JP2001523221A - 親油性物質の促進された生物学的利用能のための固形共沈物 - Google Patents
親油性物質の促進された生物学的利用能のための固形共沈物Info
- Publication number
- JP2001523221A JP2001523221A JP51187998A JP51187998A JP2001523221A JP 2001523221 A JP2001523221 A JP 2001523221A JP 51187998 A JP51187998 A JP 51187998A JP 51187998 A JP51187998 A JP 51187998A JP 2001523221 A JP2001523221 A JP 2001523221A
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- Japan
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- composition
- tpgs
- coprecipitate
- solid
- lipophilic
- Prior art date
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- Ceased
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US119176 | 1987-11-10 | ||
| IL11917696A IL119176A (en) | 1996-09-01 | 1996-09-01 | Soluble coprecipitates for enhanced oral bioavailability of lipophilic substances |
| US08/833,076 US5891469A (en) | 1997-04-02 | 1997-04-02 | Solid Coprecipitates for enhanced bioavailability of lipophilic substances |
| US08/833,076 | 1997-04-02 | ||
| PCT/US1997/015072 WO1998008490A1 (en) | 1996-09-01 | 1997-08-27 | Solid coprecipitates for enhanced bioavailability of lipophilic substances |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2001523221A true JP2001523221A (ja) | 2001-11-20 |
| JP2001523221A5 JP2001523221A5 (enExample) | 2005-05-12 |
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| Application Number | Title | Priority Date | Filing Date |
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| JP51187998A Ceased JP2001523221A (ja) | 1996-09-01 | 1997-08-27 | 親油性物質の促進された生物学的利用能のための固形共沈物 |
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| Country | Link |
|---|---|
| EP (1) | EP1017366A4 (enExample) |
| JP (1) | JP2001523221A (enExample) |
| AU (1) | AU730216B2 (enExample) |
| CA (1) | CA2264718C (enExample) |
| WO (1) | WO1998008490A1 (enExample) |
Cited By (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2005531652A (ja) * | 2002-06-07 | 2005-10-20 | フラメル・テクノロジー | α−トコフェロールを用いて機能化されたポリアミノ酸、およびその使用、特に治療学的使用 |
| JP2006517929A (ja) * | 2003-02-19 | 2006-08-03 | ハー・ルンドベック・アクチエゼルスカベット | 溶融アグロメレーションを用いてアグロメレートを製造する方法 |
| JP2007510658A (ja) * | 2003-11-03 | 2007-04-26 | リポシン， インコーポレイテッド | 可溶化剤放出が同調する薬学的組成物 |
| JP2008514607A (ja) * | 2004-09-24 | 2008-05-08 | ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド | 新規な種類の界面活性剤様物質 |
| WO2009113522A1 (ja) * | 2008-03-11 | 2009-09-17 | あすか製薬株式会社 | 固体分散体とその医薬組成物、並びにそれらの製造方法 |
| JP2010150264A (ja) * | 2005-12-19 | 2010-07-08 | Ind Technol Res Inst | グルタチオンベースデリバリーシステム |
| WO2010092925A1 (ja) * | 2009-02-12 | 2010-08-19 | あすか製薬株式会社 | 固体分散体とその医薬組成物、並びにそれらの製造方法 |
| JP2012516346A (ja) * | 2009-01-29 | 2012-07-19 | ノバルティス アーゲー | ピリドピリミジノンの経口用固体製剤 |
| JP2012524092A (ja) * | 2009-04-14 | 2012-10-11 | ブリストル−マイヤーズ スクイブ カンパニー | アモルファスアルファ−（ｎ−スルホンアミド）アセトアミド化合物の生物学的に利用可能なカプセル組成物 |
| US8673863B2 (en) | 2005-12-19 | 2014-03-18 | Industrial Technology Research Institute | Glutathione-based delivery system |
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- 1997-08-27 AU AU42373/97A patent/AU730216B2/en not_active Ceased
- 1997-08-27 JP JP51187998A patent/JP2001523221A/ja not_active Ceased
- 1997-08-27 WO PCT/US1997/015072 patent/WO1998008490A1/en not_active Ceased
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Also Published As
| Publication number | Publication date |
|---|---|
| EP1017366A4 (en) | 2006-03-22 |
| AU730216B2 (en) | 2001-03-01 |
| AU4237397A (en) | 1998-03-19 |
| CA2264718C (en) | 2006-05-30 |
| CA2264718A1 (en) | 1998-03-05 |
| EP1017366A1 (en) | 2000-07-12 |
| WO1998008490A1 (en) | 1998-03-05 |
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