IL79189A - Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them - Google Patents

Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them

Info

Publication number
IL79189A
IL79189A IL79189A IL7918986A IL79189A IL 79189 A IL79189 A IL 79189A IL 79189 A IL79189 A IL 79189A IL 7918986 A IL7918986 A IL 7918986A IL 79189 A IL79189 A IL 79189A
Authority
IL
Israel
Prior art keywords
sup
acid derivatives
naphthyridine
quinoline
oxo
Prior art date
Application number
IL79189A
Other languages
English (en)
Other versions
IL79189A0 (en
Original Assignee
Daiichi Seiyaku Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co
Publication of IL79189A0 publication Critical patent/IL79189A0/xx
Publication of IL79189A publication Critical patent/IL79189A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Table Devices Or Equipment (AREA)
  • Stringed Musical Instruments (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL79189A 1985-06-26 1986-06-23 Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them IL79189A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP13983085 1985-06-26
JP27999185 1985-12-12

Publications (2)

Publication Number Publication Date
IL79189A0 IL79189A0 (en) 1986-09-30
IL79189A true IL79189A (en) 1990-07-12

Family

ID=26472527

Family Applications (1)

Application Number Title Priority Date Filing Date
IL79189A IL79189A (en) 1985-06-26 1986-06-23 Quinoline and/or naphthyridine-4-oxo-3-carboxylic acid derivatives,process for their preparation and pharmaceutical compositions comprising them

Country Status (18)

Country Link
US (4) US5098912A (de)
EP (1) EP0207420B1 (de)
JP (2) JPH0745491B2 (de)
KR (1) KR930005001B1 (de)
AT (1) ATE75740T1 (de)
AU (1) AU589978B2 (de)
CA (1) CA1301760C (de)
DE (1) DE3685157D1 (de)
DK (1) DK170641B1 (de)
ES (1) ES8707520A1 (de)
FI (1) FI87071C (de)
GR (1) GR861649B (de)
IE (1) IE59188B1 (de)
IL (1) IL79189A (de)
NO (1) NO167090C (de)
PH (1) PH24886A (de)
PT (1) PT82839B (de)
YU (1) YU46526B (de)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3508816A1 (de) * 1985-01-10 1986-07-10 Bayer Ag, 5090 Leverkusen 6,7-disubstituierte 1-cyclopropyl-1,4-dihydro-4-oxo-1,8-naphtyridin-3-carbonsaeuren
US4920120A (en) * 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents
US5585491A (en) * 1988-01-25 1996-12-17 Otsuka Pharmaceutical Co., Ltd. Antibacterial agents
CA1332605C (en) * 1988-10-03 1994-10-18 Yasuhiro Nishitani Pyridonecarboxylic acids
US5364861A (en) * 1990-11-30 1994-11-15 Warner-Lambert Company Optical isomers of 7-[3-(1,1-dialkylmethyl-1-amino-1-pyrrolidinyl]-quinolones and naphthyridones as antibacterial agents
DE69131428T2 (de) * 1990-11-30 2000-01-05 Warner-Lambert Co., Ann Arbor Individuelle stereoisomere von 7-[3-(aminoalkyl)-1-pyrrolidinyl]-quinolone und naphthyridone als antibakterielle wirkstoffe
US5157128A (en) * 1990-11-30 1992-10-20 Warner-Lambert Company Certain optically active substituted α,α-dialkyl-pyrrolidine-3-methamines useful as intermediates
US5258528A (en) * 1990-11-30 1993-11-02 Warner-Lambert Company Individual stereoisomers of pyrrolidine methanamines substituted on the ring nitrogen by a 1-phenylethyl group
EP0550016A1 (de) * 1991-12-31 1993-07-07 Korea Research Institute Of Chemical Technology Chinoloncarbonsäure-Derivate und Verfahren zu ihrer Herstellung
PT807630E (pt) * 1995-02-02 2003-08-29 Daiichi Seiyaku Co Compostos heterociclicos
JP4040091B2 (ja) * 1995-11-22 2008-01-30 第一三共株式会社 置換アミノシクロアルキルピロリジン誘導体
US6121285A (en) 1995-11-22 2000-09-19 Daiichi Pharmaceutical Co., Ltd. Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
AU3459797A (en) 1996-07-12 1998-02-09 Daiichi Pharmaceutical Co., Ltd. Cis-substituted aminocyclopropane derivatives
CN1263527A (zh) * 1997-05-21 2000-08-16 第一制药株式会社 顺式取代－取代氨基环烷基吡咯烷衍生物
MY119816A (en) * 1997-05-30 2005-07-29 Daiichi Seiyaku Co Substituted cyclobutylamine derivatives
US6387928B1 (en) 1997-09-15 2002-05-14 The Procter & Gamble Co. Antimicrobial quinolones, their compositions and uses
CN1264837C (zh) * 1997-09-15 2006-07-19 普罗克特和甘保尔公司 喹诺酮抗微生物剂、其组合物和应用
EP1082300B1 (de) * 1998-05-29 2003-09-10 PHARMACIA & UPJOHN COMPANY 3-[(1'-n-methylamino)ethyl-n-benzyl]pyrrolidin-monomethanesulfonat
CN1258531C (zh) 1999-03-10 2006-06-07 第一制药株式会社 芳香族取代基取代的氨基甲基吡咯烷衍生物
US6569686B2 (en) * 2000-01-28 2003-05-27 Pion, Inc. Measurement of solubility-pH profiles
PT1336611E (pt) * 2000-11-20 2007-12-06 Daiichi Sankyo Co Ltd Compostos desalogenados
PL1666477T3 (pl) 2003-09-10 2013-11-29 Kyorin Seiyaku Kk Pochodna kwasu 7-(4-podstawionego-3-cyklopropyloaminometylo-1- pirolidynylo)chinolonokarboksylowego
WO2005030752A1 (ja) * 2003-09-29 2005-04-07 Daiichi Pharmaceutical Co., Ltd. ８−シアノキノロンカルボン酸誘導体
ES2366150T3 (es) * 2006-03-28 2011-10-17 Warner Chilcott Company, Llc Malatos de polimorfos de ácido (3s,5s)-7-[3-amino-5-metil-piperidinil]-1-ciclopropil-1,4-dihidro-8-metoxi-4-oxo-3-quinolinocarboxílico.
CA2647454A1 (en) * 2006-03-28 2007-10-04 The Procter & Gamble Company A coupling process for preparing quinolone intermediates
BRPI0709209A2 (pt) * 2006-03-28 2011-06-28 Procter & Gamble processo de redução de hidreto para preparo de intermediários de quinolona
JP5322927B2 (ja) * 2007-05-24 2013-10-23 杏林製薬株式会社 １４位置換基に複素芳香環カルボン酸構造を有するムチリン誘導体
CN116606280A (zh) * 2023-03-13 2023-08-18 广东工业大学 一种氟喹诺酮类化合物及其在制备抗菌药物中的应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4665079A (en) * 1984-02-17 1987-05-12 Warner-Lambert Company Antibacterial agents
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
DE3318145A1 (de) * 1983-05-18 1984-11-22 Bayer Ag, 5090 Leverkusen 7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
JPS60228479A (ja) * 1984-04-26 1985-11-13 Toyama Chem Co Ltd １，４−ジヒドロ−４−オキソナフチリジン誘導体およびその塩
IE58742B1 (en) * 1984-07-20 1993-11-05 Warner Lambert Co Substituted-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7h-pyrido[1,2,3-de] [1,4]benzoxauine-6-carboxylic acids; sibstituted-5-amino-6-6fluoro-4-oxo.1,4-dihydroquinoline-3 carboxylic acids; substituted-5-amino-6-fluoro-1,4-dihydro-4-oxo-1.8-naphthyridine-3-carboxylic acids; derivatives thereof; pharmaceutical compositions comprising the compounds; and processes for producing the compounds
DE3509546A1 (de) * 1985-03-16 1986-09-25 Bayer Ag, 5090 Leverkusen 7-amino-1-(subst.cyclopropyl)-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
US4657913A (en) * 1985-04-18 1987-04-14 Warner-Lambert Company Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents
EP0242789A3 (de) * 1986-04-25 1990-09-05 Dainippon Pharmaceutical Co., Ltd. Chinolinderivate und Verfahren zu ihrer Herstellung
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
US4920120A (en) * 1988-01-25 1990-04-24 Warner-Lambert Company Antibacterial agents

Also Published As

Publication number Publication date
FI87071B (fi) 1992-08-14
DK304686A (da) 1987-02-23
JPH09143157A (ja) 1997-06-03
JPS62234082A (ja) 1987-10-14
KR870000321A (ko) 1987-02-17
US5380874A (en) 1995-01-10
EP0207420A3 (en) 1988-04-20
PT82839B (pt) 1988-04-21
US5416222A (en) 1995-05-16
YU46526B (sh) 1993-11-16
EP0207420B1 (de) 1992-05-06
AU589978B2 (en) 1989-10-26
FI87071C (fi) 1992-11-25
IL79189A0 (en) 1986-09-30
AU5924586A (en) 1987-01-08
ATE75740T1 (de) 1992-05-15
PT82839A (en) 1986-07-01
ES556754A0 (es) 1987-08-01
NO167090B (no) 1991-06-24
YU112086A (en) 1991-04-30
IE861696L (en) 1986-12-26
EP0207420A2 (de) 1987-01-07
DE3685157D1 (de) 1992-06-11
NO862559L (no) 1986-12-29
IE59188B1 (en) 1994-01-26
DK304686D0 (da) 1986-06-26
PH24886A (en) 1990-12-26
GR861649B (en) 1986-10-30
FI862688L (fi) 1986-12-27
JPH0745491B2 (ja) 1995-05-17
JP2686705B2 (ja) 1997-12-08
NO862559D0 (no) 1986-06-25
FI862688A0 (fi) 1986-06-24
DK170641B1 (da) 1995-11-20
KR930005001B1 (ko) 1993-06-11
NO167090C (no) 1991-10-02
CA1301760C (en) 1992-05-26
ES8707520A1 (es) 1987-08-01
US5098912A (en) 1992-03-24
US5476950A (en) 1995-12-19

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