IL93262A - Preparation of optically active 3-thiolnyl sulfonate esters - Google Patents

Preparation of optically active 3-thiolnyl sulfonate esters

Info

Publication number
IL93262A
IL93262A IL9326290A IL9326290A IL93262A IL 93262 A IL93262 A IL 93262A IL 9326290 A IL9326290 A IL 9326290A IL 9326290 A IL9326290 A IL 9326290A IL 93262 A IL93262 A IL 93262A
Authority
IL
Israel
Prior art keywords
formula
optically active
solvent
reaction
preparation
Prior art date
Application number
IL9326290A
Other languages
English (en)
Hebrew (he)
Other versions
IL93262A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/308,868 external-priority patent/US4864046A/en
Priority claimed from US07/378,888 external-priority patent/US4921972A/en
Application filed by Pfizer filed Critical Pfizer
Publication of IL93262A0 publication Critical patent/IL93262A0/xx
Publication of IL93262A publication Critical patent/IL93262A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/16—Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/64—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms
    • C07C309/65—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to acyclic carbon atoms of a saturated carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C309/06—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing halogen atoms, or nitro or nitroso groups bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/63—Esters of sulfonic acids
    • C07C309/72—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C309/73—Esters of sulfonic acids having sulfur atoms of esterified sulfo groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton to carbon atoms of non-condensed six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30—Hetero atoms other than halogen
    • C07D333/32—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
IL9326290A 1989-02-09 1990-02-02 Preparation of optically active 3-thiolnyl sulfonate esters IL93262A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US07/308,868 US4864046A (en) 1989-02-09 1989-02-09 Process for optically active 3-thiolanyl sulfonate esters
US07/378,888 US4921972A (en) 1989-05-17 1989-07-12 Process for optically active 3-thiolanyl sulfonate esters

Publications (2)

Publication Number Publication Date
IL93262A0 IL93262A0 (en) 1990-11-29
IL93262A true IL93262A (en) 1994-08-26

Family

ID=26976494

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9326290A IL93262A (en) 1989-02-09 1990-02-02 Preparation of optically active 3-thiolnyl sulfonate esters

Country Status (13)

Country Link
EP (1) EP0382418A3 (ja)
JP (1) JPH0643355B2 (ja)
KR (1) KR920010181B1 (ja)
AU (1) AU609348B2 (ja)
CA (1) CA2009457A1 (ja)
DK (1) DK0382418T3 (ja)
FI (1) FI92583C (ja)
HU (1) HU203545B (ja)
IL (1) IL93262A (ja)
MY (1) MY105176A (ja)
NO (1) NO173443C (ja)
NZ (1) NZ232425A (ja)
PT (1) PT93075A (ja)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005314374A (ja) * 2004-03-31 2005-11-10 Daiso Co Ltd ３−ヒドロキシチオランの新規製法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1988008845A1 (en) * 1987-05-11 1988-11-17 Pfizer Inc. Diastereomeric 5r,6s-6-(1r-hydroxyethyl)-2-(cis-1-oxo-3-thiolanylthio)-2-penem-3-carboxylic acids
US4992543A (en) * 1988-10-19 1991-02-12 Pfizer Inc. Penem derivatives
US4864046A (en) * 1989-02-09 1989-09-05 Pfizer Inc. Process for optically active 3-thiolanyl sulfonate esters

Also Published As

Publication number Publication date
NO173443B (no) 1993-09-06
FI92583B (fi) 1994-08-31
HU203545B (en) 1991-08-28
NO173443C (no) 1993-12-15
PT93075A (pt) 1990-08-31
EP0382418A2 (en) 1990-08-16
AU4937890A (en) 1990-08-16
NO900603D0 (no) 1990-02-08
NZ232425A (en) 1991-05-28
HUT52768A (en) 1990-08-28
JPH02240077A (ja) 1990-09-25
HU900727D0 (en) 1990-04-28
AU609348B2 (en) 1991-04-26
JPH0643355B2 (ja) 1994-06-08
CA2009457A1 (en) 1990-08-09
EP0382418A3 (en) 1991-10-23
FI92583C (fi) 1994-12-12
FI900626A0 (fi) 1990-02-08
KR920010181B1 (ko) 1992-11-19
KR900012923A (ko) 1990-09-03
MY105176A (en) 1994-08-30
IL93262A0 (en) 1990-11-29
NO900603L (no) 1990-08-10
DK0382418T3 (da) 1991-10-23

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Legal Events

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