IL88047A - Aminomethyl oxooxazolidinyl aroylbenzene derivatives,their preparation and pharmaceutical compositions containing them - Google Patents
Aminomethyl oxooxazolidinyl aroylbenzene derivatives,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL88047A IL88047A IL88047A IL8804788A IL88047A IL 88047 A IL88047 A IL 88047A IL 88047 A IL88047 A IL 88047A IL 8804788 A IL8804788 A IL 8804788A IL 88047 A IL88047 A IL 88047A
- Authority
- IL
- Israel
- Prior art keywords
- aroylbenzene
- derivatives
- preparation
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10903287A | 1987-10-16 | 1987-10-16 |
Publications (2)
Publication Number | Publication Date |
---|---|
IL88047A0 IL88047A0 (en) | 1989-06-30 |
IL88047A true IL88047A (en) | 1992-11-15 |
Family
ID=22325458
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL88047A IL88047A (en) | 1987-10-16 | 1988-10-14 | Aminomethyl oxooxazolidinyl aroylbenzene derivatives,their preparation and pharmaceutical compositions containing them |
Country Status (20)
Country | Link |
---|---|
EP (1) | EP0312000B1 (no) |
JP (1) | JPH01132570A (no) |
KR (1) | KR890006602A (no) |
AT (1) | ATE73783T1 (no) |
AU (1) | AU617366B2 (no) |
CA (1) | CA1320730C (no) |
DE (1) | DE3869310D1 (no) |
DK (1) | DK573988A (no) |
ES (1) | ES2033394T3 (no) |
FI (1) | FI884755A (no) |
GR (1) | GR3004973T3 (no) |
HU (1) | HU199810B (no) |
IE (1) | IE60426B1 (no) |
IL (1) | IL88047A (no) |
MY (1) | MY103784A (no) |
NO (1) | NO174551C (no) |
NZ (1) | NZ226582A (no) |
PT (1) | PT88765B (no) |
SU (1) | SU1616517A3 (no) |
ZA (1) | ZA887683B (no) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
US5231188A (en) * | 1989-11-17 | 1993-07-27 | The Upjohn Company | Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents |
ATE146783T1 (de) * | 1991-11-01 | 1997-01-15 | Upjohn Co | Substituierte aryl- und heteroaryl- phenyloxazolidinone |
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
EP0673370B1 (en) * | 1992-12-08 | 1998-01-07 | PHARMACIA & UPJOHN COMPANY | Tropone-substituted phenyloxazolidinone antibacterial agents |
US5688792A (en) * | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
NZ274966A (en) * | 1993-11-22 | 1998-01-26 | Upjohn Co | Substituted-hydroxyacetyl piperazine phenyl oxazolidinone derivatives, use in pharmaceutical compositions |
DE4425609A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | Benzofuranyl- und Benzothienyloxazolidinone |
DE4425613A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
DE4425612A1 (de) * | 1994-07-20 | 1996-04-04 | Bayer Ag | 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone |
DE19514313A1 (de) | 1994-08-03 | 1996-02-08 | Bayer Ag | Benzoxazolyl- und Benzothiazolyloxazolidinone |
CN1046520C (zh) * | 1994-11-15 | 1999-11-17 | 法玛西雅厄普约翰美国公司 | 二环噁嗪及噻嗪噁唑烷酮抗菌剂 |
RU2154645C2 (ru) * | 1995-02-03 | 2000-08-20 | Фармация Энд Апджон Компани | Фенилоксазолидиноны, замещенные в кольце гетероароматическими кольцами, в качестве антимикробных агентов |
HRP960159A2 (en) * | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
DE69614847T2 (de) * | 1995-05-11 | 2002-04-04 | Upjohn Co | Spirocyclische und bicyclische diazinyl- und carbazinyloxazolidinone |
MX9703040A (es) * | 1995-09-12 | 1997-07-31 | Upjohn Co | Antimicrobianos de feniloxazolidinona. |
DE19601265A1 (de) * | 1996-01-16 | 1997-07-17 | Bayer Ag | 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone |
GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
HRP970049A2 (en) | 1996-02-06 | 1998-04-30 | Bayer Ag | New heteroaryl oxazolidinones |
DE19604223A1 (de) | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
GB9702213D0 (en) | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
GB9609919D0 (en) | 1996-05-11 | 1996-07-17 | Zeneca Ltd | Chemical compounds |
GB9717804D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
GB9717807D0 (en) | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
EP1007525A1 (en) * | 1997-08-29 | 2000-06-14 | Zeneca Limited | Aminometyl oxooxazolidinyl benzene derivatives |
EP1030852B1 (en) * | 1997-11-12 | 2003-09-17 | PHARMACIA & UPJOHN COMPANY | Oxazolidinone derivatives and pharmaceutical compositions |
GB9725244D0 (en) | 1997-11-29 | 1998-01-28 | Zeneca Ltd | Chemical compounds |
WO1999037630A1 (en) * | 1998-01-23 | 1999-07-29 | Versicor, Inc. | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
US6562844B2 (en) | 1998-01-23 | 2003-05-13 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
US7002020B1 (en) | 1998-01-23 | 2006-02-21 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
AU1379900A (en) * | 1998-11-17 | 2000-06-05 | Bayer Aktiengesellschaft | Novel substituted phenyloxazolidone derivatives |
AU2001269370B2 (en) | 2000-07-17 | 2005-10-27 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
US6956040B2 (en) | 2001-07-16 | 2005-10-18 | Ranbaxy Laboratories Limited | Oxazolidinone piperazinyl derivatives as potential antimicrobials |
KR100854211B1 (ko) | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
CN101220002B (zh) * | 2007-12-28 | 2011-07-13 | 天津药物研究院 | 作为抗菌剂的噁唑烷酮类化合物 |
KR101023174B1 (ko) * | 2008-09-24 | 2011-03-18 | 주식회사 레고켐 바이오사이언스 | 사이클릭 아미독심 또는 사이클릭 아미드라존 기를 가지는 신규한 옥사졸리디논 유도체 및 이를 함유하는 의약 조성물 |
US8604209B2 (en) | 2008-10-10 | 2013-12-10 | Trius Therapeutics, Inc. | Methods for preparing oxazolidinones and compositions containing them |
CN102439006A (zh) | 2009-02-03 | 2012-05-02 | 特留斯治疗学公司 | (r)-3-(4-(2-(2-甲基四唑-5-基)吡啶-5-基)-3-氟苯基)-5-羟甲基噁唑烷-2-酮二氢磷酸酯的晶型 |
US8580767B2 (en) | 2009-05-28 | 2013-11-12 | Trius Therapeutics, Inc. | Oxazolidinone containing dimer compounds, compositions and methods to make and use |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1222708A (en) * | 1968-10-22 | 1971-02-17 | Delalande Sa | Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation |
FR2500450A1 (fr) * | 1981-02-25 | 1982-08-27 | Delalande Sa | Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique |
ES8506659A1 (es) * | 1983-06-07 | 1985-08-01 | Du Pont | Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno. |
CA1260948A (en) * | 1984-12-05 | 1989-09-26 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents |
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
-
1988
- 1988-10-11 CA CA000579796A patent/CA1320730C/en not_active Expired - Fee Related
- 1988-10-12 AT AT88116903T patent/ATE73783T1/de not_active IP Right Cessation
- 1988-10-12 DE DE8888116903T patent/DE3869310D1/de not_active Expired - Fee Related
- 1988-10-12 ES ES198888116903T patent/ES2033394T3/es not_active Expired - Lifetime
- 1988-10-12 EP EP88116903A patent/EP0312000B1/en not_active Expired - Lifetime
- 1988-10-14 FI FI884755A patent/FI884755A/fi not_active Application Discontinuation
- 1988-10-14 JP JP63257417A patent/JPH01132570A/ja active Pending
- 1988-10-14 IE IE311988A patent/IE60426B1/en not_active IP Right Cessation
- 1988-10-14 PT PT88765A patent/PT88765B/pt not_active IP Right Cessation
- 1988-10-14 HU HU885297A patent/HU199810B/hu not_active IP Right Cessation
- 1988-10-14 NZ NZ226582A patent/NZ226582A/xx unknown
- 1988-10-14 KR KR1019880013394A patent/KR890006602A/ko not_active Application Discontinuation
- 1988-10-14 IL IL88047A patent/IL88047A/xx unknown
- 1988-10-14 ZA ZA887683A patent/ZA887683B/xx unknown
- 1988-10-14 SU SU884356643A patent/SU1616517A3/ru active
- 1988-10-14 DK DK573988A patent/DK573988A/da not_active Application Discontinuation
- 1988-10-14 NO NO884594A patent/NO174551C/no unknown
- 1988-10-14 MY MYPI88001159A patent/MY103784A/en unknown
- 1988-10-17 AU AU23962/88A patent/AU617366B2/en not_active Ceased
-
1992
- 1992-06-18 GR GR920401308T patent/GR3004973T3/el unknown
Also Published As
Publication number | Publication date |
---|---|
ATE73783T1 (de) | 1992-04-15 |
HUT49864A (en) | 1989-11-28 |
JPH01132570A (ja) | 1989-05-25 |
NO174551B (no) | 1994-02-14 |
IE60426B1 (en) | 1994-07-13 |
KR890006602A (ko) | 1989-06-14 |
EP0312000A1 (en) | 1989-04-19 |
ZA887683B (en) | 1990-06-27 |
IE883119L (en) | 1989-04-16 |
DE3869310D1 (de) | 1992-04-23 |
CA1320730C (en) | 1993-07-27 |
AU617366B2 (en) | 1991-11-28 |
NO884594L (no) | 1989-04-17 |
PT88765B (pt) | 1992-12-31 |
SU1616517A3 (ru) | 1990-12-23 |
DK573988D0 (da) | 1988-10-14 |
DK573988A (da) | 1989-04-17 |
FI884755A (fi) | 1989-04-17 |
IL88047A0 (en) | 1989-06-30 |
NZ226582A (en) | 1990-06-26 |
AU2396288A (en) | 1989-04-20 |
MY103784A (en) | 1993-09-30 |
HU199810B (en) | 1990-03-28 |
NO174551C (no) | 1994-05-25 |
ES2033394T3 (es) | 1993-03-16 |
NO884594D0 (no) | 1988-10-14 |
EP0312000B1 (en) | 1992-03-18 |
FI884755A0 (fi) | 1988-10-14 |
GR3004973T3 (no) | 1993-04-28 |
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