IL96134A0 - Substituted cycloalkano(b)-dihydroindole-and-indolesulphonamides,their preparation and pharmaceutical compositions containing them - Google Patents
Substituted cycloalkano(b)-dihydroindole-and-indolesulphonamides,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL96134A0 IL96134A0 IL96134A IL9613490A IL96134A0 IL 96134 A0 IL96134 A0 IL 96134A0 IL 96134 A IL96134 A IL 96134A IL 9613490 A IL9613490 A IL 9613490A IL 96134 A0 IL96134 A0 IL 96134A0
- Authority
- IL
- Israel
- Prior art keywords
- dihydroindole
- indolesulphonamides
- preparation
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/82—Carbazoles; Hydrogenated carbazoles
- C07D209/88—Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB898924392A GB8924392D0 (en) | 1989-10-30 | 1989-10-30 | Substituted cycloalkano/b/dihydroindole-and-indolesulphonamides |
Publications (1)
Publication Number | Publication Date |
---|---|
IL96134A0 true IL96134A0 (en) | 1991-07-18 |
Family
ID=10665396
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL96134A IL96134A0 (en) | 1989-10-30 | 1990-10-26 | Substituted cycloalkano(b)-dihydroindole-and-indolesulphonamides,their preparation and pharmaceutical compositions containing them |
Country Status (21)
Country | Link |
---|---|
US (3) | US5039670A (pt) |
EP (1) | EP0425906B1 (pt) |
JP (1) | JPH03151360A (pt) |
KR (1) | KR910007876A (pt) |
CN (1) | CN1051354A (pt) |
AT (1) | ATE102185T1 (pt) |
AU (1) | AU628665B2 (pt) |
CA (1) | CA2028621A1 (pt) |
DE (1) | DE59004764D1 (pt) |
DK (1) | DK0425906T3 (pt) |
ES (1) | ES2062250T3 (pt) |
FI (1) | FI905294A0 (pt) |
GB (1) | GB8924392D0 (pt) |
HU (1) | HUT57190A (pt) |
IE (1) | IE903869A1 (pt) |
IL (1) | IL96134A0 (pt) |
NO (1) | NO904487L (pt) |
NZ (1) | NZ235860A (pt) |
PH (1) | PH27484A (pt) |
PT (1) | PT95728A (pt) |
ZA (1) | ZA908637B (pt) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE59208448D1 (de) * | 1991-08-15 | 1997-06-12 | Ciba Geigy Ag | N-Acyl-N-Heterocyclyl- oder Naphthylalkyl-Aminosäuren als Angiotensin II Antagonisten |
DE19506739A1 (de) * | 1995-02-27 | 1996-08-29 | Bayer Ag | [3-Amino]-tetrahydrocarbazol-propansäureester |
US5708187A (en) * | 1996-06-27 | 1998-01-13 | Eli Lilly And Company | 6-substituted-1,2,3,4-tetrahydro-9H-carbazoles and 7-substituted-10H-cyclohepta 7,6-B!indoles: New 5-HT1F agonists |
WO2003097598A1 (fr) * | 2002-05-16 | 2003-11-27 | Shionogi & Co., Ltd. | Composé comprenant un antagonisme du récepteur de pdg2 |
WO2003097042A1 (fr) * | 2002-05-16 | 2003-11-27 | Shionogi & Co., Ltd. | Antagoniste de recepteur de pdg2 |
CA2528321A1 (en) * | 2003-06-10 | 2004-12-23 | Smithkline Beecham Corporation | Tetrahydrocarbazole derivatives and their pharmaceutical use |
DK1902026T3 (da) * | 2005-06-24 | 2010-04-26 | Lilly Co Eli | Tetrahydrocarbazol-derivater, der kan anvendes som androgen-receptor-modulatorer (SARM) |
US7662831B2 (en) | 2006-07-27 | 2010-02-16 | Wyeth Llc | Tetracyclic indoles as potassium channel modulators |
US7601856B2 (en) | 2006-07-27 | 2009-10-13 | Wyeth | Benzofurans as potassium ion channel modulators |
UA98777C2 (en) * | 2006-11-20 | 2012-06-25 | Эли Лилли Энд Компани | Tetrahydrocyclopenta[b]indole compounds as androgen receptor modulators |
CN101434571B (zh) * | 2007-11-13 | 2012-05-30 | 杭州容立医药科技有限公司 | 环烷并[1,2-b]吲哚磺酰胺、其异构体或其盐的合成方法 |
BRPI0912394A2 (pt) * | 2008-05-16 | 2016-07-26 | Lilly Co Eli | moduladores do receptor de androgênio à base de tetra-hidrociclopenta[b]indol |
CN106103435B (zh) | 2014-03-17 | 2018-11-16 | 爱杜西亚药品有限公司 | 氮杂吲哚乙酸衍生物及彼等作为前列腺素d2受体调节剂的用途 |
CN108026093B (zh) | 2015-09-15 | 2021-11-16 | 爱杜西亚药品有限公司 | 结晶形式 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3514696A1 (de) * | 1985-04-24 | 1986-11-06 | Bayer Ag, 5090 Leverkusen | N-indolylethyl-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung |
DE3525801A1 (de) * | 1985-07-19 | 1987-01-22 | Hoechst Ag | Tertiaere hydroxyalkylxanthine, verfahren zu ihrer herstellung, die sie enthaltenden arzneimittel und ihre verwendung |
ES2038653T3 (es) * | 1986-01-23 | 1993-08-01 | Merck Frosst Canada Inc. | Acidos 1-alcanoicos tetrahidrocarbazol. |
US4808608A (en) * | 1986-01-23 | 1989-02-28 | Merck & Co., Inc. | Tetrahydrocarbazole 1-alkanoic acids, pharmaceutical compositions and use |
DE3631824A1 (de) * | 1986-02-21 | 1988-03-31 | Bayer Ag | Cycloalkano(1.2-b)indol-sulfonamide |
US4940719A (en) * | 1986-03-27 | 1990-07-10 | Merck Frosst Canada, Inc. | Tetrahydrocarbazole esters, pharmaceutical compositions and use |
DE3613623A1 (de) * | 1986-04-23 | 1987-10-29 | Bayer Ag | N-dihydroindolylethyl-sulfonamide |
-
1989
- 1989-10-30 GB GB898924392A patent/GB8924392D0/en active Pending
-
1990
- 1990-10-05 AU AU63848/90A patent/AU628665B2/en not_active Ceased
- 1990-10-17 US US07/599,321 patent/US5039670A/en not_active Expired - Fee Related
- 1990-10-17 NO NO90904487A patent/NO904487L/no unknown
- 1990-10-18 DE DE90119974T patent/DE59004764D1/de not_active Expired - Fee Related
- 1990-10-18 EP EP90119974A patent/EP0425906B1/de not_active Expired - Lifetime
- 1990-10-18 DK DK90119974.5T patent/DK0425906T3/da active
- 1990-10-18 ES ES90119974T patent/ES2062250T3/es not_active Expired - Lifetime
- 1990-10-18 AT AT90119974T patent/ATE102185T1/de not_active IP Right Cessation
- 1990-10-25 JP JP2286009A patent/JPH03151360A/ja active Pending
- 1990-10-26 FI FI905294A patent/FI905294A0/fi not_active Application Discontinuation
- 1990-10-26 IL IL96134A patent/IL96134A0/xx unknown
- 1990-10-26 CA CA002028621A patent/CA2028621A1/en not_active Abandoned
- 1990-10-26 IE IE386990A patent/IE903869A1/en unknown
- 1990-10-26 NZ NZ235860A patent/NZ235860A/en unknown
- 1990-10-29 KR KR1019900017353A patent/KR910007876A/ko not_active Application Discontinuation
- 1990-10-29 PT PT95728A patent/PT95728A/pt not_active Application Discontinuation
- 1990-10-29 HU HU906925A patent/HUT57190A/hu unknown
- 1990-10-29 ZA ZA908637A patent/ZA908637B/xx unknown
- 1990-10-30 PH PH41465A patent/PH27484A/en unknown
- 1990-10-30 CN CN90108726A patent/CN1051354A/zh active Pending
-
1991
- 1991-03-28 US US07/678,563 patent/US5096897A/en not_active Expired - Fee Related
-
1993
- 1993-04-05 US US08/042,857 patent/US5374647A/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
EP0425906A3 (en) | 1992-01-22 |
HU906925D0 (en) | 1991-05-28 |
FI905294A0 (fi) | 1990-10-26 |
DK0425906T3 (da) | 1994-04-11 |
AU6384890A (en) | 1991-06-20 |
IE903869A1 (en) | 1991-05-08 |
AU628665B2 (en) | 1992-09-17 |
KR910007876A (ko) | 1991-05-30 |
GB8924392D0 (en) | 1989-12-20 |
US5039670A (en) | 1991-08-13 |
PH27484A (en) | 1993-07-23 |
EP0425906A2 (de) | 1991-05-08 |
NO904487D0 (no) | 1990-10-17 |
HUT57190A (en) | 1991-11-28 |
CA2028621A1 (en) | 1991-05-01 |
EP0425906B1 (de) | 1994-03-02 |
NO904487L (no) | 1991-05-02 |
DE59004764D1 (de) | 1994-04-07 |
ATE102185T1 (de) | 1994-03-15 |
JPH03151360A (ja) | 1991-06-27 |
NZ235860A (en) | 1992-09-25 |
US5096897A (en) | 1992-03-17 |
US5374647A (en) | 1994-12-20 |
ES2062250T3 (es) | 1994-12-16 |
CN1051354A (zh) | 1991-05-15 |
PT95728A (pt) | 1991-09-13 |
ZA908637B (en) | 1991-08-28 |
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