9040538B2 (en) * 2009-05-21 2015-05-26 Universite Laval Pyrimidines as novel therapeutic agents

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GB2359078A (en) 2000-02-11 2001-08-15 Astrazeneca Uk Ltd Pharmaceutically active pyrimidine derivatives
GB2359551A (en) 2000-02-23 2001-08-29 Astrazeneca Uk Ltd Pharmaceutically active pyrimidine derivatives
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