JP2002504535A5 - - Google Patents
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- Publication number
- JP2002504535A5 JP2002504535A5 JP2000533402A JP2000533402A JP2002504535A5 JP 2002504535 A5 JP2002504535 A5 JP 2002504535A5 JP 2000533402 A JP2000533402 A JP 2000533402A JP 2000533402 A JP2000533402 A JP 2000533402A JP 2002504535 A5 JP2002504535 A5 JP 2002504535A5
- Authority
- JP
- Japan
- Prior art keywords
- hydrazone
- hydroxylamine
- oxime
- hydrazine
- mol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/030,936 US6235936B1 (en) | 1998-02-26 | 1998-02-26 | Metal-catalyzed arylations of hydrazines, hydrazones, and related substrates |
| US5555798A | 1998-04-06 | 1998-04-06 | |
| US09/055,557 | 1998-04-06 | ||
| US09/030,936 | 1998-04-06 | ||
| PCT/US1999/004217 WO1999043643A2 (en) | 1998-02-26 | 1999-02-26 | Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2002504535A JP2002504535A (ja) | 2002-02-12 |
| JP2002504535A5 true JP2002504535A5 (https=) | 2006-04-20 |
| JP4647780B2 JP4647780B2 (ja) | 2011-03-09 |
Family
ID=26706608
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2000533402A Expired - Lifetime JP4647780B2 (ja) | 1998-02-26 | 1999-02-26 | ヒドラジン、ヒドラゾン、ヒドロキシルアミンおよびオキシムの金属−触媒アリール化およびビニル化 |
Country Status (6)
| Country | Link |
|---|---|
| EP (1) | EP1058678B1 (https=) |
| JP (1) | JP4647780B2 (https=) |
| AT (1) | ATE229499T1 (https=) |
| CA (1) | CA2322194C (https=) |
| DE (1) | DE69904448T2 (https=) |
| WO (1) | WO1999043643A2 (https=) |
Families Citing this family (35)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6677160B1 (en) | 1999-09-29 | 2004-01-13 | Pharmacia & Upjohn Company | Methods for creating a compound library and identifying lead chemical templates and ligands for target molecules |
| US6764858B2 (en) | 1999-09-29 | 2004-07-20 | Pharmacia & Upjohn Company | Methods for creating a compound library |
| CA2400094A1 (en) * | 1999-09-29 | 2001-04-05 | Pharmacia & Upjohn Company | Methods for creating a compound library and identifying lead chemical templates and ligands for target molecules |
| EP1130009A1 (en) * | 2000-03-01 | 2001-09-05 | Therascope AG | Generation and screening of a dynamic combinatorial library |
| US6706895B1 (en) | 2002-11-14 | 2004-03-16 | Uniroyal Chemical Company, Inc. | 4-methoxybiphenyl hydrazone derivatives |
| KR100676115B1 (ko) * | 2003-07-25 | 2007-02-02 | 아사히 가세이 케미칼즈 가부시키가이샤 | 산화 촉매 |
| FR2899897B1 (fr) | 2006-04-13 | 2008-06-27 | Oreal | Composes monochromophoriques monocationiques particuliers de type hydrazone comprenant un motif 2-, 4-pyridinium ou 2-, 4-quinolinium, leur synthese, compositions tinctoriales les comprenant, procede de coloration de fibres keratiniques |
| KR102065319B1 (ko) | 2007-03-12 | 2020-01-10 | 인트라-셀룰라 써래피스, 인코퍼레이티드. | 치환된 헤테로환 융합 감마-카르볼린 합성 |
| WO2009000411A1 (en) * | 2007-06-26 | 2008-12-31 | Sanofi-Aventis | A transition metal catalyzed synthesis of 2h-indazoles |
| BR112013001138A2 (pt) | 2010-07-16 | 2016-07-05 | Abbvie Inc | ligantes de fosfina para reações catalíticas |
| US9255074B2 (en) | 2010-07-16 | 2016-02-09 | Abbvie Inc. | Process for preparing antiviral compounds |
| US8975443B2 (en) | 2010-07-16 | 2015-03-10 | Abbvie Inc. | Phosphine ligands for catalytic reactions |
| US8895737B2 (en) | 2010-07-16 | 2014-11-25 | Shashank Shekhar | Process for preparing antiviral compounds |
| WO2013155504A1 (en) | 2012-04-14 | 2013-10-17 | Intra-Cellular Therapies, Inc. | Novel methods |
| JP6166996B2 (ja) * | 2013-09-27 | 2017-07-19 | 株式会社日本ファインケム | ヒドラジノアリールカルボン酸類の製造方法 |
| IL305990B2 (en) | 2013-12-03 | 2025-12-01 | Intra Cellular Therapies Inc | Long-acting injectable composition comprising polymeric microspheres of heterocycle fused gamma-carboline compounds or a pharmaceutical composition for sustained or delayed release comprising the compounds and their use in the treatment of bipolar disorder i and/or bipolar ii disorder |
| RU2016143091A (ru) | 2014-04-04 | 2018-05-08 | Интра-Селлулар Терапиз, Инк. | Органические соединения |
| MX365969B (es) | 2014-04-04 | 2019-06-21 | Intra Cellular Therapies Inc | Gamma-carbolinas fusionadas con heterociclos sustituidas con deuterio. |
| CN108883111B (zh) | 2016-01-26 | 2021-10-08 | 细胞内治疗公司 | 有机化合物 |
| PL3407889T3 (pl) | 2016-03-25 | 2021-11-22 | Intra-Cellular Therapies, Inc. | Związki organiczne i ich zastosowanie w leczeniu lub zapobieganiu zaburzeniom ośrodkowego układu nerwowego |
| EP3436083A4 (en) | 2016-03-28 | 2019-11-27 | Intra-Cellular Therapies, Inc. | NOVEL COMPOSITIONS AND METHOD |
| JP2019513143A (ja) | 2016-03-28 | 2019-05-23 | イントラ−セルラー・セラピーズ・インコーポレイテッドＩｎｔｒａ−Ｃｅｌｌｕｌａｒ Ｔｈｅｒａｐｉｅｓ， Ｉｎｃ． | 新規塩類および結晶 |
| US11014925B2 (en) | 2016-03-28 | 2021-05-25 | Intra-Cellular Therapies, Inc. | Co-crystals of 1-(4-fluoro-phenyl)-4-((6bR,1OaS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H- pyrido[3′,4′:4,51_pyrrolo [1,2,3-delqcuinoxalin-8-yl)-butan-1-one with nicotinamide or isonicotinamide |
| US11331316B2 (en) | 2016-10-12 | 2022-05-17 | Intra-Cellular Therapies, Inc. | Amorphous solid dispersions |
| US10961245B2 (en) | 2016-12-29 | 2021-03-30 | Intra-Cellular Therapies, Inc. | Substituted heterocycle fused gamma-carbolines for treatment of central nervous system disorders |
| US10906906B2 (en) | 2016-12-29 | 2021-02-02 | Intra-Cellular Therapies, Inc. | Organic compounds |
| IL268970B2 (en) | 2017-03-24 | 2023-12-01 | Intra Cellular Therapies Inc | Oral transmucosal formulations of substituted heterocycle fused gamma carbolines |
| JP7224333B2 (ja) | 2017-07-26 | 2023-02-17 | イントラ－セルラー・セラピーズ・インコーポレイテッド | 有機化合物 |
| JP7223742B2 (ja) | 2017-07-26 | 2023-02-16 | イントラ－セルラー・セラピーズ・インコーポレイテッド | 有機化合物 |
| AU2019240226B2 (en) | 2018-03-23 | 2024-11-28 | Intra-Cellular Therapies, Inc. | Organic compounds |
| IL321985A (en) | 2018-06-06 | 2025-09-01 | Intra Cellular Therapies Inc | New salts and crystals |
| WO2019237037A1 (en) | 2018-06-08 | 2019-12-12 | Intra-Cellular Therapies, Inc. | Novel methods |
| EP3843729A4 (en) | 2018-08-29 | 2022-06-01 | Intra-Cellular Therapies, Inc. | NOVEL COMPOSITIONS AND PROCESSES |
| CA3108558A1 (en) | 2018-08-31 | 2020-03-05 | Intra-Cellular Therapies, Inc. | Novel methods |
| CN112584837A (zh) | 2018-08-31 | 2021-03-30 | 细胞内治疗公司 | 新方法 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3867452A (en) * | 1970-12-30 | 1975-02-18 | Merrill Wilcox | 2-Nitrophenylhydrazines |
| US4374271A (en) * | 1974-12-04 | 1983-02-15 | United States Borax & Chemical Corporation | Nitrophenylhydrazine compounds |
| CH654286A5 (de) * | 1981-11-04 | 1986-02-14 | Ciba Geigy Ag | Verfahren zur pd-katalysierten arylierung von olefinen mit arylhalogeniden. |
| DE3447211A1 (de) * | 1984-12-22 | 1986-06-26 | Bayer Ag, 5090 Leverkusen | Verfahren zur herstellung von substituierten phenylhydrazinen |
| DE3617977A1 (de) * | 1985-12-05 | 1987-06-11 | Bayer Ag | 5-dichloracetamido-4-nitro-1-aryl-pyrazole |
| JP3059007B2 (ja) * | 1992-09-29 | 2000-07-04 | 協和醗酵工業株式会社 | １−（２−カルボキシフェニル）インダゾール誘導体の製造方法 |
| JPH0827109A (ja) * | 1994-07-14 | 1996-01-30 | Kuraray Co Ltd | β−（ベンジル）インドール−３−エタノールの製造方法 |
| CA2241219A1 (en) * | 1995-12-27 | 1997-07-10 | Basf Aktiengesellschaft | Iminooxyphenylacetic acid derivatives, their preparation, intermediates for their preparation, and their use |
| JPH09227485A (ja) * | 1996-02-16 | 1997-09-02 | Fuji Photo Film Co Ltd | ２−ヒドラジノナフタレン化合物の製造方法 |
| GB9610811D0 (en) * | 1996-05-23 | 1996-07-31 | Pharmacia Spa | Combinatorial solid phase synthesis of a library of indole derivatives |
| GB9610813D0 (en) * | 1996-05-23 | 1996-07-31 | Pharmacia Spa | Combinatorial solid phase synthesis of a library of benzufuran derivatives |
| US6103937A (en) * | 1996-07-01 | 2000-08-15 | E. I. Du Pont De Nemours And Company | Nickel catalyzed addition of -NH- containing compounds to vinyl and aryl halides |
| WO1998046561A1 (en) * | 1997-04-11 | 1998-10-22 | Otsuka Chemical Co., Ltd. | Benzene derivatives, benzofuran derivatives, and processes for producing these |
| DE19728760C1 (de) * | 1997-07-04 | 1998-10-29 | Celanese Gmbh | Verfahren zur Aminierung von Arylverbindungen in Gegenwart eines Palladium-Komplexkatalysators |
-
1999
- 1999-02-26 WO PCT/US1999/004217 patent/WO1999043643A2/en not_active Ceased
- 1999-02-26 CA CA2322194A patent/CA2322194C/en not_active Expired - Lifetime
- 1999-02-26 JP JP2000533402A patent/JP4647780B2/ja not_active Expired - Lifetime
- 1999-02-26 AT AT99908515T patent/ATE229499T1/de not_active IP Right Cessation
- 1999-02-26 DE DE69904448T patent/DE69904448T2/de not_active Expired - Lifetime
- 1999-02-26 EP EP99908515A patent/EP1058678B1/en not_active Expired - Lifetime
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