IL319327A - Methods of administering corticosteroids - Google Patents

Methods of administering corticosteroids

Info

Publication number
IL319327A
IL319327A IL319327A IL31932725A IL319327A IL 319327 A IL319327 A IL 319327A IL 319327 A IL319327 A IL 319327A IL 31932725 A IL31932725 A IL 31932725A IL 319327 A IL319327 A IL 319327A
Authority
IL
Israel
Prior art keywords
urinary
dose
hsd
inhibitor
composition
Prior art date
Application number
IL319327A
Other languages
English (en)
Hebrew (he)
Inventor
a katz David
Original Assignee
Sparrow Pharmaceuticals Inc
a katz David
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sparrow Pharmaceuticals Inc, a katz David filed Critical Sparrow Pharmaceuticals Inc
Publication of IL319327A publication Critical patent/IL319327A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4196—1,2,4-Triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P39/00—General protective or antinoxious agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Toxicology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
IL319327A 2018-11-20 2019-08-14 Methods of administering corticosteroids IL319327A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862769932P 2018-11-20 2018-11-20
PCT/US2019/046449 WO2020106337A1 (en) 2018-11-20 2019-08-14 Methods for administering corticosteroids

Publications (1)

Publication Number Publication Date
IL319327A true IL319327A (en) 2025-05-01

Family

ID=70774135

Family Applications (2)

Application Number Title Priority Date Filing Date
IL319327A IL319327A (en) 2018-11-20 2019-08-14 Methods of administering corticosteroids
IL283069A IL283069B2 (en) 2018-11-20 2019-08-14 Methods of administering corticosteroids

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL283069A IL283069B2 (en) 2018-11-20 2019-08-14 Methods of administering corticosteroids

Country Status (10)

Country Link
US (2) US12220412B2 (cg-RX-API-DMAC7.html)
EP (1) EP3883578A4 (cg-RX-API-DMAC7.html)
JP (2) JP7472122B2 (cg-RX-API-DMAC7.html)
CN (1) CN113329754A (cg-RX-API-DMAC7.html)
AU (2) AU2019384074B2 (cg-RX-API-DMAC7.html)
BR (1) BR112021009653A2 (cg-RX-API-DMAC7.html)
CA (1) CA3120339A1 (cg-RX-API-DMAC7.html)
IL (2) IL319327A (cg-RX-API-DMAC7.html)
MX (2) MX2021005801A (cg-RX-API-DMAC7.html)
WO (1) WO2020106337A1 (cg-RX-API-DMAC7.html)

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WO2022076398A1 (en) * 2020-10-07 2022-04-14 Surface Ophthalmics, Inc. Pharmaceutical kits and their use for treating dry eye disease
CN113329754A (zh) 2018-11-20 2021-08-31 麻雀制药股份有限公司 用于施用皮质类固醇的方法
JP2022516099A (ja) 2018-12-27 2022-02-24 サーフィス オフサルミクス，インコーポレイテッド 眼科用医薬組成物及び癌表面疾患の処置方法
BR112021015481A2 (pt) * 2019-02-08 2021-12-07 Sanofi Sa Otimização biotecnológica de micro-organismos para a 1,2-desidrogenação de esteroides
CN117979951A (zh) 2021-05-10 2024-05-03 瑟菲斯眼科股份有限公司 一种用于缓解眼部疼痛的硫酸软骨素的用途
US12440510B2 (en) 2021-05-10 2025-10-14 Surface Ophthalmics, Inc. Use of chondroitin sulfate for relieving ocular pain
IL316907A (en) * 2022-05-16 2025-01-01 Sparrow Pharmaceuticals Inc METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOD EXCESS
AU2024348222A1 (en) * 2023-09-27 2026-04-16 Sparrow Pharmaceuticals, Inc. Methods and compositions for treating glucocorticoid-mediated diseases
GB202408335D0 (en) 2024-06-11 2024-07-24 Astrazeneca Ab Therapies for wound treatment

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Also Published As

Publication number Publication date
US20250205227A1 (en) 2025-06-26
US20210393622A1 (en) 2021-12-23
CA3120339A1 (en) 2020-05-28
WO2020106337A1 (en) 2020-05-28
MX2021005801A (es) 2021-08-05
EP3883578A4 (en) 2022-07-27
CN113329754A (zh) 2021-08-31
BR112021009653A2 (pt) 2021-08-17
MX2025002836A (es) 2025-04-02
JP2022507103A (ja) 2022-01-18
IL283069B1 (en) 2025-05-01
JP7472122B2 (ja) 2024-04-22
IL283069A (en) 2021-06-30
EP3883578A1 (en) 2021-09-29
US12220412B2 (en) 2025-02-11
AU2025203033A1 (en) 2025-05-22
JP2024098991A (ja) 2024-07-24
AU2019384074B2 (en) 2025-04-10
IL283069B2 (en) 2025-09-01
AU2019384074A1 (en) 2021-06-03

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Subfigure Supplementary Figure 3. Overview of all conducted experiments where mineralocorticoid receptor agonists and mineralocorticoid receptor antagonists were administered.