JP2002526474A - 環状エステルまたはアミド誘導体 - Google Patents

環状エステルまたはアミド誘導体

Info

Publication number
JP2002526474A
JP2002526474A JP2000574071A JP2000574071A JP2002526474A JP 2002526474 A JP2002526474 A JP 2002526474A JP 2000574071 A JP2000574071 A JP 2000574071A JP 2000574071 A JP2000574071 A JP 2000574071A JP 2002526474 A JP2002526474 A JP 2002526474A
Authority
JP
Japan
Prior art keywords
compound
independently
cycloalkyl
fkbp
cycloalkenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000574071A
Other languages
English (en)
Japanese (ja)
Inventor
グレゴリー エス． ハミルトン、
デイヴィッド スィー． リンバーグ、
Original Assignee
ジーピーアイ ニル ホールディングス インコーポレイテッド
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ジーピーアイ ニル ホールディングス インコーポレイテッド filed Critical ジーピーアイ ニル ホールディングス インコーポレイテッド
Publication of JP2002526474A publication Critical patent/JP2002526474A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Immunology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Transplantation (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2000574071A 1998-09-21 1999-09-17 環状エステルまたはアミド誘導体 Pending JP2002526474A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US09/157,566 US6462072B1 (en) 1998-09-21 1998-09-21 Cyclic ester or amide derivatives
US09/157,566 1998-09-21
PCT/US1999/021290 WO2000017161A1 (en) 1998-09-21 1999-09-17 Cyclic ester or amide derivatives

Publications (1)

Publication Number Publication Date
JP2002526474A true JP2002526474A (ja) 2002-08-20

Family

ID=22564303

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000574071A Pending JP2002526474A (ja) 1998-09-21 1999-09-17 環状エステルまたはアミド誘導体

Country Status (11)

Country Link
US (1) US6462072B1 (US06462072-20021008-C00001.png)
EP (1) EP1115703A1 (US06462072-20021008-C00001.png)
JP (1) JP2002526474A (US06462072-20021008-C00001.png)
KR (1) KR20010089253A (US06462072-20021008-C00001.png)
CN (1) CN1323294A (US06462072-20021008-C00001.png)
AU (1) AU6390599A (US06462072-20021008-C00001.png)
CA (1) CA2341036A1 (US06462072-20021008-C00001.png)
HU (1) HUP0103565A3 (US06462072-20021008-C00001.png)
IL (1) IL141552A0 (US06462072-20021008-C00001.png)
WO (1) WO2000017161A1 (US06462072-20021008-C00001.png)
ZA (1) ZA200101934B (US06462072-20021008-C00001.png)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001060814A2 (en) * 2000-02-15 2001-08-23 Sugen, Inc. Pyrrole substituted 2-indolinone protein kinase inhibitors
AR042586A1 (es) 2001-02-15 2005-06-29 Sugen Inc 3-(4-amidopirrol-2-ilmetiliden)-2-indolinona como inhibidores de la protein quinasa; sus composiciones farmaceuticas; un metodo para la modulacion de la actividad catalitica de la proteinquinasa; un metodo para tratar o prevenir una afeccion relacionada con la proteinquinasa
EP1434774A1 (en) 2001-10-10 2004-07-07 Sugen, Inc. 3-(4-substituted heterocyclyl)-pyrrol-2-ylmethylidene)-2-indolinone derivatives as protein kinase inhibitors
US20060063828A1 (en) * 2004-06-28 2006-03-23 Weingarten M D 1,2-Bis-(substituted-phenyl)-2-propen-1-ones and pharmaceutical compositions thereof

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Also Published As

Publication number Publication date
IL141552A0 (en) 2002-03-10
HUP0103565A3 (en) 2002-02-28
ZA200101934B (en) 2002-09-18
WO2000017161A1 (en) 2000-03-30
HUP0103565A2 (hu) 2002-01-28
US6462072B1 (en) 2002-10-08
AU6390599A (en) 2000-04-10
CA2341036A1 (en) 2000-03-30
EP1115703A1 (en) 2001-07-18
CN1323294A (zh) 2001-11-21
KR20010089253A (ko) 2001-09-29

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