IL238453A0 - Trans-clomiphene for use in cancer treatment - Google Patents

Trans-clomiphene for use in cancer treatment

Info

Publication number
IL238453A0
IL238453A0 IL238453A IL23845315A IL238453A0 IL 238453 A0 IL238453 A0 IL 238453A0 IL 238453 A IL238453 A IL 238453A IL 23845315 A IL23845315 A IL 23845315A IL 238453 A0 IL238453 A0 IL 238453A0
Authority
IL
Israel
Prior art keywords
clomiphene
trans
cancer therapy
cancer
therapy
Prior art date
Application number
IL238453A
Other languages
English (en)
Hebrew (he)
Original Assignee
Repros Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Repros Therapeutics Inc filed Critical Repros Therapeutics Inc
Publication of IL238453A0 publication Critical patent/IL238453A0/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
IL238453A 2012-11-02 2015-04-26 Trans-clomiphene for use in cancer treatment IL238453A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261722013P 2012-11-02 2012-11-02
PCT/US2013/066141 WO2014070523A1 (en) 2012-11-02 2013-10-22 Trans-clomiphene for use in cancer therapy

Publications (1)

Publication Number Publication Date
IL238453A0 true IL238453A0 (en) 2015-06-30

Family

ID=50627954

Family Applications (1)

Application Number Title Priority Date Filing Date
IL238453A IL238453A0 (en) 2012-11-02 2015-04-26 Trans-clomiphene for use in cancer treatment

Country Status (10)

Country Link
US (1) US9687458B2 (enExample)
EP (1) EP2914294A1 (enExample)
JP (3) JP2015535283A (enExample)
CN (1) CN104994877A (enExample)
AU (1) AU2013338311A1 (enExample)
CA (1) CA2889770A1 (enExample)
HK (1) HK1216502A1 (enExample)
IL (1) IL238453A0 (enExample)
MX (1) MX2015005160A (enExample)
WO (1) WO2014070523A1 (enExample)

Families Citing this family (6)

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US20170217914A1 (en) * 2014-08-05 2017-08-03 The Penn State Research Foundation Novel Triarylethylene Compounds and Methods Using Same
US11633382B2 (en) 2015-11-10 2023-04-25 Paracrine Therapeutics Ab Treatment of ER-negative breast cancer with an PDGF-CC inhibitor and anti-estrogen
JP2018002619A (ja) * 2016-06-29 2018-01-11 国立大学法人 東京大学 オートファジー阻害剤
US20200030259A1 (en) * 2016-09-26 2020-01-30 Repros Therapeutics Inc. Antiestrogens and/or Aromatase Inhibitors for Use in Treating Obesity and Related Symptoms
CN108420806A (zh) * 2017-02-15 2018-08-21 武汉华杰世纪生物医药有限公司 具有靶向性的抗肿瘤药物
WO2019236209A2 (en) * 2018-04-27 2019-12-12 Jin Byung Ju Methods for high-content drug screening

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Also Published As

Publication number Publication date
WO2014070523A1 (en) 2014-05-08
EP2914294A1 (en) 2015-09-09
US20150283099A1 (en) 2015-10-08
JP2021046448A (ja) 2021-03-25
CA2889770A1 (en) 2014-05-08
AU2013338311A1 (en) 2015-05-14
CN104994877A (zh) 2015-10-21
JP2018123168A (ja) 2018-08-09
MX2015005160A (es) 2015-07-17
HK1216502A1 (zh) 2016-11-18
US9687458B2 (en) 2017-06-27
JP2015535283A (ja) 2015-12-10

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