IL165505A0 - 2-heteroaryl carboxamides - Google Patents
2-heteroaryl carboxamidesInfo
- Publication number
- IL165505A0 IL165505A0 IL16550504A IL16550504A IL165505A0 IL 165505 A0 IL165505 A0 IL 165505A0 IL 16550504 A IL16550504 A IL 16550504A IL 16550504 A IL16550504 A IL 16550504A IL 165505 A0 IL165505 A0 IL 165505A0
- Authority
- IL
- Israel
- Prior art keywords
- heteroaryl carboxamides
- carboxamides
- heteroaryl
- prophylaxis
- learning
- Prior art date
Links
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 230000008447 perception Effects 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10225536 | 2002-06-10 | ||
| DE10257078A DE10257078A1 (de) | 2002-12-06 | 2002-12-06 | 2-Heteroarylcarbonsäureamide |
| DE2002157537 DE10257537A1 (de) | 2002-12-10 | 2002-12-10 | 2-Heteroarylcarbonsäureamide |
| DE10305922A DE10305922A1 (de) | 2002-06-10 | 2003-02-13 | 2-Heteroarylcarbonsäureamide |
| PCT/EP2003/005735 WO2003104227A1 (de) | 2002-01-20 | 2003-06-02 | 2-heteroarylcarbonsäureamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL165505A0 true IL165505A0 (en) | 2006-01-15 |
Family
ID=29740887
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL16550504A IL165505A0 (en) | 2002-06-10 | 2004-12-02 | 2-heteroaryl carboxamides |
Country Status (16)
| Country | Link |
|---|---|
| US (5) | US7977485B2 (enExample) |
| EP (1) | EP1515967B1 (enExample) |
| JP (1) | JP4542891B2 (enExample) |
| CN (1) | CN1675204A (enExample) |
| AT (1) | ATE344262T1 (enExample) |
| AU (1) | AU2003238450A1 (enExample) |
| BR (1) | BR0312446A (enExample) |
| CA (1) | CA2488761C (enExample) |
| DE (1) | DE50305587D1 (enExample) |
| ES (1) | ES2276072T3 (enExample) |
| IL (1) | IL165505A0 (enExample) |
| MX (1) | MXPA04012439A (enExample) |
| NO (1) | NO20050063L (enExample) |
| PL (1) | PL374551A1 (enExample) |
| UY (1) | UY27841A1 (enExample) |
| WO (1) | WO2003104227A1 (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10164139A1 (de) | 2001-12-27 | 2003-07-10 | Bayer Ag | 2-Heteroarylcarbonsäureamide |
| ATE344262T1 (de) * | 2002-06-10 | 2006-11-15 | Bayer Healthcare Ag | 2-heteroarylcarbonsäureamide |
| AU2003276919B2 (en) | 2002-09-25 | 2013-05-16 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof |
| DE602004031124D1 (de) | 2003-08-13 | 2011-03-03 | Neurosearch As | Neue chinuklidinderivative und deren pharmazeutische verwendung |
| WO2005063767A2 (en) | 2003-12-22 | 2005-07-14 | Memory Pharmaceuticals Corporation | Indoles, 1h-indazoles, 1,2-benzisoxazoles, and 1,2-benzisothiazoles, and preparation and uses thereof |
| US20050234095A1 (en) | 2004-03-25 | 2005-10-20 | Wenge Xie | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
| US7514450B2 (en) | 2004-05-19 | 2009-04-07 | Neurosearch A/S | Azabicyclic aryl derivatives |
| CN100588657C (zh) | 2004-10-15 | 2010-02-10 | 神经研究公司 | 新的氮杂双环芳基衍生物及其医药用途 |
| US8106066B2 (en) * | 2005-09-23 | 2012-01-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof |
| CN101910159B (zh) | 2007-12-26 | 2013-06-19 | 卫材R&D管理有限公司 | 杂环取代吡啶衍生物的制备方法 |
| US8367676B2 (en) * | 2009-06-30 | 2013-02-05 | Astrazeneca Ab | 2-carboxamide-7-piperazinyl-benzofuran derivatives 774 |
| JP5749797B2 (ja) | 2010-05-17 | 2015-07-15 | フォルム ファーマシューティカルズ、インコーポレイテッド | (r)−7−クロロ−n−(キヌクリジン−3−イル)ベンゾ[b]チオフェン−2−カルボキサミド塩酸塩一水和物の結晶形 |
| KR20130132932A (ko) | 2010-12-20 | 2013-12-05 | 아스트라제네카 아베 | 2-카르복스아미드-4-피페라지닐-벤조푸란 유도체 |
| KR101928505B1 (ko) * | 2011-01-28 | 2018-12-12 | 에스케이바이오팜 주식회사 | 피리돈 유도체 및 이를 포함하는 약학적 조성물 |
| CA2872005A1 (en) | 2012-05-08 | 2013-11-14 | Forum Pharmaceuticals, Inc. | Methods of maintaining, treating or improving cognitive function |
| CN111205283A (zh) * | 2020-01-20 | 2020-05-29 | 广州九植医药科技有限公司 | 一种盐酸帕洛诺司琼有关物质b的合成方法 |
| CN111205284A (zh) * | 2020-01-20 | 2020-05-29 | 广州九植医药科技有限公司 | 一种盐酸帕洛诺司琼有关物质a的合成方法 |
| EP4213832A4 (en) * | 2020-09-18 | 2024-10-16 | Merck Sharp & Dohme LLC | Modified benzofuran-carboxamides as glucosylceramide synthase inhibitors |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0000540D0 (sv) * | 2000-02-18 | 2000-02-18 | Astrazeneca Ab | New compounds |
| JP4616971B2 (ja) * | 2000-07-18 | 2011-01-19 | 田辺三菱製薬株式会社 | 1−アザビシクロアルカン化合物およびその医薬用途 |
| AR036040A1 (es) | 2001-06-12 | 2004-08-04 | Upjohn Co | Compuestos de heteroarilo multiciclicos sustituidos con quinuclidinas y composiciones farmaceuticas que los contienen |
| EA007429B1 (ru) | 2001-10-02 | 2006-10-27 | Фармация Энд Апджон Компани | Азабициклические замещённые конденсированные гетероарильные соединения |
| DE10164139A1 (de) | 2001-12-27 | 2003-07-10 | Bayer Ag | 2-Heteroarylcarbonsäureamide |
| ATE344262T1 (de) * | 2002-06-10 | 2006-11-15 | Bayer Healthcare Ag | 2-heteroarylcarbonsäureamide |
| DE10234424A1 (de) | 2002-07-29 | 2004-02-12 | Bayer Ag | Benzothiophen-, Benzofuran- und Indolharnstoffe |
-
2003
- 2003-06-02 AT AT03732517T patent/ATE344262T1/de not_active IP Right Cessation
- 2003-06-02 AU AU2003238450A patent/AU2003238450A1/en not_active Abandoned
- 2003-06-02 CA CA2488761A patent/CA2488761C/en not_active Expired - Fee Related
- 2003-06-02 PL PL03374551A patent/PL374551A1/xx not_active Application Discontinuation
- 2003-06-02 MX MXPA04012439A patent/MXPA04012439A/es unknown
- 2003-06-02 CN CNA038188511A patent/CN1675204A/zh active Pending
- 2003-06-02 US US10/516,777 patent/US7977485B2/en not_active Expired - Fee Related
- 2003-06-02 BR BR0312446-0A patent/BR0312446A/pt not_active Application Discontinuation
- 2003-06-02 EP EP03732517A patent/EP1515967B1/de not_active Expired - Lifetime
- 2003-06-02 JP JP2004511297A patent/JP4542891B2/ja not_active Expired - Fee Related
- 2003-06-02 WO PCT/EP2003/005735 patent/WO2003104227A1/de not_active Ceased
- 2003-06-02 ES ES03732517T patent/ES2276072T3/es not_active Expired - Lifetime
- 2003-06-02 DE DE50305587T patent/DE50305587D1/de not_active Expired - Lifetime
- 2003-06-10 UY UY27841A patent/UY27841A1/es not_active Application Discontinuation
-
2004
- 2004-12-02 IL IL16550504A patent/IL165505A0/xx unknown
-
2005
- 2005-01-06 NO NO20050063A patent/NO20050063L/no not_active Application Discontinuation
-
2011
- 2011-07-11 US US13/179,957 patent/US20110263591A1/en not_active Abandoned
-
2012
- 2012-03-06 US US13/412,946 patent/US20120258964A1/en not_active Abandoned
-
2014
- 2014-04-25 US US14/261,616 patent/US9067931B2/en not_active Expired - Fee Related
-
2015
- 2015-06-08 US US14/733,804 patent/US10214524B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US20060160877A1 (en) | 2006-07-20 |
| UY27841A1 (es) | 2003-12-31 |
| PL374551A1 (en) | 2005-10-31 |
| NO20050063L (no) | 2005-01-06 |
| US20120258964A1 (en) | 2012-10-11 |
| US7977485B2 (en) | 2011-07-12 |
| US10214524B2 (en) | 2019-02-26 |
| CA2488761C (en) | 2011-05-31 |
| WO2003104227A1 (de) | 2003-12-18 |
| EP1515967B1 (de) | 2006-11-02 |
| AU2003238450A1 (en) | 2003-12-22 |
| US20160122337A1 (en) | 2016-05-05 |
| BR0312446A (pt) | 2005-04-19 |
| CN1675204A (zh) | 2005-09-28 |
| JP4542891B2 (ja) | 2010-09-15 |
| US20140350008A1 (en) | 2014-11-27 |
| MXPA04012439A (es) | 2005-04-19 |
| JP2005533052A (ja) | 2005-11-04 |
| DE50305587D1 (en) | 2006-12-14 |
| EP1515967A1 (de) | 2005-03-23 |
| US9067931B2 (en) | 2015-06-30 |
| ATE344262T1 (de) | 2006-11-15 |
| ES2276072T3 (es) | 2007-06-16 |
| CA2488761A1 (en) | 2003-12-18 |
| US20110263591A1 (en) | 2011-10-27 |
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