ATE87622T1 - Pharmazeutisch nuetzliche thiazolidin-4karbons|ure-derivate. - Google Patents
Pharmazeutisch nuetzliche thiazolidin-4karbons|ure-derivate.Info
- Publication number
- ATE87622T1 ATE87622T1 AT87201313T AT87201313T ATE87622T1 AT E87622 T1 ATE87622 T1 AT E87622T1 AT 87201313 T AT87201313 T AT 87201313T AT 87201313 T AT87201313 T AT 87201313T AT E87622 T1 ATE87622 T1 AT E87622T1
- Authority
- AT
- Austria
- Prior art keywords
- 4carbons
- thiazolidin
- ure
- derivatives
- compounds
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 150000001299 aldehydes Chemical class 0.000 abstract 1
- 230000000202 analgesic effect Effects 0.000 abstract 1
- 230000003110 anti-inflammatory effect Effects 0.000 abstract 1
- 230000001754 anti-pyretic effect Effects 0.000 abstract 1
- 239000002221 antipyretic Substances 0.000 abstract 1
- XUJNEKJLAYXESH-UHFFFAOYSA-N cysteine Natural products SCC(N)C(O)=O XUJNEKJLAYXESH-UHFFFAOYSA-N 0.000 abstract 1
- 235000018417 cysteine Nutrition 0.000 abstract 1
- 230000006378 damage Effects 0.000 abstract 1
- 230000002496 gastric effect Effects 0.000 abstract 1
- 208000028867 ischemia Diseases 0.000 abstract 1
- 150000002576 ketones Chemical class 0.000 abstract 1
- 230000000510 mucolytic effect Effects 0.000 abstract 1
- 230000010410 reperfusion Effects 0.000 abstract 1
- 208000011580 syndromic disease Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D277/06—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biomedical Technology (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT21112/86A IT1196485B (it) | 1986-07-14 | 1986-07-14 | Derivati dell'acido tiazolidin-4-carbossilico ad attivita' farmaceutica |
| EP87201313A EP0254354B1 (de) | 1986-07-14 | 1987-07-09 | Pharmazeutisch nützliche Thiazolidin-4-Karbonsäure-Derivate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE87622T1 true ATE87622T1 (de) | 1993-04-15 |
Family
ID=11176919
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT87201313T ATE87622T1 (de) | 1986-07-14 | 1987-07-09 | Pharmazeutisch nuetzliche thiazolidin-4karbons|ure-derivate. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US4840936A (de) |
| EP (1) | EP0254354B1 (de) |
| JP (1) | JP2603639B2 (de) |
| AT (1) | ATE87622T1 (de) |
| AU (1) | AU609406B2 (de) |
| CA (1) | CA1322074C (de) |
| DE (1) | DE3785104T2 (de) |
| ES (1) | ES2054654T3 (de) |
| IE (1) | IE60205B1 (de) |
| IT (1) | IT1196485B (de) |
| ZA (1) | ZA875099B (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1030415A (zh) * | 1987-02-20 | 1989-01-18 | 山之内制药株式会社 | 饱和的杂环碳酰胺衍生物和它的制备方法 |
| IT1223565B (it) * | 1987-12-21 | 1990-09-19 | Zambon Spa | Derivati dell'acido tiazolidin 4 carbossilico ad attivita' farmaceutica |
| DE3818850A1 (de) * | 1988-06-03 | 1989-12-07 | Hoechst Ag | Oligopeptide mit zyklischen prolin-analogen aminosaeuren |
| IT1230706B (it) * | 1989-02-10 | 1991-10-29 | Poli Ind Chimica Spa | Derivati dell'acido 3 piroglutamoil tiazolidin 4 carbossilico e loro proprieta' farmacologiche. |
| IT1250736B (it) * | 1991-08-01 | 1995-04-21 | Zambon Spa | Processo per la preparazione dell'acido 5-(2',4'-difluorofenil) salicilico in forma ii pura |
| DE19711052C2 (de) * | 1997-03-03 | 1999-09-23 | Hans Rommelspacher | Verwendung von 2-Methyl-thiazolidin-2,4-dicarbonsäure als Mukolytikum |
| KR20010025470A (ko) * | 2000-12-29 | 2001-04-06 | 강덕영 | 치아졸리딘-4-카르복실산 염의 제조방법 |
| AU2003211367A1 (en) | 2002-02-28 | 2003-09-09 | Mitsubishi Chemical Corporation | Novel dehydrogenase and gene encoding the same |
| WO2023003497A1 (ru) * | 2021-07-23 | 2023-01-26 | Общество С Ограниченной Ответственностью "Валента-Интеллект" | Соединения с лизосомотропной и противовирусной активностью |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2210230A1 (de) * | 1972-03-03 | 1973-09-06 | Kolmar Laboratories | Verwendung bestimmter thioaether als antimikrobielle und zytostatische mittel |
| AU528115B2 (en) * | 1978-04-08 | 1983-04-14 | Santen Pharmaceutical Co. Ltd. | Antihypertensive 4-thiazolidine/carboxylic acids |
| DE3002989A1 (de) * | 1980-01-29 | 1981-07-30 | Hoechst Ag, 6000 Frankfurt | Hydroxyphenyl-thiazol, -thiazolin und -thiazolidin-carbonsaeuren, verfahren zu ihrer herstellung und ihre verwendung zur beeinflussung des kollagenstoffwechsels |
| HU195492B (en) * | 1984-07-27 | 1988-05-30 | Boehringer Biochemia Srl | Process for producing 2-substituted thiazolidine derivatives with antitussive and mucus regulating action and pharmaceuticals comprising these compounds as active ingredient |
| IT1176983B (it) * | 1984-10-16 | 1987-08-26 | Zambon Spa | Dipeptidi ad attivita' farmacologica |
-
1986
- 1986-07-14 IT IT21112/86A patent/IT1196485B/it active
-
1987
- 1987-07-09 EP EP87201313A patent/EP0254354B1/de not_active Expired - Lifetime
- 1987-07-09 ES ES87201313T patent/ES2054654T3/es not_active Expired - Lifetime
- 1987-07-09 AT AT87201313T patent/ATE87622T1/de not_active IP Right Cessation
- 1987-07-09 DE DE8787201313T patent/DE3785104T2/de not_active Expired - Fee Related
- 1987-07-10 IE IE187287A patent/IE60205B1/en not_active IP Right Cessation
- 1987-07-13 US US07/072,569 patent/US4840936A/en not_active Expired - Lifetime
- 1987-07-13 AU AU75566/87A patent/AU609406B2/en not_active Ceased
- 1987-07-13 ZA ZA875099A patent/ZA875099B/xx unknown
- 1987-07-14 CA CA000541971A patent/CA1322074C/en not_active Expired - Fee Related
- 1987-07-14 JP JP62175776A patent/JP2603639B2/ja not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| IT1196485B (it) | 1988-11-16 |
| IT8621112A0 (it) | 1986-07-14 |
| CA1322074C (en) | 1993-09-07 |
| IT8621112A1 (it) | 1988-01-14 |
| AU7556687A (en) | 1988-01-21 |
| DE3785104T2 (de) | 1993-09-02 |
| ES2054654T3 (es) | 1994-08-16 |
| DE3785104D1 (de) | 1993-05-06 |
| ZA875099B (en) | 1988-04-27 |
| EP0254354B1 (de) | 1993-03-31 |
| IE871872L (en) | 1988-01-14 |
| JPS6323876A (ja) | 1988-02-01 |
| JP2603639B2 (ja) | 1997-04-23 |
| AU609406B2 (en) | 1991-05-02 |
| EP0254354A1 (de) | 1988-01-27 |
| US4840936A (en) | 1989-06-20 |
| IE60205B1 (en) | 1994-06-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |