MX2023007265A - Inhibidores de cdk y su uso como productos farmacéuticos. - Google Patents
Inhibidores de cdk y su uso como productos farmacéuticos.Info
- Publication number
- MX2023007265A MX2023007265A MX2023007265A MX2023007265A MX2023007265A MX 2023007265 A MX2023007265 A MX 2023007265A MX 2023007265 A MX2023007265 A MX 2023007265A MX 2023007265 A MX2023007265 A MX 2023007265A MX 2023007265 A MX2023007265 A MX 2023007265A
- Authority
- MX
- Mexico
- Prior art keywords
- pharmaceuticals
- cdk inhibitors
- compounds
- formula
- cdk
- Prior art date
Links
- 229940043378 cyclin-dependent kinase inhibitor Drugs 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La descripción se dirige a compuestos de la Fórmula (I), también se describen composiciones farmacéuticas que comprenden compuestos de la Fórmula (I), así como métodos para su uso y preparación. (ver fórmula I).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202063127853P | 2020-12-18 | 2020-12-18 | |
PCT/US2021/064037 WO2022133215A1 (en) | 2020-12-18 | 2021-12-17 | Cdk inhibitors and their use as pharmaceuticals |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2023007265A true MX2023007265A (es) | 2023-08-14 |
Family
ID=80050584
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2023007265A MX2023007265A (es) | 2020-12-18 | 2021-12-17 | Inhibidores de cdk y su uso como productos farmacéuticos. |
Country Status (10)
Country | Link |
---|---|
US (1) | US20220267345A1 (es) |
EP (1) | EP4263525A1 (es) |
JP (1) | JP2023554643A (es) |
KR (1) | KR20230122096A (es) |
CN (1) | CN116940563A (es) |
AU (1) | AU2021401403A1 (es) |
CA (1) | CA3205652A1 (es) |
IL (1) | IL303779A (es) |
MX (1) | MX2023007265A (es) |
WO (1) | WO2022133215A1 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR112022004327A2 (pt) * | 2019-09-11 | 2022-05-31 | Prelude Therapeutics Inc | Inibidores de cdk e seu uso como fármacos |
US20230257394A1 (en) * | 2022-02-03 | 2023-08-17 | Prelude Therapeutics, Incorporated | CDK Inhibitors And Their Use As Pharmaceuticals |
WO2024035771A2 (en) * | 2022-08-09 | 2024-02-15 | H. Lee Moffitt Cancer Center And Research Institute, Inc. | Ulk3 inhibitors and uses thereof |
WO2024051717A1 (zh) * | 2022-09-08 | 2024-03-14 | 上海深势唯思科技有限责任公司 | 作为plk1抑制剂的化合物及其制备方法和用途 |
CN115594664B (zh) * | 2022-11-25 | 2023-02-24 | 英矽智能科技(上海)有限公司 | 一类螺环衍生物作为kif18a抑制剂 |
Family Cites Families (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3657744A (en) | 1970-05-08 | 1972-04-25 | Univ Minnesota | Method for fixing prosthetic implants in a living body |
US4733665C2 (en) | 1985-11-07 | 2002-01-29 | Expandable Grafts Partnership | Expandable intraluminal graft and method and apparatus for implanting an expandable intraluminal graft |
US5023252A (en) | 1985-12-04 | 1991-06-11 | Conrex Pharmaceutical Corporation | Transdermal and trans-membrane delivery of drugs |
US5061273A (en) | 1989-06-01 | 1991-10-29 | Yock Paul G | Angioplasty apparatus facilitating rapid exchanges |
US5040548A (en) | 1989-06-01 | 1991-08-20 | Yock Paul G | Angioplasty mehtod |
US5350395A (en) | 1986-04-15 | 1994-09-27 | Yock Paul G | Angioplasty apparatus facilitating rapid exchanges |
US4748982A (en) | 1987-01-06 | 1988-06-07 | Advanced Cardiovascular Systems, Inc. | Reinforced balloon dilatation catheter with slitted exchange sleeve and method |
US4992445A (en) | 1987-06-12 | 1991-02-12 | American Cyanamid Co. | Transdermal delivery of pharmaceuticals |
US5001139A (en) | 1987-06-12 | 1991-03-19 | American Cyanamid Company | Enchancers for the transdermal flux of nivadipine |
CA1322628C (en) | 1988-10-04 | 1993-10-05 | Richard A. Schatz | Expandable intraluminal graft |
US5674278A (en) | 1989-08-24 | 1997-10-07 | Arterial Vascular Engineering, Inc. | Endovascular support device |
US6344053B1 (en) | 1993-12-22 | 2002-02-05 | Medtronic Ave, Inc. | Endovascular support device and method |
US5292331A (en) | 1989-08-24 | 1994-03-08 | Applied Vascular Engineering, Inc. | Endovascular support device |
ES2389673T3 (es) * | 2007-09-28 | 2012-10-30 | Nerviano Medical Sciences S.R.L. | Derivados de pirrolopirimidina sustituidos, procedimiento para su preparación y su uso como inhibidores de quinasas |
CN106810536A (zh) * | 2015-11-30 | 2017-06-09 | 甘李药业股份有限公司 | 一种蛋白激酶抑制剂及其制备方法和医药用途 |
DK3665179T3 (da) | 2017-08-09 | 2021-08-16 | Prelude Therapeutics Inc | Selektive inhibitorer af proteinargininmethyltransferase 5 (prmt5) |
US10711007B2 (en) | 2018-03-14 | 2020-07-14 | Prelude Therapeutics Incorporated | Selective inhibitors of protein arginine methyltransferase 5 (PRMT5) |
CN113661164A (zh) * | 2019-04-08 | 2021-11-16 | 珠海宇繁生物科技有限责任公司 | 一种cdk激酶抑制剂及其应用 |
US20240092799A1 (en) * | 2020-08-20 | 2024-03-21 | Hepagene Therapeutics (HK) Limited | Mnk inhibitors |
-
2021
- 2021-12-17 CN CN202180092828.2A patent/CN116940563A/zh active Pending
- 2021-12-17 KR KR1020237024366A patent/KR20230122096A/ko unknown
- 2021-12-17 EP EP21848359.2A patent/EP4263525A1/en active Pending
- 2021-12-17 AU AU2021401403A patent/AU2021401403A1/en active Pending
- 2021-12-17 IL IL303779A patent/IL303779A/en unknown
- 2021-12-17 WO PCT/US2021/064037 patent/WO2022133215A1/en active Application Filing
- 2021-12-17 CA CA3205652A patent/CA3205652A1/en active Pending
- 2021-12-17 JP JP2023537129A patent/JP2023554643A/ja active Pending
- 2021-12-17 MX MX2023007265A patent/MX2023007265A/es unknown
- 2021-12-17 US US17/554,284 patent/US20220267345A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
JP2023554643A (ja) | 2023-12-28 |
KR20230122096A (ko) | 2023-08-22 |
WO2022133215A1 (en) | 2022-06-23 |
CA3205652A1 (en) | 2022-06-23 |
US20220267345A1 (en) | 2022-08-25 |
AU2021401403A1 (en) | 2023-07-13 |
IL303779A (en) | 2023-08-01 |
EP4263525A1 (en) | 2023-10-25 |
CN116940563A (zh) | 2023-10-24 |
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