IT1150697B - Ammido-ammino acidi ad attivita' farmacologica e relativo procedimento di preparazione - Google Patents
Ammido-ammino acidi ad attivita' farmacologica e relativo procedimento di preparazioneInfo
- Publication number
- IT1150697B IT1150697B IT20259/82A IT2025982A IT1150697B IT 1150697 B IT1150697 B IT 1150697B IT 20259/82 A IT20259/82 A IT 20259/82A IT 2025982 A IT2025982 A IT 2025982A IT 1150697 B IT1150697 B IT 1150697B
- Authority
- IT
- Italy
- Prior art keywords
- amid
- amino acids
- pharmacological activity
- preparation procedure
- related preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
- C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/022—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
- C07K5/0222—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Heart & Thoracic Surgery (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Cardiology (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US24540781A | 1981-03-19 | 1981-03-19 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IT8220259A0 IT8220259A0 (it) | 1982-03-18 |
| IT1150697B true IT1150697B (it) | 1986-12-17 |
Family
ID=22926526
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IT20259/82A IT1150697B (it) | 1981-03-19 | 1982-03-18 | Ammido-ammino acidi ad attivita' farmacologica e relativo procedimento di preparazione |
Country Status (21)
| Country | Link |
|---|---|
| JP (1) | JPS57165355A (ko) |
| KR (1) | KR890001146B1 (ko) |
| AU (1) | AU558451B2 (ko) |
| BE (1) | BE892552A (ko) |
| CH (1) | CH658455A5 (ko) |
| DE (1) | DE3209708A1 (ko) |
| DK (1) | DK120982A (ko) |
| ES (3) | ES8307718A1 (ko) |
| FI (1) | FI820974L (ko) |
| FR (1) | FR2502149A1 (ko) |
| GB (1) | GB2095252B (ko) |
| IE (1) | IE53076B1 (ko) |
| IL (1) | IL65247A (ko) |
| IN (1) | IN156096B (ko) |
| IT (1) | IT1150697B (ko) |
| NL (1) | NL8201066A (ko) |
| NO (1) | NO820903L (ko) |
| NZ (1) | NZ200047A (ko) |
| PH (1) | PH18657A (ko) |
| SE (1) | SE8201654L (ko) |
| ZA (1) | ZA821833B (ko) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3242599A1 (de) * | 1982-11-18 | 1984-05-24 | Dr. Karl Thomae Gmbh, 7950 Biberach | Neue benzazepinderivate, ihre herstellung und ihre verwendung als arzneimittel |
| US4410520A (en) * | 1981-11-09 | 1983-10-18 | Ciba-Geigy Corporation | 3-Amino-[1]-benzazepin-2-one-1-alkanoic acids |
| US4555502A (en) * | 1982-09-30 | 1985-11-26 | Merck & Co., Inc. | Aminoacyl-containing dipeptide derivatives useful as antihypertensives |
| US4410807A (en) * | 1982-03-26 | 1983-10-18 | Kay Industries, Inc. | Regulating device for polyphase electrical circuits |
| US4473575A (en) * | 1982-07-19 | 1984-09-25 | Ciba-Geigy Corporation | 3-Amino-(1)-benzazepin-2-one-1-alkanoic acids |
| US4520025A (en) * | 1982-07-21 | 1985-05-28 | William H. Rorer, Inc. | Bicyclic nitrogen heterocyclic ethers and thioethers, and their pharmaceutical uses |
| DE3302125A1 (de) * | 1983-01-22 | 1984-07-26 | Boehringer Ingelheim KG, 6507 Ingelheim | Aminosaeure-derivate, verfahren zu ihrer herstellung und verwendung |
| DK156484A (da) * | 1983-03-16 | 1984-09-17 | Usv Pharma Corp | Aminosyrederivater |
| DE3333454A1 (de) * | 1983-09-16 | 1985-04-11 | Hoechst Ag, 6230 Frankfurt | Verfahren zur herstellung von n-alkylierten dipeptiden und deren estern |
| DE3622297A1 (de) * | 1986-07-03 | 1988-01-07 | Basf Ag | Disazothiophenfarbstoffe |
| US5246943A (en) * | 1992-05-19 | 1993-09-21 | Warner-Lambert Company | Substituted 1,2,3,4-tetahydroisoquinolines with angiotensin II receptor antagonist properties |
| ES2122941B1 (es) | 1997-05-29 | 1999-07-01 | Esteve Quimica Sa | Procedimiento para la obtencion de quinapril clorhidrato y solvatos utiles para el aislamiento y purificacion de quinapril clorhidrato. |
| ES2289060T3 (es) | 2002-01-30 | 2008-02-01 | Les Laboratoires Servier | Proceso para la preparacion de perindopril de alta pureza y de intermedios utiles en su sintesis. |
| ATE360616T1 (de) | 2002-12-16 | 2007-05-15 | Lupin Ltd | Kristalline form von quinapril hydrochlorid und verfahren zu dessen herstellung |
| CA2517205C (en) * | 2003-02-28 | 2010-08-24 | Lupin Limited | Process for preparation of perindopril and salts thereof |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2503155A2 (fr) * | 1980-10-02 | 1982-10-08 | Science Union & Cie | Nouveaux imino diacides substitues, leurs procedes de preparation et leur emploi comme inhibiteur d'enzyme |
| DE3177130D1 (de) * | 1980-08-30 | 1990-01-11 | Hoechst Ag | Aminosaeurederivate, verfahren zu ihrer herstellung, diese enthaltende mittel und deren verwendung. |
| US4344949A (en) * | 1980-10-03 | 1982-08-17 | Warner-Lambert Company | Substituted acyl derivatives of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids |
| GB2086390B (en) * | 1980-11-03 | 1984-06-06 | Ciba Geigy Ag | 1-carboxy-azaalkanoylindoline-2-carboxylic acids process for their manufacture pharmaceutical preparations containing these compounds and their therapeutic application |
-
1982
- 1982-03-08 IN IN265/CAL/82A patent/IN156096B/en unknown
- 1982-03-15 NL NL8201066A patent/NL8201066A/nl not_active Application Discontinuation
- 1982-03-15 IL IL65247A patent/IL65247A/xx unknown
- 1982-03-15 PH PH26998A patent/PH18657A/en unknown
- 1982-03-16 AU AU81584/82A patent/AU558451B2/en not_active Ceased
- 1982-03-16 SE SE8201654A patent/SE8201654L/xx not_active Application Discontinuation
- 1982-03-17 DE DE19823209708 patent/DE3209708A1/de not_active Withdrawn
- 1982-03-17 GB GB8207770A patent/GB2095252B/en not_active Expired
- 1982-03-17 ES ES510498A patent/ES8307718A1/es not_active Expired
- 1982-03-18 KR KR8201157A patent/KR890001146B1/ko active
- 1982-03-18 IT IT20259/82A patent/IT1150697B/it active
- 1982-03-18 ZA ZA821833A patent/ZA821833B/xx unknown
- 1982-03-18 NZ NZ200047A patent/NZ200047A/en unknown
- 1982-03-18 CH CH1691/82A patent/CH658455A5/de not_active IP Right Cessation
- 1982-03-18 DK DK120982A patent/DK120982A/da not_active Application Discontinuation
- 1982-03-18 NO NO820903A patent/NO820903L/no unknown
- 1982-03-18 JP JP57041801A patent/JPS57165355A/ja active Pending
- 1982-03-18 BE BE0/207610A patent/BE892552A/fr not_active IP Right Cessation
- 1982-03-19 FR FR8204738A patent/FR2502149A1/fr active Granted
- 1982-03-19 FI FI820974A patent/FI820974L/fi not_active Application Discontinuation
- 1982-03-19 IE IE635/82A patent/IE53076B1/en unknown
-
1983
- 1983-03-16 ES ES521030A patent/ES521030A0/es active Granted
- 1983-03-16 ES ES521031A patent/ES8501363A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| IT8220259A0 (it) | 1982-03-18 |
| NO820903L (no) | 1982-09-20 |
| DK120982A (da) | 1982-09-20 |
| FR2502149A1 (fr) | 1982-09-24 |
| IL65247A0 (en) | 1982-05-31 |
| IL65247A (en) | 1987-07-31 |
| ES521031A0 (es) | 1984-12-01 |
| KR830009065A (ko) | 1983-12-17 |
| ES510498A0 (es) | 1983-08-01 |
| NZ200047A (en) | 1985-07-12 |
| FI820974L (fi) | 1982-09-20 |
| SE8201654L (sv) | 1982-09-20 |
| KR890001146B1 (ko) | 1989-04-25 |
| GB2095252B (en) | 1985-04-17 |
| AU8158482A (en) | 1982-09-23 |
| IN156096B (ko) | 1985-05-11 |
| JPS57165355A (en) | 1982-10-12 |
| FR2502149B1 (ko) | 1985-01-18 |
| ES8307718A1 (es) | 1983-08-01 |
| BE892552A (fr) | 1982-09-20 |
| IE820635L (en) | 1982-09-19 |
| GB2095252A (en) | 1982-09-29 |
| ZA821833B (en) | 1983-01-26 |
| DE3209708A1 (de) | 1982-10-21 |
| ES8404317A1 (es) | 1984-05-16 |
| ES521030A0 (es) | 1984-05-16 |
| PH18657A (en) | 1985-08-29 |
| NL8201066A (nl) | 1982-10-18 |
| ES8501363A1 (es) | 1984-12-01 |
| CH658455A5 (de) | 1986-11-14 |
| IE53076B1 (en) | 1988-06-08 |
| AU558451B2 (en) | 1987-01-29 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IT1142170B (it) | Composti eterosiclici dotati di attivita' farmacologica e procedimento per la loro preparazione | |
| IT8519512A0 (it) | Derivati naturali ad attivita'farmacologica | |
| IT1197038B (it) | Composizione farmaceutica ad attivita' analgesica | |
| IT1190375B (it) | N-benzidrildiazacicloalchil-alcanilidi ad attivita' antianafilattica ed antibroncospastica | |
| IT7849577A0 (it) | Derivati spiroamminici ad attivita'farmacologica e relativo procedimento di produzione | |
| IT1150697B (it) | Ammido-ammino acidi ad attivita' farmacologica e relativo procedimento di preparazione | |
| IT1196348B (it) | Composti ad attivita'antiinfiammatoria | |
| IT1186717B (it) | Benzoil-uree ad attivita' insetticida | |
| IT1150622B (it) | Polisaccaridi dotati di attivita' ant-carcinogena e procedimento per la loro preparazione | |
| IT1187756B (it) | Isoindolinil-alchil-piperazine ad attivita' farmaceutica | |
| AR231144A1 (es) | Procedimiento para la preparacion de 5'-desoxi-5'-metilticadenosina con actividad antiinflamatoria y analgesica | |
| IT1178792B (it) | Acilammino mitosani ad attivita'antitumorale e relativo procedimento di preparazione | |
| IT1190130B (it) | Acidi 3-acilammino-2-osso-1-azetidinsolfonici | |
| IT1164826B (it) | Composti di acido epossisuccinammico dotati di proprieta' farmacologiche e procedimento di preparazione | |
| IT1117779B (it) | Alchil-tiofenossialchilammine ad attivita'biologica ed aventi proprieta'farmacologiche | |
| IT7920398A0 (it) | Derivato ad attivita' analgesica antiinfiammatoria potenziata eprocedimento per la sua preparazione. | |
| IT1128706B (it) | Procedimento per la preparazione di acidi arilpropionici dotati di attivita' farmacologica | |
| BE893322A (fr) | Preparation d'acides carboxyliques | |
| BE880495A (fr) | Derives mercaptoacyles d'acides 4,5-dihydro-1h-pyrrole-2-carboxyliques et d'acides 1,4,5,6-tetrahydro-pyridine-2-carboxyliques | |
| IT8721328A0 (it) | Acidi idrossimici di eteri e ditioeteri 7 ossabicicloeptansostituiti. | |
| IT8247833A0 (it) | Derivato di colesterolo idrosolubile dotato di attivita' farmacologica e procedimento di preparazione | |
| NO862548D0 (no) | Fremstilling av 3-amino-4-hydroksy-benzosyrer. | |
| IT1188557B (it) | Acidi 8-osso-2-ossa-1-azabiciclo (4.2.0)ottano-3-carbossilici | |
| IT8249095A0 (it) | Derivati di 4-piridilpiridazinone dotati di attivita' antiinfiammatoria ed analgesica | |
| FR2510117B1 (fr) | Nouveaux derives d'hydrazonocephem et leur application pharmacologique |