IL44906A - Derivatives of 1,3-disubstituted 2,4 (1h,3h)-quinazolinediones - Google Patents

Derivatives of 1,3-disubstituted 2,4 (1h,3h)-quinazolinediones

Info

Publication number
IL44906A
IL44906A IL44906A IL4490674A IL44906A IL 44906 A IL44906 A IL 44906A IL 44906 A IL44906 A IL 44906A IL 4490674 A IL4490674 A IL 4490674A IL 44906 A IL44906 A IL 44906A
Authority
IL
Israel
Prior art keywords
propyl
phenyl
quinazolinedione
piperazinyl
compound
Prior art date
Application number
IL44906A
Other languages
English (en)
Other versions
IL44906A0 (en
Original Assignee
Miles Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Miles Lab filed Critical Miles Lab
Publication of IL44906A0 publication Critical patent/IL44906A0/xx
Publication of IL44906A publication Critical patent/IL44906A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL44906A 1973-06-18 1974-05-28 Derivatives of 1,3-disubstituted 2,4 (1h,3h)-quinazolinediones IL44906A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US371277A US3879393A (en) 1973-06-18 1973-06-18 Derivatives of 1,3-disubstituted 2,4(1h,3h)-quinazolinediones

Publications (2)

Publication Number Publication Date
IL44906A0 IL44906A0 (en) 1974-07-31
IL44906A true IL44906A (en) 1977-12-30

Family

ID=23463289

Family Applications (1)

Application Number Title Priority Date Filing Date
IL44906A IL44906A (en) 1973-06-18 1974-05-28 Derivatives of 1,3-disubstituted 2,4 (1h,3h)-quinazolinediones

Country Status (9)

Country Link
US (1) US3879393A (de)
AU (1) AU470731B2 (de)
CA (1) CA1016170A (de)
DE (1) DE2428858A1 (de)
FR (1) FR2233063B1 (de)
GB (1) GB1467471A (de)
IL (1) IL44906A (de)
NL (1) NL7407910A (de)
ZA (1) ZA743366B (de)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4058612A (en) * 1974-12-02 1977-11-15 Schering Corporation 6-(Polyhaloisopropyl)quinazoline-2,4-diones
EP0040793B1 (de) * 1980-05-22 1985-08-28 Masayuki Ishikawa Chinazolindion-Verbindungen, Verfahren zu deren Herstellung und deren pharmazeutische Verwendung
US5969079A (en) * 1985-09-05 1999-10-19 The Boeing Company Oligomers with multiple chemically functional end caps
US5210213A (en) * 1983-06-17 1993-05-11 The Boeing Company Dimensional, crosslinkable oligomers
US5714566A (en) * 1981-11-13 1998-02-03 The Boeing Company Method for making multiple chemically functional oligomers
US5521014A (en) * 1981-11-13 1996-05-28 The Boeing Company Extended multidimensional ether or ester oligomers
US5512676A (en) * 1987-09-03 1996-04-30 The Boeing Company Extended amideimide hub for multidimensional oligomers
US5705598A (en) 1985-04-23 1998-01-06 The Boeing Company Polyester sulfone oligomers and blends
US5693741A (en) * 1988-03-15 1997-12-02 The Boeing Company Liquid molding compounds
JPS58159480A (ja) * 1982-03-17 1983-09-21 Chugai Pharmaceut Co Ltd 新規なフエニルピペラジン誘導体
JPS608274A (ja) * 1983-06-27 1985-01-17 Fujisawa Pharmaceut Co Ltd 新規キナゾリノン誘導体およびその製造法・並びに抗アレルギ−剤
US4639518A (en) * 1984-09-24 1987-01-27 Ortho Pharmaceutical Corporation Substituted quinazolinediones
DE3563964D1 (en) * 1984-10-16 1988-09-01 Synthelabo Piperidine derivatives, their preparation and their therapeutical application
US5618907A (en) * 1985-04-23 1997-04-08 The Boeing Company Thallium catalyzed multidimensional ester oligomers
US5817744A (en) * 1988-03-14 1998-10-06 The Boeing Company Phenylethynyl capped imides
US6521630B1 (en) 1999-08-31 2003-02-18 Pfizer Inc. Tetrahydroquinazoline-2,4-diones and therapeutic uses thereof
DE10101324C1 (de) * 2001-01-13 2001-12-13 Ibfb Gmbh Privates Inst Fuer B 1-Dimercaptoalkylchinazolin-2,4-(1H,3H)-dione als Matrix-Metalloproteinase(MMP)-Inhibitoren
DE60235400D1 (de) * 2001-12-04 2010-04-01 Active Implants Corp Kissenlagerungsimplantate für lasttragende anwendungen
EP1687277B1 (de) 2003-11-20 2018-04-04 Janssen Pharmaceutica NV 6-alkenyl- und 6-phenylalkylsubstituierte 2-chinolinone und 2-chinoxalinone als poly(adp-ribose)-polymerase-inhibitoren
CN1882549B (zh) * 2003-11-20 2011-02-23 詹森药业有限公司 用作聚(adp-核糖)聚合酶抑制剂的7-苯基烷基取代的2-喹啉酮和2-喹喔啉酮
UA89618C2 (ru) * 2003-12-05 2010-02-25 Янссен Фармацевтика Н.В. 6-замещенные 2-хинолиноны и 2-хиноксалиноны как ингибиторы поли(адф-рибоза)полимеразы
EP1771175B1 (de) * 2004-06-30 2015-12-23 Janssen Pharmaceutica NV Phthalazin-derivate als parp-hemmer
NZ551801A (en) * 2004-06-30 2009-11-27 Janssen Pharmaceutica Nv Quinazolinedione derivatives as PARP inhibitors
AU2005259188B2 (en) 2004-06-30 2011-03-31 Janssen Pharmaceutica N.V. Quinazolinone derivatives as PARP inhibitors
AU2007208139B2 (en) 2006-01-24 2012-09-27 Janssen Pharmaceutica N.V. 2-substituted benzimidazoles as selective androgen receptor modulators (sarms)
DK2134691T3 (da) 2007-03-08 2012-05-07 Janssen Pharmaceutica Nv Quinolinonderivativer som parp- og tank-inhibitorer
US8107260B2 (en) * 2007-11-15 2012-01-31 Illinois Tool Works Inc. EMI shielding and environmental seal device
EP2271626B1 (de) 2008-03-27 2014-11-26 Janssen Pharmaceutica, N.V. Tetrahydrophenanthridinone und tetrahydrocyclopentachinolinone als parp- und tubulinpolymerisierungshemmer
WO2010099503A1 (en) 2009-02-26 2010-09-02 Reviva Pharmaceuticals, Inc. Compositions, synthesis, and methods of utilizing quinazolinedione derivatives
FR2944206B1 (fr) * 2009-04-09 2012-12-28 Sanofi Aventis Applications therapeutiques dans le domaine cardiovasculaire de derives de quinazolinedione
FR2944282B1 (fr) 2009-04-09 2013-05-03 Sanofi Aventis Derives de quinazolinedione, leur preparation et leurs diverses applications therapeutiques
EP3174864A4 (de) * 2014-07-31 2018-02-14 Oregon Health & Science University Vmat-hemmende verbindungen

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3274194A (en) * 1963-03-29 1966-09-20 Miles Lab Quinazolinedione derivatives
DE1803210A1 (de) * 1968-10-16 1970-05-14 Troponwerke Dinklage & Co 2-Methyl-3-(3-[4-phenylpiperazinyl-(1)]-2-hydroxypropyl)-chinazolinon-(4) und Verfahren zu seiner Herstellung
DE1934037A1 (de) * 1969-07-04 1971-01-07 Cassella Farbwerke Mainkur Ag Basisch substituierte Derivate des 2,4-(1H,3H)-Chinazolindions

Also Published As

Publication number Publication date
US3879393A (en) 1975-04-22
GB1467471A (en) 1977-03-16
AU470731B2 (en) 1976-03-25
AU6945074A (en) 1975-12-04
CA1016170A (en) 1977-08-23
FR2233063B1 (de) 1978-07-28
NL7407910A (de) 1974-12-20
ZA743366B (en) 1975-05-28
FR2233063A1 (de) 1975-01-10
IL44906A0 (en) 1974-07-31
DE2428858A1 (de) 1975-01-09

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