JP2002503674A5 - - Google Patents

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Publication number
JP2002503674A5
JP2002503674A5 JP2000531467A JP2000531467A JP2002503674A5 JP 2002503674 A5 JP2002503674 A5 JP 2002503674A5 JP 2000531467 A JP2000531467 A JP 2000531467A JP 2000531467 A JP2000531467 A JP 2000531467A JP 2002503674 A5 JP2002503674 A5 JP 2002503674A5
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JP
Japan
Prior art keywords
chemical
compound according
nrr
ring
nhr
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000531467A
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English (en)
Japanese (ja)
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JP2002503674A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1998/002891 external-priority patent/WO1999041276A1/en
Publication of JP2002503674A publication Critical patent/JP2002503674A/ja
Publication of JP2002503674A5 publication Critical patent/JP2002503674A5/ja
Pending legal-status Critical Current

Links

JP2000531467A 1998-02-12 1998-02-12 βシート模倣物およびその使用に関する方法 Pending JP2002503674A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/US1998/002891 WO1999041276A1 (en) 1998-02-12 1998-02-12 β-SHEET MIMETICS AND METHODS RELATING TO THE USE THEREOF

Publications (2)

Publication Number Publication Date
JP2002503674A JP2002503674A (ja) 2002-02-05
JP2002503674A5 true JP2002503674A5 (cg-RX-API-DMAC7.html) 2005-12-22

Family

ID=22266392

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000531467A Pending JP2002503674A (ja) 1998-02-12 1998-02-12 βシート模倣物およびその使用に関する方法

Country Status (9)

Country Link
EP (1) EP1053246B1 (cg-RX-API-DMAC7.html)
JP (1) JP2002503674A (cg-RX-API-DMAC7.html)
KR (1) KR20010040939A (cg-RX-API-DMAC7.html)
AT (1) ATE230414T1 (cg-RX-API-DMAC7.html)
AU (1) AU748887B2 (cg-RX-API-DMAC7.html)
CA (1) CA2319766A1 (cg-RX-API-DMAC7.html)
DE (1) DE69810513T2 (cg-RX-API-DMAC7.html)
ES (1) ES2192764T3 (cg-RX-API-DMAC7.html)
WO (1) WO1999041276A1 (cg-RX-API-DMAC7.html)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2003525294A (ja) * 2000-02-29 2003-08-26 ブリストル−マイヤーズ スクイブ ファーマ カンパニー C型肝炎ウイルスns3プロテアーゼの阻害剤
US6534651B2 (en) 2000-04-06 2003-03-18 Inotek Pharmaceuticals Corp. 7-Substituted isoindolinone inhibitors of inflammation and reperfusion injury and methods of use thereof
US20060276497A1 (en) 2000-05-09 2006-12-07 Cephalon, Inc. Novel multicyclic compounds and the use thereof
US7122679B2 (en) 2000-05-09 2006-10-17 Cephalon, Inc. Multicyclic compounds and the use thereof
CN1642550A (zh) * 2002-02-14 2005-07-20 美瑞德生物工程公司 β-折叠模拟物和组合物及其有关方法
JP2011525927A (ja) * 2008-06-25 2011-09-29 シェーリング コーポレイション 複素環式抗菌剤の合成および使用
BR112017006920A8 (pt) 2014-10-06 2023-03-07 Quince Therapeutics Inc Inibidores de lisina gingipaína
EP3374352A4 (en) 2015-11-09 2019-10-02 Cortexyme, Inc. GINGIPAINE ARGININE INHIBITORS
PL3486242T3 (pl) 2016-08-31 2022-03-21 Jiangsu Hengrui Medicine Co. Ltd. Pochodna oksopikolinamidu, sposób jej wytwarzania i zastosowanie farmaceutyczne
MX2019003087A (es) 2016-09-16 2019-08-12 Cortexyme Inc Inhibidores cetónicos de gingipain de lisina.
EP3822264A4 (en) 2018-07-02 2021-11-10 Jiangsu Hengrui Medicine Co., Ltd. CRYSTALLINE FORMS OF AN OXYPYRIDINE AMIDE DERIVATIVE AND THEIR PREPARATION PROCESS
WO2021057818A1 (zh) 2019-09-27 2021-04-01 深圳信立泰药业股份有限公司 FXIa抑制剂及其制备方法和医药用途

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2117123T3 (es) * 1992-02-14 1998-08-01 Merrell Pharma Inc Derivados de aminocetilmercaptoacetilamida utilizados como inhibidores de la encefalinasa y del enzima de conversion de angiotensina.
ES2138622T3 (es) * 1992-05-15 2000-01-16 Merrell Pharma Inc Derivados de mercaptoacetilamido piridazo(1,2-a)(1,2)diazepina utilizados como inhibidores de encefalinasa y eca.
EP0618223A3 (en) * 1993-03-08 1996-06-12 Sandoz Ltd Peptides, the release of Interleukin 1-Bêta, useful as anti-inflammatory agents.
SK83897A3 (en) * 1994-12-22 1998-05-06 Iaf Biochem Int Low molecular weight bicyclic thrombin inhibitors
EP0815123B1 (en) * 1995-03-24 2001-10-04 Molecumetics, Ltd. Beta-sheet mimetics and use thereof as protease inhibitors
WO1996030396A1 (en) * 1995-03-24 1996-10-03 Molecumetics Ltd. β-SHEET MIMETICS AND USE THEREOF AS PROTEASE INHIBITORS
US5877313A (en) * 1995-05-17 1999-03-02 Bristol-Myers Squibb Benzo-fused azepinone and piperidinone compounds useful in the inhibition of ACE and NEP
IT1277405B1 (it) * 1995-08-01 1997-11-10 Menarini Farma Ind Derivati di lattami biciclici come inibitori della trombina
WO1998005333A1 (en) * 1996-08-05 1998-02-12 Molecumetics Ltd. Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors

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