IN2012DN04867A - - Google Patents

Download PDF

Info

Publication number
IN2012DN04867A
IN2012DN04867A IN4867DEN2012A IN2012DN04867A IN 2012DN04867 A IN2012DN04867 A IN 2012DN04867A IN 4867DEN2012 A IN4867DEN2012 A IN 4867DEN2012A IN 2012DN04867 A IN2012DN04867 A IN 2012DN04867A
Authority
IN
India
Prior art keywords
women
additional
benefits
compositions
antiovulatory
Prior art date
Application number
Other languages
English (en)
Inventor
Regine Sitruk-Ware
Dario Norberto Ramon Carrara
Arnaud Grenier
Original Assignee
Population Council Inc
Antares Pharma Ipl Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Population Council Inc, Antares Pharma Ipl Ag filed Critical Population Council Inc
Publication of IN2012DN04867A publication Critical patent/IN2012DN04867A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
IN4867DEN2012 2009-12-17 2010-12-17 IN2012DN04867A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US28751409P 2009-12-17 2009-12-17
PCT/US2010/060941 WO2011084668A1 (en) 2009-12-17 2010-12-17 Nestorone®/estradiol transdermal gel

Publications (1)

Publication Number Publication Date
IN2012DN04867A true IN2012DN04867A (ru) 2015-09-25

Family

ID=43640394

Family Applications (1)

Application Number Title Priority Date Filing Date
IN4867DEN2012 IN2012DN04867A (ru) 2009-12-17 2010-12-17

Country Status (14)

Country Link
US (1) US9682087B2 (ru)
EP (1) EP2512486B1 (ru)
JP (1) JP6082249B2 (ru)
KR (2) KR20120107492A (ru)
CN (1) CN102753180A (ru)
AU (1) AU2010339867B2 (ru)
BR (1) BR112012014059B1 (ru)
CA (1) CA2782075C (ru)
ES (1) ES2641613T3 (ru)
IN (1) IN2012DN04867A (ru)
MX (1) MX363536B (ru)
NZ (1) NZ600907A (ru)
WO (1) WO2011084668A1 (ru)
ZA (1) ZA201204267B (ru)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9301920B2 (en) 2012-06-18 2016-04-05 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
ES2885523T3 (es) 2011-11-23 2021-12-14 Therapeuticsmd Inc Formulaciones y terapias de reposición hormonal de combinación naturales
CN102657661A (zh) * 2012-04-15 2012-09-12 温州医学院 Nestorone在制备治疗阿尔茨海默病的药物用途
US10806740B2 (en) 2012-06-18 2020-10-20 Therapeuticsmd, Inc. Natural combination hormone replacement formulations and therapies
US20150196640A1 (en) 2012-06-18 2015-07-16 Therapeuticsmd, Inc. Progesterone formulations having a desirable pk profile
US10806697B2 (en) 2012-12-21 2020-10-20 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US20130338122A1 (en) 2012-06-18 2013-12-19 Therapeuticsmd, Inc. Transdermal hormone replacement therapies
US11266661B2 (en) 2012-12-21 2022-03-08 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10471072B2 (en) 2012-12-21 2019-11-12 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9180091B2 (en) 2012-12-21 2015-11-10 Therapeuticsmd, Inc. Soluble estradiol capsule for vaginal insertion
US11246875B2 (en) 2012-12-21 2022-02-15 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10568891B2 (en) 2012-12-21 2020-02-25 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US10537581B2 (en) 2012-12-21 2020-01-21 Therapeuticsmd, Inc. Vaginal inserted estradiol pharmaceutical compositions and methods
US9433680B2 (en) 2013-01-31 2016-09-06 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US9446131B2 (en) 2013-01-31 2016-09-20 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US9452173B2 (en) 2013-01-31 2016-09-27 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
US8778365B1 (en) 2013-01-31 2014-07-15 Merz Pharmaceuticals, Llc Topical compositions and methods for making and using same
RU2016143081A (ru) 2014-05-22 2018-06-26 Терапьютиксмд, Инк. Натуральные комбинированные гормонозаместительные составы и терапии
JP2017523138A (ja) 2014-07-29 2017-08-17 セラピューティックスエムディー インコーポレーテッドTherapeuticsmd, Inc. 経皮クリーム
US10328087B2 (en) 2015-07-23 2019-06-25 Therapeuticsmd, Inc. Formulations for solubilizing hormones
RU2648470C2 (ru) * 2016-03-03 2018-03-26 Государственное бюджетное образовательное учреждение высшего профессионального образования "Уральский государственный медицинский университет Министерства здравоохранения Российской Федерации" (ГБОУ ВПО УГМУ Минздрава России) Способ оптимизации лечения женщин кардиотропной терапией и заместительной гормональной терапией при эстрогенодефиците с артериальной гипертензией в позднем репродуктивном периоде
US9931349B2 (en) 2016-04-01 2018-04-03 Therapeuticsmd, Inc. Steroid hormone pharmaceutical composition
US10286077B2 (en) 2016-04-01 2019-05-14 Therapeuticsmd, Inc. Steroid hormone compositions in medium chain oils
WO2022212529A1 (en) * 2021-03-30 2022-10-06 Viatris Inc. Transdermal systems having low dose estrogen and methods of making and use

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1093816A3 (en) 1990-06-01 2003-10-22 The Population Council, Inc. Use of ST1435 in hormonal therapy by transdermal application
US5122382A (en) 1990-10-29 1992-06-16 Alza Corporation Transdermal contraceptive formulations, methods and devices
US5198223A (en) * 1990-10-29 1993-03-30 Alza Corporation Transdermal formulations, methods and devices
JPH04342531A (ja) 1991-05-21 1992-11-30 Sekisui Chem Co Ltd 経皮吸収製剤
US7198801B2 (en) * 2000-08-03 2007-04-03 Antares Pharma Ipl Ag Formulations for transdermal or transmucosal application
MX347890B (es) 2009-10-19 2017-05-18 The Population Council Inc Neuroproteccion y reparacion de melina usando progestina.

Also Published As

Publication number Publication date
WO2011084668A1 (en) 2011-07-14
AU2010339867A1 (en) 2012-07-19
CN102753180A (zh) 2012-10-24
CA2782075A1 (en) 2011-07-14
JP2013514984A (ja) 2013-05-02
BR112012014059A2 (pt) 2016-07-05
BR112012014059B1 (pt) 2020-03-10
NZ600907A (en) 2013-11-29
AU2010339867B2 (en) 2014-07-24
ZA201204267B (en) 2013-01-31
MX2012006755A (es) 2012-11-23
KR101928321B1 (ko) 2018-12-12
KR20180084149A (ko) 2018-07-24
ES2641613T3 (es) 2017-11-10
EP2512486A1 (en) 2012-10-24
US9682087B2 (en) 2017-06-20
MX363536B (es) 2019-03-27
US20130045953A1 (en) 2013-02-21
EP2512486B1 (en) 2017-06-28
CA2782075C (en) 2015-06-30
BR112012014059A8 (pt) 2017-12-26
JP6082249B2 (ja) 2017-02-15
KR20120107492A (ko) 2012-10-02

Similar Documents

Publication Publication Date Title
IN2012DN04867A (ru)
MX2012012026A (es) Formas de dosificacion solidas orales con dosis muy bajas para la hrt.
PL2131847T3 (pl) Lek zawierający przynajmniej jeden gestagen
MX2009004616A (es) Metodos de tratamiento hormonal que utilizan regimenes de ciclo extendido de dosis ascendente.
EA200900491A1 (ru) Применение эстрадиола валерата или 17в-эстрадиола в комбинации с диеногестом для перорального лечения для поддержания и/или повышения полового влечения у особи женского пола
MX353713B (es) Composiciones de administracion dermica y metodos.
MX2017013565A (es) Ligandos degradadores selectivos del receptor androgénico (sard) y sus métodos uso.
MY161549A (en) Progesterone antagonists such as cdb-4124 in the treatment of breast cancer
GB2479337A (en) Combination of a 17 alpha-hydroxylase/c17, 20-lyase inhibitor with an additional therapeutic agent
GB201104241D0 (en) Dosages for menstrual suppression, contraception, and hormone replacement therapy, and methods of administrating same
MX338290B (es) Tratamiento de enfermedad de alzheimer, perdida de cognición, perdida de memoria y demencia con precursores de esteroides sexuales en conbinación con moduladores selectivos del receptor de estrógenos.
CU20120175A7 (es) Compuestos derivados de 6,7-dihidro-5h-benzo[7]anulenos
AU2012293593A8 (en) Use of estetrol as emergency contraceptive
PH12015500062A1 (en) 3-substituted estra-1,3,5(10),16-tetraene derivatives, methods for the production thereof, pharmaceutical preparations containing same, and use thereof for the production of medicaments
SE0400346D0 (sv) Steroids for cancer treatment
DK201270089A (en) Fulvestrant in a dosage of 50mg for the treatment of advanced cancer
TW200612962A (en) Estriol and estetrol prodrugs
JP2013500324A5 (ru)
MX2019014677A (es) Compuestos de estra-1,3,5(10)-trien-17-ona sustituida con 15.beta.-[3-propanamido] y sus 17-oximas para usarse en la inhibicion de 17.beta.-hidroxiesteroides deshidrogenasas.
UA99918C2 (ru) 8-бета-замещенные эстратриены как селективно активные эстрогены
NZ627242A (en) Transdermal hormone delivery
MX2023001868A (es) Composicion de anticonceptivo oral de liberacion modificada.
MX2021006426A (es) Sistema de suministro de farmaco para combinaciones de estrogeno de dosis ultra-baja y metodos y usos del mismo.
Frey Ethinylestradiol/drospirenone/norelgestromin
Elia Various toxicities: 12 case reports