JP2003516394A5 - - Google Patents

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Publication number
JP2003516394A5
JP2003516394A5 JP2001543523A JP2001543523A JP2003516394A5 JP 2003516394 A5 JP2003516394 A5 JP 2003516394A5 JP 2001543523 A JP2001543523 A JP 2001543523A JP 2001543523 A JP2001543523 A JP 2001543523A JP 2003516394 A5 JP2003516394 A5 JP 2003516394A5
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JP
Japan
Prior art keywords
crystalline form
celecoxib
phase purity
crystalline
degrees
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2001543523A
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English (en)
Japanese (ja)
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JP2003516394A (ja
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Publication date
Application filed filed Critical
Priority claimed from PCT/US2000/032760 external-priority patent/WO2001042222A1/en
Publication of JP2003516394A publication Critical patent/JP2003516394A/ja
Publication of JP2003516394A5 publication Critical patent/JP2003516394A5/ja
Withdrawn legal-status Critical Current

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JP2001543523A 1999-12-08 2000-12-01 セレコキシブの多型結晶形態 Withdrawn JP2003516394A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16985699P 1999-12-08 1999-12-08
US60/169,856 1999-12-08
PCT/US2000/032760 WO2001042222A1 (en) 1999-12-08 2000-12-01 Polymorphic crystalline forms of celecoxib

Publications (2)

Publication Number Publication Date
JP2003516394A JP2003516394A (ja) 2003-05-13
JP2003516394A5 true JP2003516394A5 (enExample) 2008-01-24

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001543523A Withdrawn JP2003516394A (ja) 1999-12-08 2000-12-01 セレコキシブの多型結晶形態

Country Status (27)

Country Link
US (1) US7476744B2 (enExample)
EP (2) EP1528058A1 (enExample)
JP (1) JP2003516394A (enExample)
AT (1) ATE288897T1 (enExample)
AU (1) AU750978B2 (enExample)
BR (1) BR0008088A (enExample)
CA (1) CA2362675A1 (enExample)
CY (1) CY1106307T1 (enExample)
CZ (1) CZ20013210A3 (enExample)
DE (1) DE60018040T2 (enExample)
DK (1) DK1150960T3 (enExample)
DZ (1) DZ3140A1 (enExample)
EA (1) EA003464B1 (enExample)
EE (1) EE200100419A (enExample)
GE (1) GEP20043180B (enExample)
HR (1) HRP20010589A2 (enExample)
IL (1) IL144799A (enExample)
IS (1) IS6042A (enExample)
MX (1) MXPA01008161A (enExample)
NO (1) NO321062B1 (enExample)
NZ (1) NZ514059A (enExample)
PL (1) PL349224A1 (enExample)
SI (1) SI1150960T1 (enExample)
SK (1) SK11522001A3 (enExample)
UA (1) UA74539C2 (enExample)
WO (1) WO2001042222A1 (enExample)
ZA (1) ZA200207445B (enExample)

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CN102775396B (zh) 2005-11-08 2014-10-08 沃泰克斯药物股份有限公司 Atp-结合弹夹转运蛋白的杂环调控剂
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EP2231606B1 (en) 2007-12-07 2013-02-13 Vertex Pharmaceuticals Incorporated Processes for producing cycloalkylcarboxiamido-pyridine benzoic acids
ES2647531T3 (es) 2008-02-28 2017-12-22 Vertex Pharmaceuticals Incorporated Derivados de heteroarilo como moduladores de CFTR
CN102089051A (zh) * 2008-07-11 2011-06-08 巴斯夫欧洲公司 作为形态学改变剂的两亲性蛋白质
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US20110213159A1 (en) * 2010-03-01 2011-09-01 Vamsee Krishna Muppidi Process for preparation of celecoxib crystalline form
ES3017582T3 (en) 2010-04-07 2025-05-13 Vertex Pharma Pharmaceutical compositions of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxol-5-yl) cyclopropanecarboxamido)-3-methylpyriodin-2-yl)benzoic acid and administration thereof
EP2468258A1 (en) * 2010-12-22 2012-06-27 LEK Pharmaceuticals d.d. Process for the preparation of a pharmaceutical composition comprising a low soluble pharmaceutically active ingredient
CN103193677A (zh) * 2013-03-22 2013-07-10 南开大学 美索巴莫磷酸二钠盐的多晶型及其制备方法
CN103130684A (zh) * 2013-03-22 2013-06-05 南开大学 美索巴莫磷酸二钾盐的多晶型及其制备方法
CN105848657B (zh) 2013-11-12 2020-05-22 沃泰克斯药物股份有限公司 制备用于治疗cftr介导的疾病的药物组合物的方法
SI3221692T1 (sl) 2014-11-18 2021-11-30 Vertex Pharmaceuticals Inc. Postopek za izvajanje testov visoke prepustnosti z visoko zmogljivostno tekočinsko kromatografijo
KR20160098029A (ko) * 2015-01-13 2016-08-18 오토텔릭 엘엘씨 개별화된 약물 치료요법을 위한 방법
JP6499948B2 (ja) * 2015-09-09 2019-04-10 株式会社トクヤマ セレコキシブｉｉ型結晶の製造方法
TWI805601B (zh) 2017-08-11 2023-06-21 南韓商愛茉莉太平洋股份有限公司 醫藥組成物及抑制其形成結晶的方法
KR102518632B1 (ko) 2018-04-18 2023-04-06 (주)아모레퍼시픽 (r)-n-[1-(3,5-다이플루오로-4-메테인설폰일아미노-페닐)-에틸]-3-(2-프로필-6-트라이플루오로메틸-피리딘-3-일)-아크릴아마이드를 함유하는 약학 조성물
CN113005176A (zh) * 2019-12-20 2021-06-22 深圳市帝迈生物技术有限公司 稳定剂、凝血酶原时间检测试剂及其制备方法、试剂盒
CN119656108B (zh) * 2025-02-21 2025-05-30 墨格微流科技(汕头)有限公司 一种米诺地尔纳米晶混悬液及其制备方法

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