IT8621112A0 - Derivati dell'acido tiazolidin-4-carbossilico adattivita' farmaceutica. - Google Patents

Derivati dell'acido tiazolidin-4-carbossilico adattivita' farmaceutica.

Info

Publication number
IT8621112A0
IT8621112A0 IT8621112A IT2111286A IT8621112A0 IT 8621112 A0 IT8621112 A0 IT 8621112A0 IT 8621112 A IT8621112 A IT 8621112A IT 2111286 A IT2111286 A IT 2111286A IT 8621112 A0 IT8621112 A0 IT 8621112A0
Authority
IT
Italy
Prior art keywords
adaptivity
thiazolidin
derivatives
carboxylic acid
acid pharmaceutical
Prior art date
Application number
IT8621112A
Other languages
English (en)
Other versions
IT1196485B (it
IT8621112A1 (it
Inventor
Franco Pellacini
Davide Della Bella
Angelo Carenzi
Dario Chiarino
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of IT8621112A0 publication Critical patent/IT8621112A0/it
Priority to IT21112/86A priority Critical patent/IT1196485B/it
Priority to EP87201313A priority patent/EP0254354B1/en
Priority to DE8787201313T priority patent/DE3785104T2/de
Priority to AT87201313T priority patent/ATE87622T1/de
Priority to ES87201313T priority patent/ES2054654T3/es
Priority to IE187287A priority patent/IE60205B1/en
Priority to ZA875099A priority patent/ZA875099B/xx
Priority to AU75566/87A priority patent/AU609406B2/en
Priority to US07/072,569 priority patent/US4840936A/en
Priority to JP62175776A priority patent/JP2603639B2/ja
Priority to CA000541971A priority patent/CA1322074C/en
Publication of IT8621112A1 publication Critical patent/IT8621112A1/it
Application granted granted Critical
Publication of IT1196485B publication Critical patent/IT1196485B/it

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT21112/86A 1986-07-14 1986-07-14 Derivati dell'acido tiazolidin-4-carbossilico ad attivita' farmaceutica IT1196485B (it)

Priority Applications (11)

Application Number Priority Date Filing Date Title
IT21112/86A IT1196485B (it) 1986-07-14 1986-07-14 Derivati dell'acido tiazolidin-4-carbossilico ad attivita' farmaceutica
EP87201313A EP0254354B1 (en) 1986-07-14 1987-07-09 Pharmaceutically useful derivatives of thiazolidine-4-carboxylic acid
DE8787201313T DE3785104T2 (de) 1986-07-14 1987-07-09 Pharmazeutisch nuetzliche thiazolidin-4-karbonsaeure-derivate.
AT87201313T ATE87622T1 (de) 1986-07-14 1987-07-09 Pharmazeutisch nuetzliche thiazolidin-4karbons|ure-derivate.
ES87201313T ES2054654T3 (es) 1986-07-14 1987-07-09 Derivados farmaceuticamente utiles de acido tiazolidina-4-carboxilico.
IE187287A IE60205B1 (en) 1986-07-14 1987-07-10 Pharmaceutically useful derivatives of thiazolidine-4-carboxylic acid
ZA875099A ZA875099B (en) 1986-07-14 1987-07-13 Pharmaceutically useful derivatives of thiazolidine-4-carboxylic acid
AU75566/87A AU609406B2 (en) 1986-07-14 1987-07-13 Pharmaceutically useful derivatives of thiazolidine-4-carboxylic acid
US07/072,569 US4840936A (en) 1986-07-14 1987-07-13 Pharmaceutically useful derivatives of thiazolidine-4-carboxylic acid
JP62175776A JP2603639B2 (ja) 1986-07-14 1987-07-14 チアゾリジン―４―カルボン酸化合物、その製造方法、この化合物を含有する解熱消炎鎮痛剤および虚血・リパーフュージョン症候群治療薬
CA000541971A CA1322074C (en) 1986-07-14 1987-07-14 Pharmaceutically useful derivatives of thiazolidine-4- carboxylic acid

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT21112/86A IT1196485B (it) 1986-07-14 1986-07-14 Derivati dell'acido tiazolidin-4-carbossilico ad attivita' farmaceutica

Publications (3)

Publication Number Publication Date
IT8621112A0 true IT8621112A0 (it) 1986-07-14
IT8621112A1 IT8621112A1 (it) 1988-01-14
IT1196485B IT1196485B (it) 1988-11-16

Family

ID=11176919

Family Applications (1)

Application Number Title Priority Date Filing Date
IT21112/86A IT1196485B (it) 1986-07-14 1986-07-14 Derivati dell'acido tiazolidin-4-carbossilico ad attivita' farmaceutica

Country Status (11)

Country Link
US (1) US4840936A (it)
EP (1) EP0254354B1 (it)
JP (1) JP2603639B2 (it)
AT (1) ATE87622T1 (it)
AU (1) AU609406B2 (it)
CA (1) CA1322074C (it)
DE (1) DE3785104T2 (it)
ES (1) ES2054654T3 (it)
IE (1) IE60205B1 (it)
IT (1) IT1196485B (it)
ZA (1) ZA875099B (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1030415A (zh) * 1987-02-20 1989-01-18 山之内制药株式会社 饱和的杂环碳酰胺衍生物和它的制备方法
IT1223565B (it) * 1987-12-21 1990-09-19 Zambon Spa Derivati dell'acido tiazolidin 4 carbossilico ad attivita' farmaceutica
DE3818850A1 (de) * 1988-06-03 1989-12-07 Hoechst Ag Oligopeptide mit zyklischen prolin-analogen aminosaeuren
IT1230706B (it) * 1989-02-10 1991-10-29 Poli Ind Chimica Spa Derivati dell'acido 3 piroglutamoil tiazolidin 4 carbossilico e loro proprieta' farmacologiche.
IT1250736B (it) * 1991-08-01 1995-04-21 Zambon Spa Processo per la preparazione dell'acido 5-(2',4'-difluorofenil) salicilico in forma ii pura
DE19711052C2 (de) 1997-03-03 1999-09-23 Hans Rommelspacher Verwendung von 2-Methyl-thiazolidin-2,4-dicarbonsäure als Mukolytikum
KR20010025470A (ko) * 2000-12-29 2001-04-06 강덕영 치아졸리딘-4-카르복실산 염의 제조방법
EP1479762B1 (en) 2002-02-28 2011-09-28 Mitsubishi Chemical Corporation Novel dehydrogenase and gene encoding the same
WO2023003497A1 (ru) * 2021-07-23 2023-01-26 Общество С Ограниченной Ответственностью "Валента-Интеллект" Соединения с лизосомотропной и противовирусной активностью

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2210230A1 (de) * 1972-03-03 1973-09-06 Kolmar Laboratories Verwendung bestimmter thioaether als antimikrobielle und zytostatische mittel
AU528115B2 (en) * 1978-04-08 1983-04-14 Santen Pharmaceutical Co. Ltd. Antihypertensive 4-thiazolidine/carboxylic acids
DE3002989A1 (de) * 1980-01-29 1981-07-30 Hoechst Ag, 6000 Frankfurt Hydroxyphenyl-thiazol, -thiazolin und -thiazolidin-carbonsaeuren, verfahren zu ihrer herstellung und ihre verwendung zur beeinflussung des kollagenstoffwechsels
HU195492B (en) * 1984-07-27 1988-05-30 Boehringer Biochemia Srl Process for producing 2-substituted thiazolidine derivatives with antitussive and mucus regulating action and pharmaceuticals comprising these compounds as active ingredient
IT1176983B (it) * 1984-10-16 1987-08-26 Zambon Spa Dipeptidi ad attivita' farmacologica

Also Published As

Publication number Publication date
EP0254354A1 (en) 1988-01-27
ATE87622T1 (de) 1993-04-15
IE871872L (en) 1988-01-14
US4840936A (en) 1989-06-20
AU609406B2 (en) 1991-05-02
EP0254354B1 (en) 1993-03-31
DE3785104T2 (de) 1993-09-02
AU7556687A (en) 1988-01-21
JPS6323876A (ja) 1988-02-01
JP2603639B2 (ja) 1997-04-23
DE3785104D1 (de) 1993-05-06
IE60205B1 (en) 1994-06-15
ZA875099B (en) 1988-04-27
CA1322074C (en) 1993-09-07
ES2054654T3 (es) 1994-08-16
IT1196485B (it) 1988-11-16
IT8621112A1 (it) 1988-01-14

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