JP2001510200A5 - - Google Patents

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Publication number
JP2001510200A5
JP2001510200A5 JP2000503098A JP2000503098A JP2001510200A5 JP 2001510200 A5 JP2001510200 A5 JP 2001510200A5 JP 2000503098 A JP2000503098 A JP 2000503098A JP 2000503098 A JP2000503098 A JP 2000503098A JP 2001510200 A5 JP2001510200 A5 JP 2001510200A5
Authority
JP
Japan
Prior art keywords
estrone
compound
compounds
sulfatase
estrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2000503098A
Other languages
English (en)
Japanese (ja)
Other versions
JP2001510200A (ja
Filing date
Publication date
Priority claimed from US08/897,247 external-priority patent/US5880115A/en
Application filed filed Critical
Publication of JP2001510200A publication Critical patent/JP2001510200A/ja
Publication of JP2001510200A5 publication Critical patent/JP2001510200A5/ja
Pending legal-status Critical Current

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JP2000503098A 1997-07-18 1998-07-08 ステロイドスルファターゼ阻害剤並びにその製造及び使用方法 Pending JP2001510200A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/897,247 1997-07-18
US08/897,247 US5880115A (en) 1997-07-18 1997-07-18 Steroid sulfatase inhibitors and methods for making and using the same
PCT/US1998/014206 WO1999003876A1 (en) 1997-07-18 1998-07-08 Steroid sulfatase inhibitors and methods for making and using the same

Publications (2)

Publication Number Publication Date
JP2001510200A JP2001510200A (ja) 2001-07-31
JP2001510200A5 true JP2001510200A5 (enExample) 2006-01-05

Family

ID=25407613

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2000503098A Pending JP2001510200A (ja) 1997-07-18 1998-07-08 ステロイドスルファターゼ阻害剤並びにその製造及び使用方法

Country Status (8)

Country Link
US (1) US5880115A (enExample)
EP (1) EP1009755B1 (enExample)
JP (1) JP2001510200A (enExample)
AT (1) ATE250077T1 (enExample)
AU (1) AU729325B2 (enExample)
CA (1) CA2296498A1 (enExample)
DE (1) DE69818278T2 (enExample)
WO (1) WO1999003876A1 (enExample)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6476011B1 (en) * 1991-08-28 2002-11-05 Sterix Limited Methods for introducing an estrogenic compound
GB9118478D0 (en) * 1991-08-29 1991-10-16 Imperial College Steroid sulphatase inhibitors
US6011024A (en) 1991-08-28 2000-01-04 Imperial College Of Science Technology & Medicine Steroid sulphatase inhibitors
US6288050B1 (en) 1997-07-18 2001-09-11 Duquesne University Of The Holy Ghost Steroid sulfatase inhibitors and methods for making and using the same
US6376687B1 (en) * 1997-07-18 2002-04-23 Duquesne University Of The Holy Ghost Steroid sulfatase inhibitors and methods for making and using the same
ATE473759T1 (de) 1998-05-22 2010-07-15 Univ Leland Stanford Junior Bifunktionelle moleküle sowie darauf basierende therapien.
AU765386B2 (en) 1998-06-10 2003-09-18 Sterix Limited Pharmaceutical composition with tumor necrosis factor a and 2-methoxyestrone-3-(o)-sulphamate for inhibition of estrone sulphatase
US6248780B1 (en) 1998-10-01 2001-06-19 Duquesne University Of The Holy Ghost Compounds for the treatment of estrogen-dependent illnesses and methods for making and using the same
JP2000309599A (ja) 1999-04-13 2000-11-07 Kyowa Hakko Kogyo Co Ltd エストラ−１，３，５（１０），１６−テトラエン誘導体
US7078395B1 (en) 1999-06-16 2006-07-18 Sterix Limited Methods for treating or preventing cancer by preventing, inhibiting or arresting cell cycling
NZ515061A (en) 1999-04-30 2004-04-30 Sterix Ltd Use of a cyclic compound in cell cycling
US7335650B2 (en) * 2000-01-14 2008-02-26 Sterix Limited Composition
AU2001248849A1 (en) * 2000-04-24 2001-11-07 Kyowa Hakko Kogyo Co. Ltd. Estra-1,3,5(10)-triene derivatives
GB0025788D0 (en) * 2000-10-20 2000-12-06 Sterix Ltd Use
US7125565B2 (en) 2000-12-01 2006-10-24 Kyowa Hakko Kogyo Co., Ltd. Composition improved in the solubility or oral absorbability
EP2147679B1 (en) 2001-07-25 2014-06-25 Raptor Pharmaceutical, Inc. Compositions for blood-brain barrier transport
US8026229B2 (en) * 2001-08-13 2011-09-27 Sterix Limited Antitumor-active 2-alkoxyestradiol sulfamates
GB0306718D0 (en) * 2003-03-24 2003-04-30 Sterix Ltd Compound
EP2392258B1 (en) 2005-04-28 2014-10-08 Proteus Digital Health, Inc. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
PL3395372T3 (pl) 2009-02-20 2022-07-25 EnhanX Biopharm Inc. Układ do dostarczania leków na bazie glutationu
CN102458374A (zh) 2009-05-06 2012-05-16 实验室护肤股份有限公司 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其使用方法
CN111647037B (zh) * 2020-06-02 2021-12-07 南宁师范大学 17-酰胺雌甾类化合物及其制备方法和应用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE86393C (enExample) *
GB9118478D0 (en) * 1991-08-29 1991-10-16 Imperial College Steroid sulphatase inhibitors
US5556847A (en) * 1994-10-27 1996-09-17 Duquesne University Of The Holy Ghost Methods of effecting memory enhancement mediated by steroid sulfatase inhibitors
US5571933A (en) * 1994-11-17 1996-11-05 Duquesne University Of The Holy Ghost Derivatives of estra 1,3,5(10)triene-17-one, 3-amino compounds and their use
US5567831A (en) * 1995-08-16 1996-10-22 Duguesne University Of The Holy Ghost Non-steroidal sulfatase inhibitor compounds and their method of use

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