IL201627A - Process for Preparation of 6 - {4 - [3 - ((r) -2 - Methyl-Pyrrolidine-1-Il) -Propoxy] -Phenyl} -2H-Pyridazine-3-On - Google Patents
Process for Preparation of 6 - {4 - [3 - ((r) -2 - Methyl-Pyrrolidine-1-Il) -Propoxy] -Phenyl} -2H-Pyridazine-3-OnInfo
- Publication number
- IL201627A IL201627A IL201627A IL20162709A IL201627A IL 201627 A IL201627 A IL 201627A IL 201627 A IL201627 A IL 201627A IL 20162709 A IL20162709 A IL 20162709A IL 201627 A IL201627 A IL 201627A
- Authority
- IL
- Israel
- Prior art keywords
- methylpyrrolidine
- tartrate
- methyl
- phenyl
- propoxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/06—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with radicals, containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Cosmetics (AREA)
- Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US92735607P | 2007-05-03 | 2007-05-03 | |
| PCT/US2008/005702 WO2008137087A1 (en) | 2007-05-03 | 2008-05-02 | Processes for preparing (r)-2-methylpyrrolidine and (s)-2-methylpyrrolidine and tartrate salts thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| IL201627A0 IL201627A0 (en) | 2010-05-31 |
| IL201627A true IL201627A (en) | 2014-06-30 |
Family
ID=39688886
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL201627A IL201627A (en) | 2007-05-03 | 2009-10-19 | Process for Preparation of 6 - {4 - [3 - ((r) -2 - Methyl-Pyrrolidine-1-Il) -Propoxy] -Phenyl} -2H-Pyridazine-3-On |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP2152669A1 (pt) |
| JP (1) | JP5698887B2 (pt) |
| KR (1) | KR20100017565A (pt) |
| CN (1) | CN101679237A (pt) |
| AU (1) | AU2008248168B2 (pt) |
| BR (1) | BRPI0810330A2 (pt) |
| CA (1) | CA2686033A1 (pt) |
| EA (1) | EA019031B1 (pt) |
| IL (1) | IL201627A (pt) |
| MX (1) | MX2009011787A (pt) |
| NZ (1) | NZ580948A (pt) |
| UA (1) | UA99913C2 (pt) |
| WO (1) | WO2008137087A1 (pt) |
| ZA (1) | ZA200907643B (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL2069312T3 (pl) | 2006-07-25 | 2013-03-29 | Cephalon Inc | Pochodne pirydazynonu |
| US8383657B2 (en) | 2007-12-21 | 2013-02-26 | Abbott Laboratories | Thiazolylidine urea and amide derivatives and methods of use thereof |
| ES2479440T3 (es) * | 2008-01-30 | 2014-07-24 | Cephalon, Inc. | Derivados de piridazina sustituidos que tienen actividad antagonista de histamina H3 |
| JP6849594B2 (ja) * | 2014-12-23 | 2021-03-24 | セファロン、インク． | 縮合二環式２，４−ジアミノピリミジン誘導体を調整する方法 |
Family Cites Families (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3329974A1 (de) | 1983-08-19 | 1985-02-28 | Bayer Ag, 5090 Leverkusen | Herstellung von hydrierten nitrilkautschuken |
| DE3433392A1 (de) | 1984-09-12 | 1986-03-20 | Bayer Ag, 5090 Leverkusen | Hydrierung nitrilgruppenhaltiger ungesaettigter polymerer |
| FR2714849B1 (fr) | 1994-01-13 | 1996-04-05 | Inst Francais Du Petrole | Procédé de préparation d'un catalyseur d'hydrogénation soluble en phase liquide organique. |
| DE4403479A1 (de) | 1994-02-04 | 1995-08-10 | Basf Ag | Verfahren zur Herstellung von Hydroxylammoniumsalzen |
| WO2004024707A2 (en) * | 2002-09-16 | 2004-03-25 | Abbott Laboratories | Process for preparing amine type substituted benzofurans |
| US7153889B2 (en) | 2002-11-12 | 2006-12-26 | Abbott Laboratories | Bicyclic-substituted amines as histamine-3 receptor ligands |
| US8110519B2 (en) | 2004-03-08 | 2012-02-07 | Japan Science & Technology Agency | Polymer-supported metal cluster composition |
| US7145005B2 (en) | 2004-05-12 | 2006-12-05 | Abbott Laboratories | 2-(6-{2-[(2R)-2-Methyl-1-pyrrolidin-1-yl]-ethyl}-2-naphthalen-2-yl)-2H-pyridazin-3-one salts and their preparation |
| PL1755593T3 (pl) | 2004-06-02 | 2008-06-30 | Hoffmann La Roche | Pochodne naftalenu przydatne jako ligandy 3-receptora histaminowego |
| US8158652B2 (en) | 2004-12-01 | 2012-04-17 | Msd K.K. | Substituted pyridone derivative |
| DE602005026169D1 (de) | 2004-12-17 | 2011-03-10 | Janssen Pharmaceutica Nv | Tetrahydroisochinolinverbindungen zur behandlung von zns-erkrankungen |
| JP2008526895A (ja) | 2005-01-21 | 2008-07-24 | シェーリング コーポレイション | ヒスタミンｈ３アンタゴニストとして有用なイミダゾールおよびベンゾイミダゾール誘導体 |
| WO2006103045A1 (en) | 2005-03-31 | 2006-10-05 | Ucb Pharma S.A. | Compounds comprising an oxazole or thiazole moiety, processes for making them, and their uses |
| GB0514812D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
| US7943605B2 (en) | 2005-10-27 | 2011-05-17 | Ucb Pharma S.A. | Compounds comprising a lactam or a lactam derivative moiety, processes for making them, and their uses |
| WO2007094962A2 (en) | 2006-02-09 | 2007-08-23 | Athersys, Inc. | Pyrazoles for the treatment of obesity and other cns disorders |
| WO2007099423A1 (en) | 2006-03-02 | 2007-09-07 | Pfizer Products Inc. | 1-pyrrolidine indane derivatives as histamine-3 receptor antagonists |
| WO2007105053A2 (en) | 2006-03-13 | 2007-09-20 | Pfizer Products Inc. | Tetralines antagonists of the h-3 receptor |
| WO2008005338A1 (en) | 2006-06-29 | 2008-01-10 | Arena Pharmaceuticals, Inc. | Modulators of the histamine h3-receptor useful for the treatment of disorders related thereto |
| PL2069312T3 (pl) * | 2006-07-25 | 2013-03-29 | Cephalon Inc | Pochodne pirydazynonu |
-
2008
- 2008-05-02 BR BRPI0810330-5A2A patent/BRPI0810330A2/pt not_active IP Right Cessation
- 2008-05-02 MX MX2009011787A patent/MX2009011787A/es active IP Right Grant
- 2008-05-02 KR KR1020097025141A patent/KR20100017565A/ko not_active Application Discontinuation
- 2008-05-02 NZ NZ580948A patent/NZ580948A/en not_active IP Right Cessation
- 2008-05-02 AU AU2008248168A patent/AU2008248168B2/en not_active Ceased
- 2008-05-02 EP EP08754205A patent/EP2152669A1/en not_active Withdrawn
- 2008-05-02 CN CN200880021225A patent/CN101679237A/zh active Pending
- 2008-05-02 WO PCT/US2008/005702 patent/WO2008137087A1/en active Application Filing
- 2008-05-02 EA EA200971019A patent/EA019031B1/ru not_active IP Right Cessation
- 2008-05-02 UA UAA200912476A patent/UA99913C2/ru unknown
- 2008-05-02 JP JP2010507416A patent/JP5698887B2/ja not_active Expired - Fee Related
- 2008-05-02 CA CA002686033A patent/CA2686033A1/en not_active Abandoned
-
2009
- 2009-10-19 IL IL201627A patent/IL201627A/en not_active IP Right Cessation
- 2009-10-30 ZA ZA2009/07643A patent/ZA200907643B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EA019031B1 (ru) | 2013-12-30 |
| ZA200907643B (en) | 2014-03-26 |
| EA200971019A1 (ru) | 2010-04-30 |
| UA99913C2 (ru) | 2012-10-25 |
| JP5698887B2 (ja) | 2015-04-08 |
| KR20100017565A (ko) | 2010-02-16 |
| EP2152669A1 (en) | 2010-02-17 |
| JP2010526142A (ja) | 2010-07-29 |
| CA2686033A1 (en) | 2008-11-13 |
| WO2008137087A1 (en) | 2008-11-13 |
| CN101679237A (zh) | 2010-03-24 |
| BRPI0810330A2 (pt) | 2014-10-14 |
| AU2008248168A1 (en) | 2008-11-13 |
| AU2008248168B2 (en) | 2013-03-21 |
| MX2009011787A (es) | 2009-11-13 |
| NZ580948A (en) | 2011-04-29 |
| IL201627A0 (en) | 2010-05-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FF | Patent granted | ||
| KB | Patent renewed | ||
| MM9K | Patent not in force due to non-payment of renewal fees |