ATE344262T1 - 2-heteroarylcarbonsäureamide - Google Patents

2-heteroarylcarbonsäureamide

Info

Publication number
ATE344262T1
ATE344262T1 AT03732517T AT03732517T ATE344262T1 AT E344262 T1 ATE344262 T1 AT E344262T1 AT 03732517 T AT03732517 T AT 03732517T AT 03732517 T AT03732517 T AT 03732517T AT E344262 T1 ATE344262 T1 AT E344262T1
Authority
AT
Austria
Prior art keywords
heteroaryl
carbonic acid
acid amides
prophylaxis
learning
Prior art date
Application number
AT03732517T
Other languages
German (de)
English (en)
Inventor
Joachim Luithle
Frank-Gerhard Boess
Christina Erb
Frank-Thorsten Hafner
Katrin Schnizler
Timo Flessner
Kampen Marja Van
Der Staay Franz-Josef Van
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10257078A external-priority patent/DE10257078A1/de
Priority claimed from DE2002157537 external-priority patent/DE10257537A1/de
Priority claimed from DE10305922A external-priority patent/DE10305922A1/de
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Application granted granted Critical
Publication of ATE344262T1 publication Critical patent/ATE344262T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
AT03732517T 2002-06-10 2003-06-02 2-heteroarylcarbonsäureamide ATE344262T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE10225536 2002-06-10
DE10257078A DE10257078A1 (de) 2002-12-06 2002-12-06 2-Heteroarylcarbonsäureamide
DE2002157537 DE10257537A1 (de) 2002-12-10 2002-12-10 2-Heteroarylcarbonsäureamide
DE10305922A DE10305922A1 (de) 2002-06-10 2003-02-13 2-Heteroarylcarbonsäureamide

Publications (1)

Publication Number Publication Date
ATE344262T1 true ATE344262T1 (de) 2006-11-15

Family

ID=29740887

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03732517T ATE344262T1 (de) 2002-06-10 2003-06-02 2-heteroarylcarbonsäureamide

Country Status (16)

Country Link
US (5) US7977485B2 (enExample)
EP (1) EP1515967B1 (enExample)
JP (1) JP4542891B2 (enExample)
CN (1) CN1675204A (enExample)
AT (1) ATE344262T1 (enExample)
AU (1) AU2003238450A1 (enExample)
BR (1) BR0312446A (enExample)
CA (1) CA2488761C (enExample)
DE (1) DE50305587D1 (enExample)
ES (1) ES2276072T3 (enExample)
IL (1) IL165505A0 (enExample)
MX (1) MXPA04012439A (enExample)
NO (1) NO20050063L (enExample)
PL (1) PL374551A1 (enExample)
UY (1) UY27841A1 (enExample)
WO (1) WO2003104227A1 (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10164139A1 (de) 2001-12-27 2003-07-10 Bayer Ag 2-Heteroarylcarbonsäureamide
ATE344262T1 (de) * 2002-06-10 2006-11-15 Bayer Healthcare Ag 2-heteroarylcarbonsäureamide
AU2003276919B2 (en) 2002-09-25 2013-05-16 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof
DE602004031124D1 (de) 2003-08-13 2011-03-03 Neurosearch As Neue chinuklidinderivative und deren pharmazeutische verwendung
WO2005063767A2 (en) 2003-12-22 2005-07-14 Memory Pharmaceuticals Corporation Indoles, 1h-indazoles, 1,2-benzisoxazoles, and 1,2-benzisothiazoles, and preparation and uses thereof
US20050234095A1 (en) 2004-03-25 2005-10-20 Wenge Xie Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof
US7514450B2 (en) 2004-05-19 2009-04-07 Neurosearch A/S Azabicyclic aryl derivatives
CN100588657C (zh) 2004-10-15 2010-02-10 神经研究公司 新的氮杂双环芳基衍生物及其医药用途
US8106066B2 (en) * 2005-09-23 2012-01-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
CN101910159B (zh) 2007-12-26 2013-06-19 卫材R&D管理有限公司 杂环取代吡啶衍生物的制备方法
US8367676B2 (en) * 2009-06-30 2013-02-05 Astrazeneca Ab 2-carboxamide-7-piperazinyl-benzofuran derivatives 774
JP5749797B2 (ja) 2010-05-17 2015-07-15 フォルム ファーマシューティカルズ、インコーポレイテッド (r)−7−クロロ−n−(キヌクリジン−3−イル)ベンゾ[b]チオフェン−2−カルボキサミド塩酸塩一水和物の結晶形
KR20130132932A (ko) 2010-12-20 2013-12-05 아스트라제네카 아베 2-카르복스아미드-4-피페라지닐-벤조푸란 유도체
KR101928505B1 (ko) * 2011-01-28 2018-12-12 에스케이바이오팜 주식회사 피리돈 유도체 및 이를 포함하는 약학적 조성물
CA2872005A1 (en) 2012-05-08 2013-11-14 Forum Pharmaceuticals, Inc. Methods of maintaining, treating or improving cognitive function
CN111205283A (zh) * 2020-01-20 2020-05-29 广州九植医药科技有限公司 一种盐酸帕洛诺司琼有关物质b的合成方法
CN111205284A (zh) * 2020-01-20 2020-05-29 广州九植医药科技有限公司 一种盐酸帕洛诺司琼有关物质a的合成方法
EP4213832A4 (en) * 2020-09-18 2024-10-16 Merck Sharp & Dohme LLC Modified benzofuran-carboxamides as glucosylceramide synthase inhibitors

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0000540D0 (sv) * 2000-02-18 2000-02-18 Astrazeneca Ab New compounds
JP4616971B2 (ja) * 2000-07-18 2011-01-19 田辺三菱製薬株式会社 1−アザビシクロアルカン化合物およびその医薬用途
AR036040A1 (es) 2001-06-12 2004-08-04 Upjohn Co Compuestos de heteroarilo multiciclicos sustituidos con quinuclidinas y composiciones farmaceuticas que los contienen
EA007429B1 (ru) 2001-10-02 2006-10-27 Фармация Энд Апджон Компани Азабициклические замещённые конденсированные гетероарильные соединения
DE10164139A1 (de) 2001-12-27 2003-07-10 Bayer Ag 2-Heteroarylcarbonsäureamide
ATE344262T1 (de) * 2002-06-10 2006-11-15 Bayer Healthcare Ag 2-heteroarylcarbonsäureamide
DE10234424A1 (de) 2002-07-29 2004-02-12 Bayer Ag Benzothiophen-, Benzofuran- und Indolharnstoffe

Also Published As

Publication number Publication date
US20060160877A1 (en) 2006-07-20
UY27841A1 (es) 2003-12-31
PL374551A1 (en) 2005-10-31
NO20050063L (no) 2005-01-06
US20120258964A1 (en) 2012-10-11
US7977485B2 (en) 2011-07-12
US10214524B2 (en) 2019-02-26
CA2488761C (en) 2011-05-31
WO2003104227A1 (de) 2003-12-18
EP1515967B1 (de) 2006-11-02
AU2003238450A1 (en) 2003-12-22
US20160122337A1 (en) 2016-05-05
BR0312446A (pt) 2005-04-19
CN1675204A (zh) 2005-09-28
JP4542891B2 (ja) 2010-09-15
IL165505A0 (en) 2006-01-15
US20140350008A1 (en) 2014-11-27
MXPA04012439A (es) 2005-04-19
JP2005533052A (ja) 2005-11-04
DE50305587D1 (en) 2006-12-14
EP1515967A1 (de) 2005-03-23
US9067931B2 (en) 2015-06-30
ES2276072T3 (es) 2007-06-16
CA2488761A1 (en) 2003-12-18
US20110263591A1 (en) 2011-10-27

Similar Documents

Publication Publication Date Title
ATE344262T1 (de) 2-heteroarylcarbonsäureamide
WO2003055878A8 (de) 2-heteroarylcarbonsäureamide
NL300933I2 (nl) Letermovir
ATE370968T1 (de) Varianten des menschliche koagulationsfaktors vii
DE50310516D1 (de) Fredericamycin-derivate
ATE365720T1 (de) Agonisten von beta-adrenorezeptoren
DK1411932T3 (da) Kombinationsterapi med substituerede oxazolidinoner
CY1107054T1 (el) Ενωσεις διτοσυλικου αλατος κιναζολινης
WO2003078431A8 (de) Aza- bicyclische n-biarylamide mit affinität zum alpha7 nikotinischen acetylcholin-rezeptor
DE60318839D1 (de) 2,6-chinolinyl- und 2,6-naphthylderivate und deren verwendungen zur behandlung von vla-4 bezogenen krankheiten
CY1113116T1 (el) Υποκατεστημενες 4-αμινοκυκλοεξανολες
WO2003078430A8 (de) Essig- und propionsäureamide
MA28613B1 (fr) Macrocycles d'amide antibacteriens
ATE338036T1 (de) Zur behandlung hyperproliferativer erkrankungen geeignete benzofuran- und benzothiophenderivate
BR0209541A (pt) Uso das imidazotriazinonas 2-fenil-substituìdas
NO20055741L (no) Nye kjemiske forbindelser
DE602004023721D1 (de) Zusammensetzungen und methoden für die behandlung von herzerkrankungen
ECSP055844A (es) Nuevos compuestos triciclicos
EP1494696A4 (en) TREATMENT OF PULMONARY DISORDERS
UA86399C2 (ru) Применение 2,5 дигидроксибензолсульфоновой кислоты для изготовления лекарства, которые применяют для лечения болезней, зависимых от ангиогенеза
DE602004026597D1 (de) Behandlung von alzheimer-krankheit und verwandten zuständen
DE502004012196D1 (de) Verwendung von isorhamnetin zur behandlung von depressiven verstimmungen und erkrankungen
ATE359270T1 (de) Phenyl-piperidin-4-yliden-methyl-benzamidderiva e zur behandlung von schmerz oder magen-darm- erkrankungen
HUP0102116A2 (hu) Paroxetin-aszkorbát, eljárás az előállítására és gyógyászati alkalmazása
UY27475A1 (es) Amidas de ácido piperazinciclohexanocarboxílico sustituidas y su utilización

Legal Events

Date Code Title Description
REN Ceased due to non-payment of the annual fee