JP2003514876A - 新規官能化ポリマー試薬 - Google Patents

新規官能化ポリマー試薬

Info

Publication number
JP2003514876A
JP2003514876A JP2001539587A JP2001539587A JP2003514876A JP 2003514876 A JP2003514876 A JP 2003514876A JP 2001539587 A JP2001539587 A JP 2001539587A JP 2001539587 A JP2001539587 A JP 2001539587A JP 2003514876 A JP2003514876 A JP 2003514876A
Authority
JP
Japan
Prior art keywords
polymer
reagent
hydrogen
functionalized polymeric
functionalized
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2001539587A
Other languages
English (en)
Japanese (ja)
Inventor
パトリック・パージュ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
AstraZeneca AB
Original Assignee
AstraZeneca AB
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by AstraZeneca AB filed Critical AstraZeneca AB
Publication of JP2003514876A publication Critical patent/JP2003514876A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures
    • C40B40/04—Libraries containing only organic compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C291/00—Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00
    • C07C291/10—Isocyanides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78—Ring systems having three or more relevant rings
    • C07D311/80—Dibenzopyrans; Hydrogenated dibenzopyrans
    • C07D311/82—Xanthenes
    • C07D311/84—Xanthenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 9
    • C07D311/88—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
    • C08F8/00—Chemical modification by after-treatment
    • C08F8/30—Introducing nitrogen atoms or nitrogen-containing groups
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B20/00—Methods specially adapted for identifying library members
    • C40B20/04—Identifying library members by means of a tag, label, or other readable or detectable entity associated with the library members, e.g. decoding processes
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B30/00—Methods of screening libraries
    • C40B30/04—Methods of screening libraries by measuring the ability to specifically bind a target molecule, e.g. antibody-antigen binding, receptor-ligand binding
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B50/00—Methods of creating libraries, e.g. combinatorial synthesis
    • C40B50/14—Solid phase synthesis, i.e. wherein one or more library building blocks are bound to a solid support during library creation; Particular methods of cleavage from the solid support
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/11—Compounds covalently bound to a solid support

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Structural Engineering (AREA)
  • Engineering & Computer Science (AREA)
  • Polymers & Plastics (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Analytical Chemistry (AREA)
  • Toxicology (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2001539587A 1999-11-22 2000-11-16 新規官能化ポリマー試薬 Pending JP2003514876A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE9904222-8 1999-11-22
SE9904222A SE519326C2 (sv) 1999-11-22 1999-11-22 Funktionaliserade polymera reagens innefattande en syralabil isonitrildel samt förfarande för dess framställning
PCT/SE2000/002263 WO2001037983A1 (en) 1999-11-22 2000-11-16 New functionalized polymeric reagents

Publications (1)

Publication Number Publication Date
JP2003514876A true JP2003514876A (ja) 2003-04-22

Family

ID=20417810

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2001539587A Pending JP2003514876A (ja) 1999-11-22 2000-11-16 新規官能化ポリマー試薬

Country Status (6)

Country Link
EP (1) EP1239949A1 (sv)
JP (1) JP2003514876A (sv)
AU (1) AU769893B2 (sv)
CA (1) CA2389953A1 (sv)
SE (1) SE519326C2 (sv)
WO (1) WO2001037983A1 (sv)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10150077B4 (de) * 2001-10-10 2004-07-29 Morphochem Aktiengesellschaft für kombinatorische Chemie Verfahren zur Herstellung polymergebundener Isonitrile
DE10162134A1 (de) * 2001-12-18 2003-07-10 Morphochem Ag Ag Fuer Kombinat Harzgebundene Isonitrile
FR2856061A1 (fr) * 2003-06-11 2004-12-17 Chrysalon Derives polycycliques ortho-condenses de l'aminopyrrole a substituant electroattracteur chimiotheques combinatoires desdits derives et leur procede d'obtention
WO2005123140A2 (en) 2004-06-08 2005-12-29 Alza Corporation Preparation of macromolecular conjugates by four-component condensation reaction
CA2859205A1 (en) 2011-12-16 2013-06-20 Massachusetts Institute Of Technology Alpha-aminoamidine polymers and uses thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4812532A (en) * 1987-07-29 1989-03-14 Bio-Affinity Systems, Inc. Solid phase oxime reagent
AU1589099A (en) * 1997-11-18 1999-06-07 Rhone-Poulenc Rorer Pharmaceuticals Inc. Functionalized resin for the synthesis of amides and peptides

Also Published As

Publication number Publication date
AU769893B2 (en) 2004-02-05
SE9904222L (sv) 2001-05-23
CA2389953A1 (en) 2001-05-31
WO2001037983A1 (en) 2001-05-31
EP1239949A1 (en) 2002-09-18
SE9904222D0 (sv) 1999-11-22
AU1907401A (en) 2001-06-04
SE519326C2 (sv) 2003-02-11

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