JP2000502105A5 - - Google Patents

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Publication number
JP2000502105A5
JP2000502105A5 JP1997523095A JP52309597A JP2000502105A5 JP 2000502105 A5 JP2000502105 A5 JP 2000502105A5 JP 1997523095 A JP1997523095 A JP 1997523095A JP 52309597 A JP52309597 A JP 52309597A JP 2000502105 A5 JP2000502105 A5 JP 2000502105A5
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP1997523095A
Other languages
English (en)
Japanese (ja)
Other versions
JP2000502105A (ja
JP4865113B2 (ja
Filing date
Publication date
Priority claimed from US08/575,344 external-priority patent/US6201124B1/en
Application filed filed Critical
Publication of JP2000502105A publication Critical patent/JP2000502105A/ja
Publication of JP2000502105A5 publication Critical patent/JP2000502105A5/ja
Application granted granted Critical
Publication of JP4865113B2 publication Critical patent/JP4865113B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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JP52309597A 1995-12-21 1996-12-19 ピペリジン誘導体の製法 Expired - Lifetime JP4865113B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/575,344 1995-12-21
US08/575,344 US6201124B1 (en) 1995-12-21 1995-12-21 Process for production of piperidine derivatives
PCT/US1996/020769 WO1997022344A1 (en) 1995-12-21 1996-12-19 Process for production of piperidine derivatives

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2008227513A Division JP2009019059A (ja) 1995-12-21 2008-09-04 ピペリジン誘導体の製法

Publications (3)

Publication Number Publication Date
JP2000502105A JP2000502105A (ja) 2000-02-22
JP2000502105A5 true JP2000502105A5 (cg-RX-API-DMAC7.html) 2004-11-04
JP4865113B2 JP4865113B2 (ja) 2012-02-01

Family

ID=24299941

Family Applications (2)

Application Number Title Priority Date Filing Date
JP52309597A Expired - Lifetime JP4865113B2 (ja) 1995-12-21 1996-12-19 ピペリジン誘導体の製法
JP2008227513A Pending JP2009019059A (ja) 1995-12-21 2008-09-04 ピペリジン誘導体の製法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2008227513A Pending JP2009019059A (ja) 1995-12-21 2008-09-04 ピペリジン誘導体の製法

Country Status (16)

Country Link
US (7) US6201124B1 (cg-RX-API-DMAC7.html)
EP (2) EP0877733B1 (cg-RX-API-DMAC7.html)
JP (2) JP4865113B2 (cg-RX-API-DMAC7.html)
KR (2) KR100591212B1 (cg-RX-API-DMAC7.html)
AT (1) ATE335726T1 (cg-RX-API-DMAC7.html)
AU (1) AU723759B2 (cg-RX-API-DMAC7.html)
BR (1) BR9612099A (cg-RX-API-DMAC7.html)
CA (1) CA2240735C (cg-RX-API-DMAC7.html)
DE (1) DE69636439T2 (cg-RX-API-DMAC7.html)
DK (1) DK0877733T3 (cg-RX-API-DMAC7.html)
ES (1) ES2268715T3 (cg-RX-API-DMAC7.html)
HU (1) HUP9900947A3 (cg-RX-API-DMAC7.html)
NO (1) NO311718B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ326228A (cg-RX-API-DMAC7.html)
PT (1) PT877733E (cg-RX-API-DMAC7.html)
WO (1) WO1997022344A1 (cg-RX-API-DMAC7.html)

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HU226037B1 (en) * 1993-06-25 2008-03-28 Aventis Inc Process for producing antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives and novel intermediates
US6153754A (en) * 1995-12-21 2000-11-28 Albany Molecular Research, Inc. Process for production of piperidine derivatives
US6201124B1 (en) * 1995-12-21 2001-03-13 Albany Molecular Research, Inc. Process for production of piperidine derivatives
ES2151442B1 (es) * 1999-01-11 2001-07-01 Espanola Prod Quimicos Nuevo derivado del bencenoetanol.
US20030021849A1 (en) * 2001-04-09 2003-01-30 Ben-Zion Dolitzky Polymorphs of fexofenadine hydrochloride
KR20040012747A (ko) * 2001-04-09 2004-02-11 테바 파마슈티컬 인더스트리즈 리미티드 펙소페나딘 염산염의 다형체
ITRM20010260A1 (it) 2001-05-17 2002-11-18 Dinamite Dipharma S P A In For Processo per la preparazione della fexofenadina o acido 4 1-idrossi-4-4- (idrossidifenilmetil)-1-piperidinil|-butil|-alfa,alfa-dimetilbenz
EP1453509A2 (en) * 2001-11-08 2004-09-08 Teva Pharmaceutical Industries Ltd. Polymorphs of fexofenadine base
JP2005532356A (ja) * 2002-06-10 2005-10-27 テバ ファーマシューティカル インダストリーズ リミティド 塩酸フェキソフェナジンの多型体ｘｖｉ
US6949765B2 (en) 2002-11-05 2005-09-27 Chartered Semiconductor Manufacturing Ltd. Padless structure design for easy identification of bridging defects in lines by passive voltage contrast
TW200517114A (en) 2003-10-15 2005-06-01 Combinatorx Inc Methods and reagents for the treatment of immunoinflammatory disorders
EP1628959A2 (en) * 2004-04-26 2006-03-01 Teva Pharmaceutical Industries Ltd Crystalline forms of fexofenadine hydrochloride and processes for their preparation
US7498443B2 (en) * 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of carebastine
US7498345B2 (en) 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of piperidine derivatives
WO2006037042A1 (en) * 2004-09-28 2006-04-06 Teva Pharmaceutical Industries Ltd. Fexofenadine crystal form and processes for its preparation thereof
RU2008122978A (ru) 2005-11-09 2009-12-20 Комбинаторкс, Инкорпорейтед (Us) Способы, композиции и наборы для лечения медицинских состояний
CN100443470C (zh) * 2006-07-21 2008-12-17 杭州保灵有限公司 一种依巴斯汀的制备方法
ITMI20061492A1 (it) * 2006-07-27 2008-01-28 Archimica Srl Processo per la preparazione di fexofenadina.
ITMI20061491A1 (it) * 2006-07-27 2008-01-28 Archimica Srl Processo per la preparazione di fexofenadina.
ITMI20070987A1 (it) 2007-05-16 2008-11-17 Dipharma Francis Srl Procedimento per la preparazione di composti chetonici
US20100092479A1 (en) * 2008-08-18 2010-04-15 Combinatorx (Singapore) Pte. Ltd. Compositions and methods for treatment of viral diseases
US20110130711A1 (en) * 2009-11-19 2011-06-02 Follica, Inc. Hair growth treatment
EP2371817A1 (en) * 2010-04-01 2011-10-05 Arevipharma GmbH Process for the preparation of 1-[4-(1,1-dimethylethyl)phenyl]-4-[4-(diphenylmethoxy)-1-piperidinyl]-1-butanone and acid addition salts thereof
CN105254579A (zh) * 2015-09-19 2016-01-20 万全万特制药江苏有限公司 一种一锅法制备比拉斯汀中间体的方法
CN114621083A (zh) * 2022-03-30 2022-06-14 西安万隆制药股份有限公司 一种抗组胺药物盐酸非索非那定杂质及其合成方法和应用
CN114671802B (zh) * 2022-04-14 2024-05-17 江苏联环药业股份有限公司 一种高纯度依巴斯汀的制备方法
EP4647423A1 (en) * 2023-01-03 2025-11-12 Chengdu Shibeikang Biomedical Technology Co., Ltd. Crystal form and amorphous form of carebastine p-toluenesulfonate

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US4028404A (en) 1967-07-31 1977-06-07 Allen & Hanburys Limited Acetic acid derivatives
GB1242169A (en) 1969-04-09 1971-08-11 Ucb Sa Piperidine derivatives
US3839431A (en) 1970-07-13 1974-10-01 Squibb & Sons Inc Cyclopropylmethylphenylacetic acids and derivatives
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GB8321157D0 (en) 1983-08-05 1983-09-07 Fordonal Sa Piperidine derivatives
US4742175A (en) 1986-05-07 1988-05-03 Merrell Dow Pharmaceuticals Inc. Preparation of polymorphically pure terfenadine
US5382600A (en) 1988-01-22 1995-01-17 Pharmacia Aktiebolag 3,3-diphenylpropylamines and pharmaceutical compositions thereof
FR2636946B1 (fr) 1988-09-23 1990-11-02 Lipha ((diarylmethoxy)alcoyl)-1 pyrrolidines et piperidines, procedes de preparation et medicaments les contenant
DE4034218A1 (de) 1990-10-27 1992-04-30 Merck Patent Gmbh Verfahren zur herstellung von carebastin
HU211019B (en) 1991-12-02 1995-09-28 Richter Gedeon Vegyeszet Process for producing new 1,2,3,6-tetrahydropyridine and piperidine derivatives substituted with n-(hydroxylalkyl) group and compositions comprising such compounds
JP3686950B2 (ja) 1992-04-10 2005-08-24 メレル ファーマスーティカルズ インコーポレイテッド ピペリジン誘導体類の新規な方法
CA2141572C (en) 1992-08-03 2001-02-06 James W. Young Terfenadine metabolites and their optically pure isomers for treating allergic disorders
KR100387348B1 (ko) * 1993-06-24 2003-06-12 알바니 몰레큘라 리써치, 인크. 피페리딘 유도체의 제조 방법
US20020007068A1 (en) * 1999-07-16 2002-01-17 D'ambra Thomas E. Piperidine derivatives and process for their production
HU226037B1 (en) * 1993-06-25 2008-03-28 Aventis Inc Process for producing antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives and novel intermediates
US6201124B1 (en) * 1995-12-21 2001-03-13 Albany Molecular Research, Inc. Process for production of piperidine derivatives
US6153754A (en) * 1995-12-21 2000-11-28 Albany Molecular Research, Inc. Process for production of piperidine derivatives
US5925761A (en) * 1997-02-04 1999-07-20 Sepracor Inc. Synthesis of terfenadine and derivatives
US7498345B2 (en) * 2004-09-17 2009-03-03 Albany Molecular Research, Inc. Process for production of piperidine derivatives

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