JP2003516393A5 - - Google Patents

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Publication number
JP2003516393A5
JP2003516393A5 JP2001543517A JP2001543517A JP2003516393A5 JP 2003516393 A5 JP2003516393 A5 JP 2003516393A5 JP 2001543517 A JP2001543517 A JP 2001543517A JP 2001543517 A JP2001543517 A JP 2001543517A JP 2003516393 A5 JP2003516393 A5 JP 2003516393A5
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JP
Japan
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oxo
compound
acid
substituted
embedded image
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JP2001543517A
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English (en)
Japanese (ja)
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JP5021131B2 (ja
JP2003516393A (ja
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Priority claimed from PCT/US2000/033260 external-priority patent/WO2001042216A2/en
Publication of JP2003516393A publication Critical patent/JP2003516393A/ja
Publication of JP2003516393A5 publication Critical patent/JP2003516393A5/ja
Application granted granted Critical
Publication of JP5021131B2 publication Critical patent/JP5021131B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP2001543517A 1999-12-08 2000-12-08 カスパーゼインヒビターおよびその使用 Expired - Fee Related JP5021131B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US16981299P 1999-12-08 1999-12-08
US60/169,812 1999-12-08
PCT/US2000/033260 WO2001042216A2 (en) 1999-12-08 2000-12-08 Caspase inhibitors and uses thereof

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP2007315252A Division JP2008101019A (ja) 1999-12-08 2007-12-05 カスパーゼインヒビターおよびその使用
JP2011234386A Division JP2012021032A (ja) 1999-12-08 2011-10-25 カスパーゼインヒビターおよびその使用

Publications (3)

Publication Number Publication Date
JP2003516393A JP2003516393A (ja) 2003-05-13
JP2003516393A5 true JP2003516393A5 (https=) 2008-01-31
JP5021131B2 JP5021131B2 (ja) 2012-09-05

Family

ID=22617272

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2001543517A Expired - Fee Related JP5021131B2 (ja) 1999-12-08 2000-12-08 カスパーゼインヒビターおよびその使用
JP2007315252A Withdrawn JP2008101019A (ja) 1999-12-08 2007-12-05 カスパーゼインヒビターおよびその使用
JP2011234386A Withdrawn JP2012021032A (ja) 1999-12-08 2011-10-25 カスパーゼインヒビターおよびその使用

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2007315252A Withdrawn JP2008101019A (ja) 1999-12-08 2007-12-05 カスパーゼインヒビターおよびその使用
JP2011234386A Withdrawn JP2012021032A (ja) 1999-12-08 2011-10-25 カスパーゼインヒビターおよびその使用

Country Status (24)

Country Link
US (4) US7517987B2 (https=)
EP (4) EP2308845A3 (https=)
JP (3) JP5021131B2 (https=)
KR (3) KR100904697B1 (https=)
CN (2) CN101348455A (https=)
AP (1) AP2002002535A0 (https=)
AR (1) AR026748A1 (https=)
AU (3) AU2428301A (https=)
BR (1) BR0016282A (https=)
CA (2) CA2733434A1 (https=)
CO (1) CO5261609A1 (https=)
CZ (1) CZ20021970A3 (https=)
EA (1) EA200200645A1 (https=)
HU (1) HUP0300782A3 (https=)
IL (1) IL150077A0 (https=)
IS (1) IS6411A (https=)
MX (1) MXPA02005779A (https=)
NO (2) NO324776B1 (https=)
NZ (2) NZ530485A (https=)
PL (1) PL356066A1 (https=)
SK (1) SK8072002A3 (https=)
TW (1) TWI275586B (https=)
WO (1) WO2001042216A2 (https=)
ZA (1) ZA200204390B (https=)

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US8173645B2 (en) 2007-03-21 2012-05-08 Takeda San Diego, Inc. Glucokinase activators
US8791235B2 (en) 2008-05-21 2014-07-29 Novagenesis Foundation Selective caspase inhibitors and uses thereof
WO2010017408A1 (en) 2008-08-06 2010-02-11 The Buck Institute For Age Research Caspase inhibitors and uses thereof
CA2738313A1 (en) 2008-09-23 2010-04-08 Georgetown University Viral and fungal inhibitors
EP2344479B1 (en) * 2008-09-23 2015-04-08 Georgetown University 1,2-benzisothiazolinone and isoindolinone derivatives
WO2010133000A1 (en) 2009-05-21 2010-11-25 New World Laboratories Inc. Selective caspase inhibitors and uses thereof
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WO2011094426A1 (en) 2010-01-29 2011-08-04 The United State Of America, As Represented By The Secretary, Department Of Health & Human Services Caspase inhibitors
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EP2699091B1 (en) 2011-03-28 2017-06-21 DeuteRx, LLC 2',6'-dioxo-3'-deutero-piperdin-3-yl-isoindoline compounds
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WO2018133870A1 (zh) * 2017-01-23 2018-07-26 正大天晴药业集团股份有限公司 作为Caspase抑制剂的联环化合物
CN106749045B (zh) * 2017-03-03 2020-02-14 上海交通大学 一种d-氨基酸氧化酶抑制剂及其制法和应用
EP3692014B1 (en) * 2017-10-04 2023-11-22 Battelle Memorial Institute Probe for selectively characterizing enzymes involved in xenobiotic metabolism and method of making and using the same
CA3171430A1 (en) * 2020-03-13 2021-09-16 Brent R. Stockwell Gpx4 compounds and compositions and methods of treatment using same
BR112022026725A2 (pt) * 2020-08-05 2023-02-14 Lg Chemical Ltd Composição farmacêutica para aliviar ou tratar osteoartrite
KR102670554B1 (ko) * 2022-01-04 2024-05-30 주식회사 이노보테라퓨틱스 캐스파제 저해제로서의 신규한 이소인돌리논 유도체 화합물
JP2025534288A (ja) * 2022-09-26 2025-10-15 エッジワイズ セラピューティクス, インコーポレイテッド 1,4-ジヒドロキナゾリノン化合物およびその使用
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