IN2011KN04192A - - Google Patents
Info
- Publication number
- IN2011KN04192A IN2011KN04192A IN4192KON2011A IN2011KN04192A IN 2011KN04192 A IN2011KN04192 A IN 2011KN04192A IN 4192KON2011 A IN4192KON2011 A IN 4192KON2011A IN 2011KN04192 A IN2011KN04192 A IN 2011KN04192A
- Authority
- IN
- India
- Prior art keywords
- methylphenyl
- preparation
- thiazolo
- cyclopropyl
- fluoro
- Prior art date
Links
- 238000002360 preparation method Methods 0.000 abstract 2
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/42—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C331/00—Derivatives of thiocyanic acid or of isothiocyanic acid
- C07C331/02—Thiocyanates
- C07C331/04—Thiocyanates having sulfur atoms of thiocyanate groups bound to acyclic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
- C07D327/02—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
- C07D327/04—Five-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D339/00—Heterocyclic compounds containing rings having two sulfur atoms as the only ring hetero atoms
- C07D339/02—Five-membered rings
- C07D339/06—Five-membered rings having the hetero atoms in positions 1 and 3, e.g. cyclic dithiocarbonates
-
- C—CHEMISTRY; METALLURGY
- C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
- C08F—MACROMOLECULAR COMPOUNDS OBTAINED BY REACTIONS ONLY INVOLVING CARBON-TO-CARBON UNSATURATED BONDS
- C08F216/00—Copolymers of compounds having one or more unsaturated aliphatic radicals, each having only one carbon-to-carbon double bond, and at least one being terminated by an alcohol, ether, aldehydo, ketonic, acetal or ketal radical
- C08F216/12—Copolymers of compounds having one or more unsaturated aliphatic radicals, each having only one carbon-to-carbon double bond, and at least one being terminated by an alcohol, ether, aldehydo, ketonic, acetal or ketal radical by an ether radical
- C08F216/14—Monomers containing only one unsaturated aliphatic radical
- C08F216/1466—Monomers containing sulfur
- C08F216/1483—Monomers containing sulfur and nitrogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU0900267A HUP0900267A2 (en) | 2009-04-30 | 2009-04-30 | Process for preparing of thiazole amines and intermediates thereof |
| PCT/HU2010/000047 WO2010125414A1 (en) | 2009-04-30 | 2010-04-26 | Process for the preparation of [4-(2-chloro-4-methoxy-5-methylphenyl)-5-methyl-thiazolo-2-yl]-[2-cyclopropyl-1-(3-fluoro-4-methylphenyl)-ethyl]-amine |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2011KN04192A true IN2011KN04192A (ru) | 2015-10-02 |
Family
ID=89988941
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN4192KON2011 IN2011KN04192A (ru) | 2009-04-30 | 2010-04-26 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US8314249B2 (ru) |
| EP (1) | EP2424848B1 (ru) |
| JP (1) | JP5608221B2 (ru) |
| KR (1) | KR20120014005A (ru) |
| CN (1) | CN102414185B (ru) |
| AR (1) | AR076478A1 (ru) |
| AU (1) | AU2010243362B2 (ru) |
| BR (1) | BRPI1014627A2 (ru) |
| CA (1) | CA2760384A1 (ru) |
| HU (1) | HUP0900267A2 (ru) |
| IL (1) | IL216017A0 (ru) |
| IN (1) | IN2011KN04192A (ru) |
| MX (1) | MX2011011530A (ru) |
| MY (1) | MY152269A (ru) |
| RU (1) | RU2523793C2 (ru) |
| SG (1) | SG175829A1 (ru) |
| TW (1) | TWI461413B (ru) |
| UY (1) | UY32594A (ru) |
| WO (1) | WO2010125414A1 (ru) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8943551B2 (en) * | 2008-08-14 | 2015-01-27 | Microsoft Corporation | Cloud-based device information storage |
| HUP0900267A2 (en) | 2009-04-30 | 2011-03-28 | Sanofi Aventis | Process for preparing of thiazole amines and intermediates thereof |
| KR102258522B1 (ko) | 2014-01-21 | 2021-05-31 | 뉴로크린 바이오사이언시즈 인코퍼레이티드 | 선천성 부신 과형성 치료를 위한 ｃｒｆ1 수용체 길항제 |
| US10207974B1 (en) | 2017-12-05 | 2019-02-19 | Chevron Phillips Chemical Company Lp | Synthesis of gamma dicarbonyl and pyrrole compounds |
| CN113518616A (zh) * | 2018-12-07 | 2021-10-19 | 纽罗克里生物科学有限公司 | 用于治疗先天性肾上腺皮质增生症的crf1受体拮抗剂、其药物制剂和固体形式 |
| EP4034111A1 (en) * | 2019-09-27 | 2022-08-03 | Neurocrine Biosciences, Inc. | Crf receptor antagonists and methods of use |
| MA58993A1 (fr) | 2020-06-10 | 2023-09-27 | Sanofi Sa | Antagoniste du récepteur crf1 pour le traitement de l'hyperplasie surrénale congénitale |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB823251A (en) | 1955-07-02 | 1959-11-11 | Thomae Gmbh Dr K | Improvements in or relating to preparations containing benzoxathiol derivatives for the care of hair and skin |
| US3222248A (en) * | 1961-12-12 | 1965-12-07 | Stauffer Chemical Co | Method of controlling microorganisms by means of organic thiocyanates |
| US3433803A (en) | 1966-12-01 | 1969-03-18 | Olin Mathieson | Substituted imino-1,3-oxathiols and their preparation |
| IL103586A (en) | 1991-10-30 | 1997-09-30 | Astra Ab | Process for the preparation of 4-methyl-5- (2-chloroethyl)-thiazole and analogues thereof |
| JPH1036360A (ja) | 1996-02-21 | 1998-02-10 | Kuraray Co Ltd | ２−クロロ−５−クロロメチル−１，３−チアゾールの製造方法 |
| FR2796380B3 (fr) * | 1999-07-15 | 2001-08-17 | Sanofi Synthelabo | Nouveaux derives d'aminothiazoles, leur preparation et les compositions pharmaceutiques les contenant |
| HUP0900267A2 (en) | 2009-04-30 | 2011-03-28 | Sanofi Aventis | Process for preparing of thiazole amines and intermediates thereof |
-
2009
- 2009-04-30 HU HU0900267A patent/HUP0900267A2/hu unknown
-
2010
- 2010-04-26 SG SG2011079696A patent/SG175829A1/en unknown
- 2010-04-26 MX MX2011011530A patent/MX2011011530A/es active IP Right Grant
- 2010-04-26 BR BRPI1014627-0A patent/BRPI1014627A2/pt not_active IP Right Cessation
- 2010-04-26 JP JP2012507828A patent/JP5608221B2/ja not_active Expired - Fee Related
- 2010-04-26 MY MYPI2011005171 patent/MY152269A/en unknown
- 2010-04-26 WO PCT/HU2010/000047 patent/WO2010125414A1/en active Application Filing
- 2010-04-26 CA CA2760384A patent/CA2760384A1/en active Pending
- 2010-04-26 AU AU2010243362A patent/AU2010243362B2/en not_active Ceased
- 2010-04-26 RU RU2011148584/04A patent/RU2523793C2/ru not_active IP Right Cessation
- 2010-04-26 KR KR1020117028054A patent/KR20120014005A/ko not_active Application Discontinuation
- 2010-04-26 CN CN201080018790.6A patent/CN102414185B/zh not_active Expired - Fee Related
- 2010-04-26 EP EP10718684A patent/EP2424848B1/en not_active Not-in-force
- 2010-04-26 IN IN4192KON2011 patent/IN2011KN04192A/en unknown
- 2010-04-28 AR ARP100101422A patent/AR076478A1/es unknown
- 2010-04-29 TW TW099113599A patent/TWI461413B/zh not_active IP Right Cessation
- 2010-04-30 UY UY0001032594A patent/UY32594A/es not_active Application Discontinuation
-
2011
- 2011-10-27 IL IL216017A patent/IL216017A0/en unknown
- 2011-10-27 US US13/282,721 patent/US8314249B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| AR076478A1 (es) | 2011-06-15 |
| CN102414185B (zh) | 2014-02-26 |
| KR20120014005A (ko) | 2012-02-15 |
| HU0900267D0 (en) | 2009-07-28 |
| CA2760384A1 (en) | 2010-11-04 |
| WO2010125414A1 (en) | 2010-11-04 |
| UY32594A (es) | 2010-11-30 |
| MX2011011530A (es) | 2011-11-18 |
| RU2523793C2 (ru) | 2014-07-27 |
| US8314249B2 (en) | 2012-11-20 |
| AU2010243362A1 (en) | 2011-11-17 |
| RU2011148584A (ru) | 2013-06-10 |
| AU2010243362B2 (en) | 2015-07-30 |
| BRPI1014627A2 (pt) | 2015-08-25 |
| JP2012525368A (ja) | 2012-10-22 |
| HUP0900267A2 (en) | 2011-03-28 |
| EP2424848A1 (en) | 2012-03-07 |
| EP2424848B1 (en) | 2013-03-13 |
| CN102414185A (zh) | 2012-04-11 |
| US20120083608A1 (en) | 2012-04-05 |
| IL216017A0 (en) | 2012-01-31 |
| TWI461413B (zh) | 2014-11-21 |
| MY152269A (en) | 2014-09-15 |
| JP5608221B2 (ja) | 2014-10-15 |
| WO2010125414A8 (en) | 2011-04-07 |
| SG175829A1 (en) | 2011-12-29 |
| TW201105640A (en) | 2011-02-16 |
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