JP2000503321A5 - - Google Patents

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Publication number
JP2000503321A5
JP2000503321A5 JP1997526110A JP52611097A JP2000503321A5 JP 2000503321 A5 JP2000503321 A5 JP 2000503321A5 JP 1997526110 A JP1997526110 A JP 1997526110A JP 52611097 A JP52611097 A JP 52611097A JP 2000503321 A5 JP2000503321 A5 JP 2000503321A5
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JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
JP1997526110A
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English (en)
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JP2000503321A (ja
Filing date
Publication date
Priority claimed from US08/588,711 external-priority patent/US5804686A/en
Application filed filed Critical
Publication of JP2000503321A publication Critical patent/JP2000503321A/ja
Publication of JP2000503321A5 publication Critical patent/JP2000503321A5/ja
Ceased legal-status Critical Current

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Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
Figure 2000503321
JP9526110A 1996-01-19 1997-01-14 新規な融合ピロールカルボキサミド；新規な種類のｇａｂａ脳リセプタリガンド Ceased JP2000503321A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/588,711 1996-01-19
US08/588,711 US5804686A (en) 1996-01-19 1996-01-19 fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
PCT/US1997/000519 WO1997026243A1 (en) 1996-01-19 1997-01-14 Novel fused pyrrolecarboxamides; a new class of gaba brain receptor ligands

Publications (2)

Publication Number Publication Date
JP2000503321A JP2000503321A (ja) 2000-03-21
JP2000503321A5 true JP2000503321A5 (ja) 2004-11-18

Family

ID=24354983

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9526110A Ceased JP2000503321A (ja) 1996-01-19 1997-01-14 新規な融合ピロールカルボキサミド；新規な種類のｇａｂａ脳リセプタリガンド

Country Status (26)

Country Link
US (2) US5804686A (ja)
EP (1) EP1019372B1 (ja)
JP (1) JP2000503321A (ja)
KR (1) KR100490108B1 (ja)
CN (1) CN1209805A (ja)
AP (1) AP1015A (ja)
AT (1) ATE322480T1 (ja)
AU (1) AU1746697A (ja)
BG (1) BG102634A (ja)
BR (1) BR9707051A (ja)
CA (1) CA2243317C (ja)
CZ (1) CZ215498A3 (ja)
DE (1) DE69735647T2 (ja)
ES (1) ES2263170T3 (ja)
HU (1) HUP9901018A3 (ja)
IL (1) IL125391A (ja)
IS (1) IS4798A (ja)
MX (1) MX9805701A (ja)
NO (1) NO312670B1 (ja)
NZ (1) NZ330861A (ja)
OA (1) OA10811A (ja)
PL (1) PL327936A1 (ja)
RU (1) RU2167151C2 (ja)
SK (1) SK94398A3 (ja)
UA (1) UA49001C2 (ja)
WO (1) WO1997026243A1 (ja)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5750702A (en) * 1993-10-27 1998-05-12 Neurogen Corporation Certain pyrrolo pyridine-3-carboxamides; a new class of GABA brain receptor ligands
US6211365B1 (en) 1996-01-19 2001-04-03 Neurogen Corporation Fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
US5804686A (en) * 1996-01-19 1998-09-08 Neurogen Corporation fused pyrrolecarboxamides; a new class of GABA brain receptor ligands
EP0888300A1 (en) 1996-03-22 1999-01-07 Neurogen Corporation Certain fused pyrrolecarboxamides as gaba brain receptor ligands
US5723462A (en) * 1996-04-26 1998-03-03 Neurogen Corporation Certain fused pyrrolecarboxamides a new class of GABA brain receptor ligands
YU27300A (sh) * 1997-11-13 2002-10-18 Pfizer Products Inc. Postupak sinteze pirolnih amida
GT199800179A (es) * 1997-11-13 2000-05-02 Procedimiento de sintesis de pirrol amidas.
WO1999043660A1 (en) * 1998-02-26 1999-09-02 Neurogen Corporation Substituted 1,4-dihydro-4-oxonicotinic carboxamides: gaba brain receptor ligands
GB9812038D0 (en) 1998-06-04 1998-07-29 Merck Sharp & Dohme Therapeutic compound
WO2000012492A1 (en) * 1998-09-01 2000-03-09 Nissan Chemical Industries, Ltd. Benzoxazine derivatives
US20050014939A1 (en) * 1999-08-31 2005-01-20 Neurogen Corporation Fused pyrrolecarboxamides: GABA brain receptor ligands
MXPA02001709A (es) * 1999-08-31 2002-10-23 Neurogen Corp Pirrolocarboxamidas fusionadas: ligandos receptores de acido gaba-aminobutirico cerebral.
US6723332B2 (en) 2000-05-26 2004-04-20 Neurogen Corporation Oxomidazopyridine-carboxamides
WO2002020492A1 (en) * 2000-09-06 2002-03-14 Neurogen Corporation Aryl substituted tetrahydroindazoles and their use as ligands for the gaba-a receptor
US6743817B2 (en) 2000-09-06 2004-06-01 Neurogen Corporation Substituted fused pyrroleimines and pyrazoleimines
MXPA03004939A (es) * 2000-12-04 2003-09-10 Pfizer Prod Inc Sintesis de pirrolamidas.
MXPA04007606A (es) * 2002-02-07 2004-11-10 Neurogen Corp Arilamidas de acido pirazolcarboxilico fusionadas substituidas y compuestos relacionados.
JP2006502974A (ja) 2002-05-17 2006-01-26 ニューロジェン コーポレイション 置換環縮合イミダゾール誘導体：ｇａｂａａ受容体リガンド
EP2258358A3 (en) 2005-08-26 2011-09-07 Braincells, Inc. Neurogenesis with acetylcholinesterase inhibitor
EP2275095A3 (en) 2005-08-26 2011-08-17 Braincells, Inc. Neurogenesis by muscarinic receptor modulation
JP2009512711A (ja) 2005-10-21 2009-03-26 ブレインセルス，インコーポレイティド Ｐｄｅ阻害による神経新生の調節
CA2625210A1 (en) 2005-10-31 2007-05-10 Braincells, Inc. Gaba receptor mediated modulation of neurogenesis
US20100216734A1 (en) 2006-03-08 2010-08-26 Braincells, Inc. Modulation of neurogenesis by nootropic agents
AU2007249399A1 (en) 2006-05-09 2007-11-22 Braincells, Inc. Neurogenesis by modulating angiotensin
JP2009536667A (ja) 2006-05-09 2009-10-15 ブレインセルス，インコーポレイティド ５ｈｔ受容体介在性の神経新生
KR20090064418A (ko) 2006-09-08 2009-06-18 브레인셀즈 인코퍼레이션 4-아실아미노피리딘 유도체 포함 조합물
DK2074123T3 (da) 2006-10-16 2013-01-14 Bionomics Ltd Nye anxiolytiske forbindelser
US10954231B2 (en) 2006-10-16 2021-03-23 Bionomics Limited Anxiolytic compounds
WO2010099217A1 (en) 2009-02-25 2010-09-02 Braincells, Inc. Modulation of neurogenesis using d-cycloserine combinations
KR101442445B1 (ko) 2010-08-31 2014-09-22 메이지 세이카 파루마 가부시키가이샤 유해 생물 방제제
WO2012116415A1 (en) 2011-03-02 2012-09-07 Bionomics Limited Novel small-molecules as therapeutics
JP6055817B2 (ja) 2011-05-12 2016-12-27 バイオノミックス リミテッド ナフチリジンの調製方法

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3455943A (en) * 1966-10-21 1969-07-15 American Cyanamid Co Certain 5,8-dihydro-beta-carbolines
US4075343A (en) * 1976-09-13 1978-02-21 Pfizer Inc. Anti-allergenic 5-alkoxyimidazo[1,2-A]quinoline-2-carboxylic acids and derivatives thereof
DE3029980A1 (de) * 1980-08-08 1982-03-11 Boehringer Mannheim Gmbh, 6800 Mannheim Indolderivate und verfahren zu ihrer herstellung
JPS57123180A (en) * 1980-12-17 1982-07-31 Schering Ag 3-substituted beta-carboline, manufacture and psychotropic drug containing same
DE3147276A1 (de) * 1981-11-28 1983-06-09 Boehringer Mannheim Gmbh, 6800 Mannheim Verfahren zur herstellung von indolderivaten, deren verwendung als wertvolle zwischenprodukte und neue 4-hydroxyindole
DE3246932A1 (de) * 1982-12-16 1984-06-20 Schering AG, 1000 Berlin und 4709 Bergkamen Substituierte 5h-pyrimido(5,4-b)indole
DE3335323A1 (de) * 1983-09-27 1985-04-04 Schering AG, 1000 Berlin und 4709 Bergkamen Substituierte ss-carboline, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
GB8429739D0 (en) * 1984-11-24 1985-01-03 Fbc Ltd Fungicides
DE3535927A1 (de) * 1985-10-04 1987-04-09 Schering Ag 3-vinyl- und 3-ethinyl-ss-carbolinderivate, ihre herstellung und ihre verwendung als arzneimittel
CA2091986C (en) * 1990-10-09 1995-11-28 Andrew Thurkauf Certain cycloalkyl and azacycloalkyl pyrrolopyrimidines; a new class of gaba brain receptor ligands
US5243049A (en) * 1992-01-22 1993-09-07 Neurogen Corporation Certain pyrroloquinolinones: a new class of GABA brain receptor ligands
EP0626966A1 (en) * 1992-02-19 1994-12-07 PHARMACIA & UPJOHN COMPANY 3-substituted imidazo(1,5-a)quinoxalines and quinazolines with cns activity
US5266698A (en) * 1992-04-30 1993-11-30 Neurogen Corporation Certain aryl and cycloalkyl fused imidazopyrazinediones; a new class of GABA brain receptor ligands
AU6098194A (en) * 1993-01-29 1994-08-15 Ariad Pharmaceuticals, Inc. Analogs of receptor tyrosine activation motifs and therapeutic uses thereof
US5484944A (en) * 1993-10-27 1996-01-16 Neurogen Corporation Certain fused pyrrolecarboxanilides and their use as GABA brain receptor ligands
US5804686A (en) * 1996-01-19 1998-09-08 Neurogen Corporation fused pyrrolecarboxamides; a new class of GABA brain receptor ligands

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