IL52203A - Preparation of 3,4-dihydro-2-methyl-4-oxo-2h-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide,and its use as an intermediate in the preparation of the corresponding n-(2-pyridyl)-and n-(2-thiazolyl)carboxamides - Google Patents

Preparation of 3,4-dihydro-2-methyl-4-oxo-2h-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide,and its use as an intermediate in the preparation of the corresponding n-(2-pyridyl)-and n-(2-thiazolyl)carboxamides

Info

Publication number
IL52203A
IL52203A IL52203A IL5220377A IL52203A IL 52203 A IL52203 A IL 52203A IL 52203 A IL52203 A IL 52203A IL 5220377 A IL5220377 A IL 5220377A IL 52203 A IL52203 A IL 52203A
Authority
IL
Israel
Prior art keywords
preparation
benzothiazine
carboxamides
thiazolyl
pyridyl
Prior art date
Application number
IL52203A
Other languages
English (en)
Other versions
IL52203A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL52203A0 publication Critical patent/IL52203A0/xx
Publication of IL52203A publication Critical patent/IL52203A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL52203A 1976-06-10 1977-05-31 Preparation of 3,4-dihydro-2-methyl-4-oxo-2h-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide,and its use as an intermediate in the preparation of the corresponding n-(2-pyridyl)-and n-(2-thiazolyl)carboxamides IL52203A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/694,572 US4100347A (en) 1976-06-10 1976-06-10 3,4-Dihydro-2-methyl-4-oxo-2H-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide

Publications (2)

Publication Number Publication Date
IL52203A0 IL52203A0 (en) 1977-07-31
IL52203A true IL52203A (en) 1979-11-30

Family

ID=24789395

Family Applications (1)

Application Number Title Priority Date Filing Date
IL52203A IL52203A (en) 1976-06-10 1977-05-31 Preparation of 3,4-dihydro-2-methyl-4-oxo-2h-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide,and its use as an intermediate in the preparation of the corresponding n-(2-pyridyl)-and n-(2-thiazolyl)carboxamides

Country Status (37)

Country Link
US (1) US4100347A (ru)
JP (1) JPS5912673B2 (ru)
AR (1) AR215006A1 (ru)
AT (1) AT356126B (ru)
AU (1) AU511643B2 (ru)
BE (1) BE855532A (ru)
BG (1) BG41307A3 (ru)
CA (1) CA1077934A (ru)
CH (1) CH634312A5 (ru)
CS (2) CS191347B2 (ru)
CY (1) CY1128A (ru)
DD (2) DD132014A5 (ru)
DE (1) DE2726175A1 (ru)
DK (1) DK147337C (ru)
EG (1) EG12644A (ru)
ES (2) ES459601A1 (ru)
FI (1) FI62297C (ru)
FR (1) FR2354325A1 (ru)
GB (2) GB1544359A (ru)
GR (1) GR66969B (ru)
HK (2) HK31381A (ru)
HU (1) HU184665B (ru)
IE (1) IE44997B1 (ru)
IL (1) IL52203A (ru)
LU (1) LU77516A1 (ru)
MY (2) MY8100269A (ru)
NL (1) NL7706338A (ru)
NO (1) NO150761C (ru)
NZ (1) NZ184249A (ru)
PH (1) PH14751A (ru)
PL (2) PL108606B1 (ru)
PT (1) PT66639B (ru)
RO (2) RO77179A (ru)
SE (1) SE442200B (ru)
SU (2) SU657747A3 (ru)
YU (1) YU39493B (ru)
ZA (1) ZA773248B (ru)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2756113A1 (de) * 1977-12-16 1979-06-21 Thomae Gmbh Dr K Neue 4-hydroxy-2h-1,2-benzothiazin- 3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4434164A (en) 1981-06-01 1984-02-28 Pfizer Inc. Crystalline benzothiazine dioxide salts
US4474955A (en) * 1981-06-17 1984-10-02 Vincenzo Iannella Process for preparing 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-[N-(2-pyridinyl)carboxamide]-1,1-dioxide, and its phosphoric ester
IN159273B (ru) * 1981-10-05 1987-04-25 Pfizer
ATE31309T1 (de) * 1982-07-07 1987-12-15 Siegfried Ag Verfahren zur herstellung von 4-hydroxy-2-methyln-2-pyridyl-2h-1,2-benzothiazin-3-carboxamid 1,1- dioxid.
DE3311165A1 (de) * 1983-03-26 1984-09-27 Gödecke AG, 1000 Berlin Feinkristallines isoxicam
IT1194522B (it) * 1983-12-16 1988-09-22 Prodotti Antibiotici Spa Metodo di sintesi di derivanti benzotiazinici
US4530272A (en) * 1984-01-13 1985-07-23 International Business Machines Corporation Method for controlling contamination in a clean room
US5741798A (en) * 1996-06-03 1998-04-21 Boehringer Ingelheim Pharmaceuticals, Inc. 2-benzyl-4-sulfonyl-4H-isoquinolin-1,3-diones and their use as antiinflammatory agents

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3501466A (en) * 1967-11-30 1970-03-17 Mcneilab Inc 3-carbamoyl and 3-alkoxycarbonyl benzothiazine-1,1-dioxides
US3492298A (en) * 1968-02-21 1970-01-27 Mcneilab Inc Oxazino-benzothiazine-6,6-dioxides
US3591584A (en) * 1968-08-27 1971-07-06 Pfizer Benzothiazine dioxides
US3808205A (en) * 1971-09-10 1974-04-30 Warner Lambert Co Process for the preparation of 4-hydroxy-3-carbamyl-2h-1,2-benzothiazine 1,1-dioxides and 4-hydroxy-3(2h)-1,2-benzothiazine carboxylate-1,1-dioxides
US3853862A (en) * 1973-04-23 1974-12-10 Pfizer Production of 4-hydroxy-1,2-benzothiazine-3-carboxamides
US3892740A (en) * 1974-10-15 1975-07-01 Pfizer Process for the production of carboxamides of oxo-1,2-benzothiazine-1,1-dioxides
US3991584A (en) 1975-01-31 1976-11-16 Western Gear Corporation Shock absorbing and retracting system for pipe laying vessel
US3960856A (en) * 1975-06-20 1976-06-01 Warner-Lambert Company Process for the preparation of 4-hydroxy-3-(5-methyl-3-isoxazolylcarbamoyl)-2-methyl-2H-1,2-benzothiazine 1,1-dioxide

Also Published As

Publication number Publication date
DE2726175A1 (de) 1977-12-22
SE7706078L (sv) 1977-12-11
BG41307A3 (en) 1987-05-15
GB1544358A (en) 1979-04-19
AR215006A1 (es) 1979-08-31
CY1128A (en) 1982-02-19
IL52203A0 (en) 1977-07-31
YU39493B (en) 1984-12-31
PT66639A (en) 1977-07-01
RO77179A (ro) 1981-06-22
NO150761C (no) 1984-12-12
ES459601A1 (es) 1978-04-01
ZA773248B (en) 1978-04-26
EG12644A (en) 1979-06-30
US4100347A (en) 1978-07-11
IE44997L (en) 1977-12-10
GR66969B (ru) 1981-05-15
DK147337C (da) 1985-01-14
PL108606B1 (en) 1980-04-30
JPS5912673B2 (ja) 1984-03-24
RO70629A (ro) 1981-01-30
PL104307B1 (pl) 1979-08-31
FI771799A (ru) 1977-12-11
DD132014A5 (de) 1978-08-16
FR2354325B1 (ru) 1981-10-30
ATA412177A (de) 1979-09-15
IE44997B1 (en) 1982-06-02
FI62297B (fi) 1982-08-31
NZ184249A (en) 1978-11-13
GB1544359A (en) 1979-04-19
LU77516A1 (ru) 1979-01-19
HU184665B (en) 1984-09-28
ES462973A1 (es) 1978-06-16
NO771870L (no) 1977-12-13
AU2566677A (en) 1978-12-07
PL198768A1 (pl) 1978-04-10
PH14751A (en) 1981-11-20
HK31281A (en) 1981-07-10
NL7706338A (nl) 1977-12-13
CH634312A5 (de) 1983-01-31
JPS52151180A (en) 1977-12-15
MY8100274A (en) 1981-12-31
CS191341B2 (en) 1979-06-29
DK255577A (da) 1977-12-11
FR2354325A1 (fr) 1978-01-06
AU511643B2 (en) 1980-08-28
SU657747A3 (ru) 1979-04-15
NO150761B (no) 1984-09-03
AT356126B (de) 1980-04-10
YU134877A (en) 1982-08-31
CS191347B2 (en) 1979-06-29
FI62297C (fi) 1982-12-10
HK31381A (en) 1981-07-10
SE442200B (sv) 1985-12-09
SU833159A3 (ru) 1981-05-23
CA1077934A (en) 1980-05-20
PT66639B (en) 1978-11-09
BE855532A (fr) 1977-12-09
DD137104A5 (de) 1979-08-15
MY8100269A (en) 1981-12-31
DK147337B (da) 1984-06-25

Similar Documents

Publication Publication Date Title
NL7803036A (nl) 4-(5-fluormethyl-2-pyridyloxy)fenoxyalkaan- carbonzuren en derivaten daarvan.
IL52257A (en) 4-(3,4-dihydroxy-epoxy-5-hydroxy-methylhexyl-tetrahydropyran)-2-yl-3-methylbut-2e-enoic acid and its preparation
NZ185105A (en) Thiazolidine derivatives and pharmaceutical compositions
NZ183150A (en) 7-aminothiazolyl-iminoa-cetamido-cephalosporin derivatives and pharmaceutical compositions
IL51581A (en) 5,6-bis-phenyl-2,3-diydro-imidazo(2,1-b)thiazole derivatives their preparation and pharmaceutical compositions containg them
PH16512A (en) N-(phenylalkylamino-alkyl)-dihydroisoquinolinones,pharmaceutical compositions and methods employing them
IL51403A0 (en) 1,2-dithiole derivatives processes for the preparation thereof and pharmaceutical compositions containing the same
NZ183134A (en) I-i-(3-aryloxy-2-hydroxypropyl)-4-piperidyl-3-aryl-imid-azolidin or hexahydropyrimidin-2-ones; and pharmaceutical compositions
IL52203A (en) Preparation of 3,4-dihydro-2-methyl-4-oxo-2h-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide,and its use as an intermediate in the preparation of the corresponding n-(2-pyridyl)-and n-(2-thiazolyl)carboxamides
IL51402A0 (en) 1,2-dithiole derivatives processes for the preparation thereof and pharmaceutical compositions containing the same
ZA772075B (en) Novel 1,3,4-thiadiazolyl derivatives and their use as herbicides
NZ184263A (en) N-(amino-alkyl-amino)-benzamides and pharmaceutical compositions
JPS5289669A (en) Thiazolidine derivatives and preparation thereof
IL48009A (en) 2,3-dihydro-3-oxothienoisothiazole 1,1-dioxide derivatives and their manufacture
AU505649B2 (en) N-(1, 3, 4-thiadiazol-2-yl) benzamides
JPS5362834A (en) Pharmaceutical composition and use thereof
IL51955A0 (en) Novel thiazole derivatives their preparation and pharmaceutical compositions containing them
NZ184634A (en) N-(i'allyl-2-pyrrolidylmethyl)-2,3-dimethoxy-5-sulphamoyl-benzamide and pharmaceutical compositions
PH12590A (en) 4a-aryl octahydro-1h-2-pyrindines and pharmaceutical composition thereof
JPS5320433A (en) Pharmaceutical composition and application
JPS5293764A (en) Novel cysteine derivatives and preparation thereof
NZ184084A (en) 2-carboxyalkyl-pyrrolid-in or piperidin-one or-dione derivatives and pharmaceutical compositions
NZ185295A (en) 9-chloroprednisolone derivatives and pharmaceutical compositions
PH12050A (en) Benzisothiazoline-1,1-dioxide derivatives,compositions and methods of use thereof
NZ185996A (en) 6, 7-methylene-3-oxo-d-homo-17a-pregna-4, 16-dienes and pharmaceutical compositions