JP2002500618A5 - - Google Patents

Download PDF

Info

Publication number
JP2002500618A5
JP2002500618A5 JP1997525183A JP52518397A JP2002500618A5 JP 2002500618 A5 JP2002500618 A5 JP 2002500618A5 JP 1997525183 A JP1997525183 A JP 1997525183A JP 52518397 A JP52518397 A JP 52518397A JP 2002500618 A5 JP2002500618 A5 JP 2002500618A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP1997525183A
Other languages
English (en)
Japanese (ja)
Other versions
JP2002500618A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1996/017995 external-priority patent/WO1997025033A1/en
Publication of JP2002500618A publication Critical patent/JP2002500618A/ja
Publication of JP2002500618A5 publication Critical patent/JP2002500618A5/ja
Withdrawn legal-status Critical Current

Links

JP52518397A 1995-10-31 1996-10-30 抗血栓性ジアミン Withdrawn JP2002500618A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US712095P 1995-10-31 1995-10-31
US2825296P 1996-10-09 1996-10-09
US60/028,252 1996-10-09
US60/007,120 1996-10-09
PCT/US1996/017995 WO1997025033A1 (en) 1995-10-31 1996-10-30 Antithrombotic diamines

Publications (2)

Publication Number Publication Date
JP2002500618A JP2002500618A (ja) 2002-01-08
JP2002500618A5 true JP2002500618A5 (OSRAM) 2004-10-28

Family

ID=26676549

Family Applications (1)

Application Number Title Priority Date Filing Date
JP52518397A Withdrawn JP2002500618A (ja) 1995-10-31 1996-10-30 抗血栓性ジアミン

Country Status (9)

Country Link
US (3) US6025382A (OSRAM)
EP (1) EP0863755B1 (OSRAM)
JP (1) JP2002500618A (OSRAM)
AT (1) ATE284690T1 (OSRAM)
AU (1) AU7725596A (OSRAM)
CA (1) CA2236007A1 (OSRAM)
DE (1) DE69634045T2 (OSRAM)
ES (1) ES2233982T3 (OSRAM)
WO (1) WO1997025033A1 (OSRAM)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2217373A1 (en) * 1996-10-10 1998-04-10 Michael John Martin Benzo¬b|thiophene compounds, intermediates, formulations, and methods
AU7170898A (en) * 1997-04-30 1998-11-24 Eli Lilly And Company Antithrombotic agents
WO1998049161A1 (en) 1997-04-30 1998-11-05 Eli Lilly And Company Antithrombotic agents
DE69828522T2 (de) 1997-04-30 2005-12-15 Eli Lilly And Co., Indianapolis Antithrombotische mittel
WO1998048797A1 (en) 1997-04-30 1998-11-05 Eli Lilly And Company Antithrombotic agents
US6271227B1 (en) 1997-04-30 2001-08-07 Eli Lilly And Company Antithrombotic Agents
CA2287984A1 (en) 1997-05-01 1998-11-05 Gerald Floyd Smith Antithrombotic agents
US7008950B1 (en) 1997-06-05 2006-03-07 Takeda Chemical Industries, Ltd. Benzofurans as suppressors of neurodegeneration
US6017914A (en) * 1997-09-03 2000-01-25 Eli Lilly And Company Benzo[b]thiophene compounds, intermediates, formulations, and methods
US6284756B1 (en) 1998-04-30 2001-09-04 Eli Lilly And Company Antithrombotic agents
US6166069A (en) * 1998-05-12 2000-12-26 American Home Products Corporation Phenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
PT997460E (pt) * 1998-10-28 2003-03-31 Lilly Co Eli Compostos benzotiofenos como agentes antitromboticos e seus intermediarios
ATE258934T1 (de) 1998-10-30 2004-02-15 Lilly Co Eli Azaindol derivate und ihre verwendung als antithrombotische wirkstoffe
ATE259802T1 (de) * 1999-11-19 2004-03-15 Lilly Co Eli Verbindungen mit antithrombotischer wirkung
CA2444787A1 (en) 2001-05-22 2002-11-28 Eli Lilly And Company Tetrahydroquinolin derivatives for the inhibition of diseases associated with estrogen deprivation or with an aberrant physiological response to endogenous estrogen
WO2002094788A1 (en) 2001-05-22 2002-11-28 Eli Lilly And Company 2-substituted 1,2,3,4-tetrahydroquinolines and derivatives thereof, compositions and methods
US7482366B2 (en) 2001-12-21 2009-01-27 X-Ceptor Therapeutics, Inc. Modulators of LXR
AU2002351412B2 (en) 2001-12-21 2010-05-20 Exelixis Patent Company Llc Modulators of LXR
EP1530470B9 (en) * 2002-07-22 2010-04-07 Eli Lilly And Company Selective estrogen receptor modulators containing a phenylsulfonyl group
US7296361B2 (en) * 2003-07-31 2007-11-20 University Of Pittsburgh Measuring device and method of measuring
US8785403B2 (en) 2003-08-01 2014-07-22 Mitsubishi Tanabe Pharma Corporation Glucopyranoside compound
ES2649737T5 (es) 2003-08-01 2021-07-07 Mitsubishi Tanabe Pharma Corp Compuestos novedosos que tienen actividad inhibidora frente a transportador de glucosa dependiente de sodio
AU2006212726C1 (en) 2005-02-14 2013-05-16 Bionomics Limited Novel tubulin polymerisation inhibitors
GB0507577D0 (en) 2005-04-14 2005-05-18 Novartis Ag Organic compounds
UY30730A1 (es) 2006-12-04 2008-07-03 Mitsubishi Tanabe Pharma Corp Forma cristalina del hemihidrato de 1-(b (beta)-d-glucopiranosil) -4-metil-3-[5-(4-fluorofenil) -2-tienilmetil]benceno
CA2699285C (en) 2007-09-10 2016-12-13 Ahmed F. Abdel-Magid Process for the preparation of compounds useful as inhibitors of sodium-dependent glucose transporter (sglt)
CL2008003653A1 (es) 2008-01-17 2010-03-05 Mitsubishi Tanabe Pharma Corp Uso de un inhibidor de sglt derivado de glucopiranosilo y un inhibidor de dppiv seleccionado para tratar la diabetes; y composicion farmaceutica.
US9056850B2 (en) 2008-10-17 2015-06-16 Janssen Pharmaceutica N.V. Process for the preparation of compounds useful as inhibitors of SGLT
US20110009347A1 (en) 2009-07-08 2011-01-13 Yin Liang Combination therapy for the treatment of diabetes
IN2012DN03299A (OSRAM) 2009-10-14 2015-10-23 Janssen Pharmaceutica Nv
SG185525A1 (en) 2010-05-11 2012-12-28 Janssen Pharmaceutica Nv Pharmaceutical formulations comprising 1 - (beta-d-glucopyranosyl) - 2 -thienylmethylbenzene derivatives as inhibitors of sglt
AU2012241897C1 (en) 2011-04-13 2017-05-11 Janssen Pharmaceutica Nv Process for the preparation of compounds useful as inhibitors of SGLT2
US9035044B2 (en) 2011-05-09 2015-05-19 Janssen Pharmaceutica Nv L-proline and citric acid co-crystals of (2S, 3R, 4R, 5S,6R)-2-(3-((5-(4-fluorophenyl)thiopen-2-yl)methyl)4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
ES2570862T3 (es) 2011-12-15 2016-05-20 Bayer Ip Gmbh Benzotienil-pirrolotriazinas sustituidas y usos de las mismas en el tratamiento de cáncer
WO2013124316A1 (en) 2012-02-23 2013-08-29 Bayer Intellectual Property Gmbh Substituted benzothienyl-pyrrolotriazines and uses thereof
WO2016132998A1 (ja) * 2015-02-19 2016-08-25 Jnc株式会社 ベンゾチオフェンを有する液晶性化合物、液晶組成物および液晶表示素子
US20170071970A1 (en) 2015-09-15 2017-03-16 Janssen Pharmaceutica Nv Co-therapy comprising canagliflozin and phentermine for the treatment of obesity and obesity related disorders
CN114539273A (zh) 2016-06-07 2022-05-27 北京加科思新药研发有限公司 可用作shp2抑制剂的新型杂环衍生物
HRP20241239T1 (hr) 2017-03-23 2024-12-06 Jacobio Pharmaceuticals Co., Ltd. Novi heterociklički derivati korisni kao shp2 inhibitori
WO2020063760A1 (en) 2018-09-26 2020-04-02 Jacobio Pharmaceuticals Co., Ltd. Novel heterocyclic derivatives useful as shp2 inhibitors

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3274213A (en) * 1961-09-05 1966-09-20 Upjohn Co Alkoxy-substituted 2-phenyl-1-(tertiary-aminoalkoxy)phenyl-3, 4-dihydronaphthalenes
US3293263A (en) * 1963-12-09 1966-12-20 Upjohn Co Diphenylbenzocycloalkenes
GB1456323A (en) * 1974-06-06 1976-11-24 Labaz Benzothiophenes process for preparing them and pharmaceutical compositions containing the same
US4001426A (en) * 1974-10-17 1977-01-04 Smithkline Corporation Substituted benzofurans and benzothiophenes
US4133814A (en) * 1975-10-28 1979-01-09 Eli Lilly And Company 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents
CA2073776A1 (en) 1990-11-15 1992-05-16 Joerg Stuerzebecher Meta-substituted phenyl alanine derivatives
JP3157882B2 (ja) * 1991-11-15 2001-04-16 帝国臓器製薬株式会社 新規なベンゾチオフエン誘導体
US5371091A (en) * 1992-08-31 1994-12-06 Bristol-Myers Squibb Company Heteroaromatic amine thrombin inhibitors
US6756388B1 (en) * 1993-10-12 2004-06-29 Pfizer Inc. Benzothiophenes and related compounds as estrogen agonists
US5441965A (en) * 1993-12-21 1995-08-15 Eli Lilly And Company Methods of inhibiting thrombin
US5510357A (en) * 1995-02-28 1996-04-23 Eli Lilly And Company Benzothiophene compounds as anti-estrogenic agents
US5523309A (en) * 1995-03-10 1996-06-04 Eli Lilly And Company Benzofuran pharmaceutical compounds
CA2218756A1 (en) 1996-10-25 1998-04-25 Kristin Sue Marron Substituted benzo¢b!thiophene compounds having activity as selective estrogen receptor modulators
US5929090A (en) 1997-09-12 1999-07-27 Eli Lilly And Company 2-aryl-3-aminoaryloxynaphthy1 compounds, intermediates, compositions and methods

Similar Documents

Publication Publication Date Title
JP2000515716A5 (OSRAM)
JP2000500228A5 (OSRAM)
JP2000500445A5 (OSRAM)
JP2000500440A5 (OSRAM)
JP2000500327A5 (OSRAM)
JP2001504574A5 (OSRAM)
JP2000501955A5 (OSRAM)
JP2000500145A5 (OSRAM)
JP2000500155A5 (OSRAM)
JP2001526734A5 (OSRAM)
JPH11511571A5 (OSRAM)
JP2000500115A5 (OSRAM)
JP2000500322A5 (OSRAM)
JP2000500258A5 (OSRAM)
JP2000500342A5 (OSRAM)
JP2000500192A5 (OSRAM)
JPH11510414A5 (OSRAM)
JP2000500112A5 (OSRAM)
JP2002500618A5 (OSRAM)
JP2000500226A5 (OSRAM)
JP2000500611A5 (OSRAM)
JP2000500407A5 (OSRAM)
JPH10501516A5 (OSRAM)
JP2000500166A5 (OSRAM)
JP2000500125A5 (OSRAM)