JP2000507588A5 - - Google Patents

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Publication number
JP2000507588A5
JP2000507588A5 JP1997535525A JP53552597A JP2000507588A5 JP 2000507588 A5 JP2000507588 A5 JP 2000507588A5 JP 1997535525 A JP1997535525 A JP 1997535525A JP 53552597 A JP53552597 A JP 53552597A JP 2000507588 A5 JP2000507588 A5 JP 2000507588A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP1997535525A
Other languages
English (en)
Japanese (ja)
Other versions
JP2000507588A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US1997/005274 external-priority patent/WO1997036580A1/en
Publication of JP2000507588A publication Critical patent/JP2000507588A/ja
Publication of JP2000507588A5 publication Critical patent/JP2000507588A5/ja
Ceased legal-status Critical Current

Links

JP9535525A 1996-03-29 1997-03-27 プロテアーゼインヒビターとしてのアミジノヒドラゾン Ceased JP2000507588A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US1431796P 1996-03-29 1996-03-29
US60/014,317 1996-03-29
PCT/US1997/005274 WO1997036580A1 (en) 1996-03-29 1997-03-27 Amidinohydrazones as protease inhibitors

Publications (2)

Publication Number Publication Date
JP2000507588A JP2000507588A (ja) 2000-06-20
JP2000507588A5 true JP2000507588A5 (enExample) 2004-12-02

Family

ID=21764747

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9535525A Ceased JP2000507588A (ja) 1996-03-29 1997-03-27 プロテアーゼインヒビターとしてのアミジノヒドラゾン

Country Status (10)

Country Link
US (1) US5891909A (enExample)
EP (1) EP0906091B1 (enExample)
JP (1) JP2000507588A (enExample)
AT (1) ATE341317T1 (enExample)
AU (1) AU722161B2 (enExample)
CA (1) CA2250426C (enExample)
DE (1) DE69736777T2 (enExample)
ES (1) ES2273365T3 (enExample)
NZ (1) NZ332073A (enExample)
WO (1) WO1997036580A1 (enExample)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW499412B (en) 1996-11-26 2002-08-21 Dimensional Pharm Inc Aminoguanidines and alkoxyguanidines as protease inhibitors
EP1036063B1 (en) 1997-11-26 2006-11-02 Ortho-McNeil Pharmaceuticals, Inc. Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
US6344486B1 (en) * 1998-04-03 2002-02-05 3-Dimensional Pharmaceuticals, Inc. Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitors
US6417161B1 (en) 1998-04-24 2002-07-09 3-Dimensional Pharmaceuticals, Inc. Amino acid amidinohydrazones, alkoxyguanidines and aminoguanidines as protease inhibitors
EA004884B1 (ru) 1998-06-11 2004-08-26 3-Дименшенл Фамэсьютикэлс, Инк. Соединения пиразинона, фармацевтическая композиция (варианты) и лекарственная форма, способ ингибирования сериновой протеазы, способ снижения тромбообразующей способности поверхности, способ лечения нарушенного протеолиза и тромбоза, связанного с различными заболеваниями, способ снижения свертывания крови у млекопитающего
FR2786181B1 (fr) * 1998-11-24 2001-10-26 Hoechst Marion Roussel Inc Nouveaux derives d'iminoguanidines, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
AU2381600A (en) 1998-12-23 2000-07-31 Du Pont Pharmaceuticals Company Thrombin or factor xa inhibitors
EP1194428B1 (en) 1999-07-09 2003-09-17 3-Dimensional Pharmaceuticals, Inc. Heteroaryl protease inhibitors and diagnostic imaging agents
DE60006407T2 (de) 1999-09-13 2004-09-09 3-Dimensional Pharmaceuticals, Inc. Azazykloalkanone serin-protease-hemmer
US6476016B2 (en) 2000-07-17 2002-11-05 3-Dimensional Pharmaceuticals, Inc. Cyclic oxyguanidine pyrazinones as protease inhibitors
CA2417914A1 (en) 2000-08-04 2002-02-14 3-Dimensional Pharmaceuticals, Inc. Cyclic oxyguanidine protease inhibitors
US6486174B2 (en) 2000-08-07 2002-11-26 3-Dimensional Pharmaceuticals, Inc. Tetrahydroisoquinoline-3-carboxylic acid alkoxyguanidines as integrin antagonists
US6589504B1 (en) 2000-09-22 2003-07-08 Pharmacia & Upjohn Company Compounds and methods for diagnosing and treating amyloid-related conditions
DK1383756T3 (da) * 2001-04-24 2008-06-23 Aryx Therapeutics Cumarinderivater til anvendelse som antikoagulanter
BR0213824A (pt) 2001-11-06 2004-08-31 Wyeth Corp Processo para a preparação de cloretos de 2-[alquil(aril)] sulfonilbenzenossulfonila e dos seus intermediários
AU2003302238A1 (en) 2002-12-03 2004-06-23 Axys Pharmaceuticals, Inc. 2-(2-hydroxybiphenyl-3-yl)-1h-benzoimidazole-5-carboxamidine derivatives as factor viia inhibitors
US20050014786A1 (en) * 2003-07-11 2005-01-20 Chongqing Sun Tetrahydroquinoline derivatives as cannabinoid receptor modulators
GB0507577D0 (en) * 2005-04-14 2005-05-18 Novartis Ag Organic compounds
US20070086958A1 (en) * 2005-10-14 2007-04-19 Medafor, Incorporated Formation of medically useful gels comprising microporous particles and methods of use
US20070087061A1 (en) * 2005-10-14 2007-04-19 Medafor, Incorporated Method and composition for creating and/or activating a platelet-rich gel by contact with a porous particulate material, for use in wound care, tissue adhesion, or as a matrix for delivery of therapeutic components
PT2724722T (pt) 2006-10-20 2017-03-14 Neurendo Pharma Llc Método de restaurar o efeito incretina
RU2354647C2 (ru) * 2007-06-28 2009-05-10 Общество С Ограниченной Ответственностью "Бионика" Новые соединения, обладающие функцией ингибиторов тромбина, и фармацевтические композиции на их основе
RU2353619C2 (ru) * 2007-06-28 2009-04-27 Общество С Ограниченной Ответственностью "Бионика" Новые соединения, обладающие функцией антикоагулянтов, фармацевтические композиции на их основе для лечения тромботических состояний и плазмозамещающий раствор для коррекции гиперкоагуляционных нарушений при гемодилюции
GB0815784D0 (en) * 2008-08-29 2008-10-08 Xention Ltd Novel potassium channel blockers
CA2824599C (en) * 2010-12-31 2020-03-10 Corridor Pharmaceuticals, Inc. Arginase inhibitors and methods of use thereof
WO2015171558A2 (en) * 2014-05-05 2015-11-12 Lycera Corporation BENZENESULFONAMIDO AND RELATED COMPOUNDS FOR USE AS AGONISTS OF RORγ AND THE TREATEMENT OF DISEASE
EP3215154B1 (en) 2014-11-07 2020-01-29 Regents of the University of Minnesota Salts and compositions useful for treating disease
CN110407721A (zh) * 2019-08-13 2019-11-05 上海毕得医药科技有限公司 一种4-氰基-3-(三氟甲基)苯-1-磺酰氯的合成方法

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3131218A (en) * 1961-02-15 1964-04-28 Smith Kline French Lab N-amino guanidine derivatives
US3271448A (en) * 1961-11-21 1966-09-06 Pfizer & Co C Phenoxyalkyl aminoguanidines
DE1263762B (de) * 1964-04-20 1968-03-21 Bayer Ag Verfahren zur Herstellung von Steroidguanylhydrazonen
BE663481A (enExample) * 1964-05-05
US3413303A (en) * 1965-09-27 1968-11-26 Ciba Geigy Corp Aralkenyloxyguanidines
FR2390954A1 (fr) * 1976-10-13 1978-12-15 Choay Sa Nouvelles guanylhydrazones, leurs procedes de preparation et medicaments les contenant
FR2549049B1 (fr) * 1983-07-13 1986-06-20 Chauvin Blache Lab Nouvelles amidines, leur procede de preparation et leur application therapeutique
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
US4727064A (en) * 1984-04-25 1988-02-23 The United States Of America As Represented By The Department Of Health And Human Services Pharmaceutical preparations containing cyclodextrin derivatives
GB8506792D0 (en) * 1985-03-15 1985-04-17 Janssen Pharmaceutica Nv Derivatives of y-cyclodextrin
US4824849A (en) * 1985-06-03 1989-04-25 Merck & Co., Inc. α2 -adrenoceptor antagonistic arylquinolizines
US5002935A (en) * 1987-12-30 1991-03-26 University Of Florida Improvements in redox systems for brain-targeted drug delivery
FR2669927B1 (fr) * 1990-11-29 1994-04-08 Adir Cie Nouveaux derives de guanidine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US5466811A (en) * 1994-07-18 1995-11-14 Merck & Co., Inc. Dioxolenylmethyl carbamates pro moieties for amine drugs

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