JP2002501514A5 - - Google Patents

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Publication number
JP2002501514A5
JP2002501514A5 JP1999500130A JP50013099A JP2002501514A5 JP 2002501514 A5 JP2002501514 A5 JP 2002501514A5 JP 1999500130 A JP1999500130 A JP 1999500130A JP 50013099 A JP50013099 A JP 50013099A JP 2002501514 A5 JP2002501514 A5 JP 2002501514A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1999500130A
Other languages
English (en)
Japanese (ja)
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JP4447663B2 (ja
JP2002501514A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/DK1998/000225 external-priority patent/WO1998054181A1/en
Publication of JP2002501514A publication Critical patent/JP2002501514A/ja
Publication of JP2002501514A5 publication Critical patent/JP2002501514A5/ja
Application granted granted Critical
Publication of JP4447663B2 publication Critical patent/JP4447663B2/ja
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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JP50013099A 1997-05-30 1998-05-29 ニコチン性achレセプターに於けるコリン作動性リガンドとしての8−アザビシクロ(3.2.1)オクト−2−エン及びオクタン誘導体 Expired - Fee Related JP4447663B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
DK62797 1997-05-30
DK0627/97 1997-05-30
DK150297 1997-12-19
DK1502/97 1997-12-19
DK0408/98 1998-03-24
DK40898 1998-03-24
DK0534/98 1998-04-16
DK53498 1998-04-16
PCT/DK1998/000225 WO1998054181A1 (en) 1997-05-30 1998-05-29 8-azabicyclo(3,2,1)oct-2-ene and octane derivatives as cholinergic ligands at nicotinic ach receptors

Publications (3)

Publication Number Publication Date
JP2002501514A JP2002501514A (ja) 2002-01-15
JP2002501514A5 true JP2002501514A5 (enExample) 2005-12-08
JP4447663B2 JP4447663B2 (ja) 2010-04-07

Family

ID=27439314

Family Applications (1)

Application Number Title Priority Date Filing Date
JP50013099A Expired - Fee Related JP4447663B2 (ja) 1997-05-30 1998-05-29 ニコチン性achレセプターに於けるコリン作動性リガンドとしての8−アザビシクロ(3.2.1)オクト−2−エン及びオクタン誘導体

Country Status (22)

Country Link
US (2) US6645977B1 (enExample)
EP (1) EP0984965B1 (enExample)
JP (1) JP4447663B2 (enExample)
KR (1) KR100589872B1 (enExample)
CN (1) CN1157392C (enExample)
AT (1) ATE267199T1 (enExample)
AU (1) AU745964B2 (enExample)
BR (1) BR9809697A (enExample)
CA (1) CA2289574C (enExample)
CZ (1) CZ298824B6 (enExample)
DE (1) DE69823994T2 (enExample)
DK (1) DK0984965T3 (enExample)
EE (1) EE04057B1 (enExample)
HU (1) HUP0002713A3 (enExample)
IL (2) IL132437A0 (enExample)
IS (1) IS2092B (enExample)
NO (1) NO325513B1 (enExample)
NZ (1) NZ500642A (enExample)
RU (1) RU2186780C2 (enExample)
SK (1) SK284994B6 (enExample)
TR (1) TR199902942T2 (enExample)
WO (1) WO1998054181A1 (enExample)

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AU2004220327B2 (en) 2003-03-12 2010-06-24 Pfizer Products Inc. Pyridyloxymethyl and benzisoxazole azabicyclic derivatives
CA2580329C (en) 2004-09-13 2015-01-06 Chrono Therapeutics Inc. Biosynchronous transdermal drug delivery
US20060173037A1 (en) * 2005-01-10 2006-08-03 Nathalie Schlienger Aminophenyl derivatives as selective androgen receptor modulators
ATE495178T1 (de) 2005-02-16 2011-01-15 Neurosearch As Diazabicyclische arylderivate und ihre verwendung als chinolinergische liganden an nikotin- acetylcholin-rezeptoren
DE102005007859A1 (de) * 2005-02-21 2006-08-24 Lts Lohmann Therapie-Systeme Ag Vefahren für eine medikamentöse Kombinations-Behandlung, sowie hierfür geeignete Arzneimittel-Kombinationen
WO2006108790A1 (en) * 2005-04-08 2006-10-19 Neurosearch A/S (+) - and (-) -8-alkyl-3-(trifluoralkylsulfonyloxy)-8-azabicycl (3.2.1.)oct-2-ene
FR2889701B1 (fr) 2005-08-12 2007-10-05 Sanofi Aventis Sa Derives de 5-pyridinyl-1-azabicyclo[3.2.1]octane, leur preparation en therapeutique.
EP1963323B1 (en) 2005-12-06 2010-07-14 Neurosearch A/S Novel diazabicyclic aryl derivatives and their medical use
US20070134169A1 (en) * 2005-12-11 2007-06-14 Rabinoff Michael D Methods for smoking cessation or alcohol cessation or other addiction cessation
AU2007213670A1 (en) 2006-02-10 2007-08-16 Neurosearch A/S 3,9-diazabicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
US7700596B2 (en) 2006-02-10 2010-04-20 Neurosearch A/S 3,9-diazabicyclo[3.3.1]nonane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
EP1987031A1 (en) 2006-02-10 2008-11-05 NeuroSearch A/S 3-heteroaryl- 3,9-diazabicyclo[3.3.1]nonane derivatives as nicotinic acetylcholine receptor agonists
US20090247570A1 (en) * 2006-06-12 2009-10-01 Pfizer Inc Pharmaceuticals
EP1977746B8 (en) 2007-04-02 2014-09-24 Parkinson's Institute Methods and compositions for reduction of side effects of therapeutic treatments
TWI415850B (zh) * 2007-07-20 2013-11-21 Theravance Inc 製備mu類鴉片受體拮抗劑之中間物的方法
SA08290475B1 (ar) 2007-08-02 2013-06-22 Targacept Inc (2s، 3r)-n-(2-((3-بيردينيل)ميثيل)-1-آزا بيسيكلو[2، 2، 2]أوكت-3-يل)بنزو فيوران-2-كربوكساميد، وصور أملاحه الجديدة وطرق استخدامه
US8697722B2 (en) * 2007-11-02 2014-04-15 Sri International Nicotinic acetylcholine receptor modulators
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JP2012509354A (ja) * 2008-11-18 2012-04-19 ノイロサーチ アクティーゼルスカブ 8−アザビシクロ[3.2.1]オクタ−2−エン誘導体及びモノアミン神経伝達物質再取込阻害剤としてのそれらの使用
SI2889033T1 (en) 2008-11-19 2018-08-31 Forum Pharmaceuticals Inc. Treatment of negative symptoms of schizophrenia with (R) -7-chloro-N- (chonylidin-3-yl) benzo (B) thiophene-2-carboxamide and pharmaceutically acceptable salts thereof
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WO2010132423A1 (en) * 2009-05-11 2010-11-18 Envivo Pharmaceuticals, Inc. Treatment of cognitive disorders with certain alpha-7 nicotinic acid receptors in combination with acetylcholinesterase inhibitors
EP2523562B1 (en) * 2010-01-11 2019-01-02 Astraea Therapeutics, LLC Nicotinic acetylcholine receptor modulators
CN103221411B (zh) 2010-05-17 2016-05-11 富瑞姆制药公司 (R)-7-氯-N-(奎宁环-3-基)苯并[b]噻吩-2-甲酰胺盐酸盐单水合物的晶型
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WO2014011768A1 (en) * 2012-07-10 2014-01-16 Adispell, Inc. Anti-anxiety treatment
CA2974324A1 (en) 2015-01-28 2016-08-04 Zita S. Netzel Drug delivery methods and systems
US9724340B2 (en) 2015-07-31 2017-08-08 Attenua, Inc. Antitussive compositions and methods
EP3565617A1 (en) 2017-01-06 2019-11-13 Chrono Therapeutics Inc. Transdermal drug delivery devices and methods
US11596779B2 (en) 2018-05-29 2023-03-07 Morningside Venture Investments Limited Drug delivery methods and systems
CA3119992A1 (en) 2018-11-16 2020-05-22 Morningside Venture Investments Limited Thermally regulated transdermal drug delivery system
KR102272452B1 (ko) 2020-12-11 2021-07-05 (주)예광솔라 스파이럴 파일 공법 및 이에 적용되는 스파이럴 파일
KR200497569Y1 (ko) 2021-02-18 2023-12-21 주식회사 알파인랩 지주 기초용 스크루 파일

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