JOP20220202A1 - تركيبة صيدلانية تشمل مركب مشتق من بنزيميدازول - Google Patents
تركيبة صيدلانية تشمل مركب مشتق من بنزيميدازولInfo
- Publication number
- JOP20220202A1 JOP20220202A1 JOP/2022/0202A JOP20220202A JOP20220202A1 JO P20220202 A1 JOP20220202 A1 JO P20220202A1 JO P20220202 A JOP20220202 A JO P20220202A JO P20220202 A1 JOP20220202 A1 JO P20220202A1
- Authority
- JO
- Jordan
- Prior art keywords
- derivative compound
- benzimidazole derivative
- pharmaceutical composition
- present disclosure
- disclosure relates
- Prior art date
Links
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
- A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
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- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
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- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Inorganic Chemistry (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
يتعلق الكشف الحالي بتركيبة صيدلانية تحتوي على مركب مشتق من البنزيميدازول. بصفة خاصة، يتعلق الكشف الحالي بصياغة قادرة على الحفاظ على تركيز مستدام لمركب مشتق من البنزيميدازول في الدم.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20200024657 | 2020-02-27 | ||
KR20200043047 | 2020-04-08 | ||
PCT/IB2021/051609 WO2021171239A1 (en) | 2020-02-27 | 2021-02-26 | Pharmaceutical composition comprising benzimidazole derivative compound |
Publications (1)
Publication Number | Publication Date |
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JOP20220202A1 true JOP20220202A1 (ar) | 2023-01-30 |
Family
ID=77490743
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JOP/2022/0202A JOP20220202A1 (ar) | 2020-02-27 | 2021-02-26 | تركيبة صيدلانية تشمل مركب مشتق من بنزيميدازول |
Country Status (13)
Country | Link |
---|---|
US (2) | US20230087865A1 (ar) |
EP (2) | EP4110301A4 (ar) |
JP (2) | JP2023517844A (ar) |
KR (2) | KR102667902B1 (ar) |
CN (2) | CN115175669A (ar) |
AU (1) | AU2021225484A1 (ar) |
BR (1) | BR112022017017A2 (ar) |
CA (2) | CA3169318A1 (ar) |
JO (1) | JOP20220202A1 (ar) |
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WO2023182332A1 (ja) * | 2022-03-22 | 2023-09-28 | 株式会社ダイセル | 口腔内崩壊錠用の添加剤組成物 |
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US5945124A (en) * | 1995-07-05 | 1999-08-31 | Byk Gulden Chemische Fabrik Gmbh | Oral pharmaceutical composition with delayed release of active ingredient for pantoprazole |
KR100504013B1 (ko) * | 2003-02-28 | 2005-07-28 | 한국유나이티드제약 주식회사 | 제어방출형 경구 펠렛제제 및 그 제조방법 |
KR100762846B1 (ko) * | 2003-09-29 | 2007-10-04 | 씨제이 주식회사 | 서방성 제제 |
US20070122480A1 (en) * | 2003-09-29 | 2007-05-31 | Cj Corporation | Sustained release formulations |
JP4481344B2 (ja) * | 2005-12-19 | 2010-06-16 | ラクオリア創薬株式会社 | クロマン置換ベンゾイミダゾール誘導体及び酸ポンプ阻害剤としてのそれらの使用 |
ZA200806496B (en) * | 2006-01-27 | 2009-12-30 | Eurand Inc | Drug delivery systems comprising weakly basic drugs and organic acids |
KR101784001B1 (ko) | 2006-04-04 | 2017-10-23 | 케이지 액퀴지션 엘엘씨 | 항혈소판제와 산 억제제를 포함하는 경구 투여용 약학 조성물 |
US9532945B2 (en) * | 2006-04-04 | 2017-01-03 | Kg Acquisition Llc | Oral dosage forms including an antiplatelet agent and an enterically coated acid inhibitor |
EP2255797A4 (en) * | 2008-02-22 | 2011-09-07 | Hanall Biopharma Co Ltd | COMPOSITE PREPARATION |
GB201003731D0 (en) * | 2010-03-05 | 2010-04-21 | Univ Strathclyde | Immediate/delayed drug delivery |
AU2011325371A1 (en) * | 2010-10-21 | 2013-05-02 | Galderma S.A. | Sustained-release tablet and process for preparing the same |
EP2755641A4 (en) | 2011-09-14 | 2015-03-18 | Pozen Inc | CONTROLLED DOSAGE OF CLOPIDOGREL IN MAGIC ACID INHIBITION THERAPIES |
KR101675501B1 (ko) * | 2011-11-02 | 2016-11-14 | 한국유나이티드제약 주식회사 | 클로피도그렐 및 아스피린의 복합제제 |
KR20140101391A (ko) * | 2011-12-09 | 2014-08-19 | 욱크하르트 리미티드 | 심혈관 질환의 치료 방법 |
KR102241487B1 (ko) * | 2013-02-20 | 2021-04-16 | 주식회사 종근당 | 제어방출 펠릿으로 된 약제학적 조성물 |
MX2017015926A (es) * | 2015-06-08 | 2018-07-06 | Cj Healthcare Corp | Uso de derivados de bencimidazol para escape acido nocturno. |
EP3329921B1 (en) * | 2015-07-30 | 2024-03-27 | Takeda Pharmaceutical Company Limited | Tablet |
CN105030725B (zh) * | 2015-08-26 | 2019-12-10 | 迪沙药业集团有限公司 | 一种富马酸沃诺拉赞肠溶组合物及其制备方法 |
CN107224438B (zh) * | 2016-03-25 | 2021-04-06 | 江苏豪森药业集团有限公司 | 富马酸沃诺拉赞药物组合物 |
JOP20190198A1 (ar) | 2018-08-28 | 2020-02-28 | Hk Inno N Corp | تركيبة صيدلانية تشتمل على عامل مضاد للصفيحات ومثبط إفراز حمض معدي |
CN109320485B (zh) * | 2018-12-02 | 2021-06-18 | 江苏慧聚药业有限公司 | 合成特戈拉赞手性醇的方法 |
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TWI821638B (zh) | 2023-11-11 |
CN115175669A (zh) | 2022-10-11 |
US20230087865A1 (en) | 2023-03-23 |
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UY39094A (es) | 2021-07-30 |
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CN115209875A (zh) | 2022-10-18 |
JP2023517844A (ja) | 2023-04-27 |
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CA3169318A1 (en) | 2021-09-02 |
JP7493048B2 (ja) | 2024-05-30 |
EP4110301A1 (en) | 2023-01-04 |
KR102667902B1 (ko) | 2024-05-21 |
JP2023514786A (ja) | 2023-04-10 |
EP4110301A4 (en) | 2023-11-15 |
BR112022017017A2 (pt) | 2022-10-11 |
WO2021171239A1 (en) | 2021-09-02 |
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