IL56028A - Peptides and derivatives thereof exhibiting morphine agonist activity,their preparation and pharmaceutical compositions containing them - Google Patents
Peptides and derivatives thereof exhibiting morphine agonist activity,their preparation and pharmaceutical compositions containing themInfo
- Publication number
- IL56028A IL56028A IL56028A IL5602878A IL56028A IL 56028 A IL56028 A IL 56028A IL 56028 A IL56028 A IL 56028A IL 5602878 A IL5602878 A IL 5602878A IL 56028 A IL56028 A IL 56028A
- Authority
- IL
- Israel
- Prior art keywords
- peptides
- exhibiting
- derivatives
- preparation
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/675—Beta-endorphins
- C07K14/6755—Beta-endorphins with at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/665—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans derived from pro-opiomelanocortin, pro-enkephalin or pro-dynorphin
- C07K14/70—Enkephalins
- C07K14/702—Enkephalins with at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Toxicology (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB48980/77A GB1604850A (en) | 1977-11-24 | 1977-11-24 | Biologically active peptides |
Publications (2)
Publication Number | Publication Date |
---|---|
IL56028A0 IL56028A0 (en) | 1979-01-31 |
IL56028A true IL56028A (en) | 1984-03-30 |
Family
ID=10450679
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL56028A IL56028A (en) | 1977-11-24 | 1978-11-23 | Peptides and derivatives thereof exhibiting morphine agonist activity,their preparation and pharmaceutical compositions containing them |
Country Status (20)
Country | Link |
---|---|
US (5) | US4244944A (de) |
EP (1) | EP0002236B1 (de) |
JP (1) | JPS5492938A (de) |
KR (3) | KR860000453B1 (de) |
AT (1) | AT386211B (de) |
AU (1) | AU530985B2 (de) |
CA (1) | CA1197235A (de) |
DE (1) | DE2862477D1 (de) |
DK (1) | DK149612C (de) |
ES (1) | ES475324A1 (de) |
FI (1) | FI70415C (de) |
GB (1) | GB1604850A (de) |
HU (1) | HU186729B (de) |
IE (1) | IE47517B1 (de) |
IL (1) | IL56028A (de) |
IT (1) | IT1106143B (de) |
MY (1) | MY8500260A (de) |
PL (1) | PL123797B1 (de) |
SU (1) | SU1470199A3 (de) |
ZA (1) | ZA786598B (de) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FI770219A (de) | 1976-02-02 | 1977-08-03 | Sandoz Ag | |
GB1604850A (en) * | 1977-11-24 | 1981-12-16 | Wellcome Found | Biologically active peptides |
DE3163199D1 (en) * | 1980-07-17 | 1984-05-24 | Sandoz Ag | Novel pentapeptides, processes for their production, pharmaceutical compositions comprising said pentapeptides and their use |
ATE16495T1 (de) * | 1981-06-22 | 1985-11-15 | Ici Plc | Peptide und pseudopeptide, die zwei substituenten am n-terminus aufweisen. |
US4380535A (en) * | 1981-09-23 | 1983-04-19 | American Home Products Corporation | Enkephalin degrading enzyme inhibitors |
US4492779A (en) * | 1981-12-07 | 1985-01-08 | Thiokol Corporation | Aramid polymer and powder filler reinforced elastomeric composition for use as a rocket motor insulation |
DE3369327D1 (en) * | 1982-02-05 | 1987-02-26 | Wellcome Found | Pharmaceutical compounds, preparation, use and intermediates therefor and their preparation |
DE3378121D1 (de) * | 1982-10-18 | 1988-11-03 | Ici Plc | Peptide and pseudopeptide derivatives |
JPH0680079B2 (ja) * | 1984-11-09 | 1994-10-12 | エーザイ株式会社 | ポリペプチド |
GB8608818D0 (en) * | 1986-04-11 | 1986-05-14 | Reckitt & Colmann Prod Ltd | Pharmaceutical compositions |
GB8616741D0 (en) * | 1986-07-09 | 1986-08-13 | Wellcome Found | Pharmacologically active compounds |
US5688519A (en) * | 1987-04-06 | 1997-11-18 | Leonard; Robert J. | Flash-flow fused medicinal implants |
US5156787A (en) * | 1991-01-29 | 1992-10-20 | Booher Benjamin V | Pultrusion method of making brake linings |
USRE37548E1 (en) | 1991-08-12 | 2002-02-19 | Bill J. Hays | Clutch design and manufacture |
US5482772A (en) | 1992-12-28 | 1996-01-09 | Kimberly-Clark Corporation | Polymeric strands including a propylene polymer composition and nonwoven fabric and articles made therewith |
US6488649B1 (en) | 1998-11-24 | 2002-12-03 | Edward M. Lichten | Implant device |
IL165365A0 (en) | 2004-11-24 | 2006-01-15 | Q Core Ltd | Finger-type peristaltic pump |
DE112007000840A5 (de) * | 2006-04-21 | 2009-01-02 | Luk Lamellen Und Kupplungsbau Beteiligungs Kg | Mehrschichtiger, insbesondere zweischichtiger Kupplungsbelag sowie Verfahren zu dessen Herstellung |
US8005603B2 (en) | 2007-09-27 | 2011-08-23 | Continental Controls Corporation | Fuel control system and method for gas engines |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1577115A (en) * | 1976-07-27 | 1980-10-22 | Reckitt & Colmann Prod Ltd | Container closure units |
NZ183712A (en) * | 1976-04-08 | 1979-10-25 | Ici Ltd | Polypeptide analogues of enkephalins, and pharmaceutical compositions |
US4028319A (en) * | 1976-05-07 | 1977-06-07 | G. D. Searle & Co. | 2 and 3-substituted enkephalins |
US4123523A (en) * | 1976-06-21 | 1978-10-31 | Imperial Chemical Industries Limited | Analgesic and sedative polypeptides |
FR2359817A1 (fr) * | 1976-07-27 | 1978-02-24 | Reckitt & Colmann Prod Ltd | Nouveaux peptides, leur procede de preparation et composition therapeutique les contenant |
US4092304A (en) * | 1976-08-09 | 1978-05-30 | G. D. Searle & Co. | 4-Substituted enkephalin derivatives |
ZA775285B (en) * | 1976-09-01 | 1978-07-26 | A Kastin | Novel methionine enkephalin derivatives |
HU178001B (en) * | 1976-09-16 | 1982-02-28 | Gyogyszekutato Intezet | Process for preparing new pentapeptides with morphine-like activity and derivatives thereof |
US4128541A (en) * | 1976-12-27 | 1978-12-05 | American Home Products Corporation | Pentapeptide with morphine- like activity |
DE2819277A1 (de) * | 1977-05-16 | 1978-11-23 | Sandoz Ag | Neue polypeptidderivate, ihre herstellung und verwendung |
US4127533A (en) * | 1977-06-16 | 1978-11-28 | Coy David Howard | Novel octapeptides, intermediates therefor, and compositions and methods employing said octapeptides |
US4127523A (en) * | 1977-06-16 | 1978-11-28 | Coy David Howard | Novel undecapeptides, intermediates therefor, and compositions and methods employing said undecapeptides |
US4127532A (en) * | 1977-06-16 | 1978-11-28 | Coy David Howard | Novel heptapeptides, intermediates therefor, and compositions and methods employing said heptapeptides |
US4127531A (en) * | 1977-06-16 | 1978-11-28 | Coy David Howard | Novel hexapeptides, intermediates therefor, and compositions and methods employing said hexapeptides |
GB1604850A (en) * | 1977-11-24 | 1981-12-16 | Wellcome Found | Biologically active peptides |
US4103005A (en) * | 1977-10-20 | 1978-07-25 | Hoffmann-La Roche Inc. | Novel-enkephalin analogs |
-
1977
- 1977-11-24 GB GB48980/77A patent/GB1604850A/en not_active Expired
-
1978
- 1978-07-24 US US05/927,271 patent/US4244944A/en not_active Expired - Lifetime
- 1978-11-22 KR KR7803518A patent/KR860000453B1/ko active
- 1978-11-23 DK DK523078A patent/DK149612C/da not_active IP Right Cessation
- 1978-11-23 AU AU41865/78A patent/AU530985B2/en not_active Expired
- 1978-11-23 IL IL56028A patent/IL56028A/xx unknown
- 1978-11-23 EP EP78101447A patent/EP0002236B1/de not_active Expired
- 1978-11-23 IE IE2317/78A patent/IE47517B1/en unknown
- 1978-11-23 FI FI783589A patent/FI70415C/fi not_active IP Right Cessation
- 1978-11-23 SU SU782691552A patent/SU1470199A3/ru active
- 1978-11-23 HU HU78WE591A patent/HU186729B/hu not_active IP Right Cessation
- 1978-11-23 AT AT0836278A patent/AT386211B/de not_active IP Right Cessation
- 1978-11-23 CA CA000316793A patent/CA1197235A/en not_active Expired
- 1978-11-23 DE DE7878101447T patent/DE2862477D1/de not_active Expired
- 1978-11-23 IT IT52041/78A patent/IT1106143B/it active
- 1978-11-23 PL PL1978211164A patent/PL123797B1/pl unknown
- 1978-11-23 ES ES475324A patent/ES475324A1/es not_active Expired
- 1978-11-24 JP JP14521278A patent/JPS5492938A/ja active Granted
- 1978-11-24 ZA ZA786598A patent/ZA786598B/xx unknown
-
1980
- 1980-09-25 US US06/191,150 patent/US4346083A/en not_active Expired - Lifetime
- 1980-09-25 US US06/190,704 patent/US4343795A/en not_active Expired - Lifetime
- 1980-09-28 US US06/192,071 patent/US4362717A/en not_active Expired - Lifetime
- 1980-09-30 US US06/192,292 patent/US4363800A/en not_active Expired - Lifetime
-
1982
- 1982-08-30 KR KR8203911A patent/KR880002608B1/ko active
- 1982-08-30 KR KR8203912A patent/KR880002609B1/ko active
-
1985
- 1985-12-30 MY MY260/85A patent/MY8500260A/xx unknown
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