ATE344262T1 - 2-heteroarylcarbonsäureamide - Google Patents

2-heteroarylcarbonsäureamide

Info

Publication number
ATE344262T1
ATE344262T1 AT03732517T AT03732517T ATE344262T1 AT E344262 T1 ATE344262 T1 AT E344262T1 AT 03732517 T AT03732517 T AT 03732517T AT 03732517 T AT03732517 T AT 03732517T AT E344262 T1 ATE344262 T1 AT E344262T1
Authority
AT
Austria
Prior art keywords
heteroaryl
carbonic acid
acid amides
prophylaxis
learning
Prior art date
Application number
AT03732517T
Other languages
German (de)
English (en)
Inventor
Joachim Luithle
Frank-Gerhard Boess
Christina Erb
Frank-Thorsten Hafner
Katrin Schnizler
Timo Flessner
Kampen Marja Van
Der Staay Franz-Josef Van
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10257078A external-priority patent/DE10257078A1/de
Priority claimed from DE2002157537 external-priority patent/DE10257537A1/de
Priority claimed from DE10305922A external-priority patent/DE10305922A1/de
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Application granted granted Critical
Publication of ATE344262T1 publication Critical patent/ATE344262T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
AT03732517T 2002-06-10 2003-06-02 2-heteroarylcarbonsäureamide ATE344262T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE10225536 2002-06-10
DE10257078A DE10257078A1 (de) 2002-12-06 2002-12-06 2-Heteroarylcarbonsäureamide
DE2002157537 DE10257537A1 (de) 2002-12-10 2002-12-10 2-Heteroarylcarbonsäureamide
DE10305922A DE10305922A1 (de) 2002-06-10 2003-02-13 2-Heteroarylcarbonsäureamide

Publications (1)

Publication Number Publication Date
ATE344262T1 true ATE344262T1 (de) 2006-11-15

Family

ID=29740887

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03732517T ATE344262T1 (de) 2002-06-10 2003-06-02 2-heteroarylcarbonsäureamide

Country Status (16)

Country Link
US (5) US7977485B2 (enExample)
EP (1) EP1515967B1 (enExample)
JP (1) JP4542891B2 (enExample)
CN (1) CN1675204A (enExample)
AT (1) ATE344262T1 (enExample)
AU (1) AU2003238450A1 (enExample)
BR (1) BR0312446A (enExample)
CA (1) CA2488761C (enExample)
DE (1) DE50305587D1 (enExample)
ES (1) ES2276072T3 (enExample)
IL (1) IL165505A0 (enExample)
MX (1) MXPA04012439A (enExample)
NO (1) NO20050063L (enExample)
PL (1) PL374551A1 (enExample)
UY (1) UY27841A1 (enExample)
WO (1) WO2003104227A1 (enExample)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10164139A1 (de) 2001-12-27 2003-07-10 Bayer Ag 2-Heteroarylcarbonsäureamide
ES2276072T3 (es) * 2002-06-10 2007-06-16 Bayer Healthcare Ag Amidas de acidos 2-heteroarilcarboxilicos.
CA2499128C (en) 2002-09-25 2012-07-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, and benzoisothiazoles, and preparation and uses thereof
WO2005016923A1 (en) 2003-08-13 2005-02-24 Neurosearch A/S Novel quinuclidine derivatives and their pharmaceutical use
PL1697378T3 (pl) 2003-12-22 2008-04-30 Memory Pharm Corp Indole, 1h-indazole, 1,2-benzoizoksazole i 1,2-benzoizotiazole oraz ich wytwarzanie i zastosowania
WO2005092890A2 (en) 2004-03-25 2005-10-06 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof
US7514450B2 (en) 2004-05-19 2009-04-07 Neurosearch A/S Azabicyclic aryl derivatives
CA2584836A1 (en) 2004-10-15 2006-04-20 Neurosearch A/S Novel azabicyclic aryl derivatives and their medical use
US8106066B2 (en) * 2005-09-23 2012-01-31 Memory Pharmaceuticals Corporation Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof
WO2009081970A1 (ja) * 2007-12-26 2009-07-02 Eisai R & D Management Co., Ltd. ヘテロ環置換ピリジン誘導体の製造方法
US8367676B2 (en) * 2009-06-30 2013-02-05 Astrazeneca Ab 2-carboxamide-7-piperazinyl-benzofuran derivatives 774
TWI519532B (zh) 2010-05-17 2016-02-01 艾維沃製藥公司 （Ｒ）－７－氯－Ｎ－（啶－３－基）苯並［b］噻吩－２－羧醯胺鹽酸鹽單水合物之結晶形體
CA2821480A1 (en) 2010-12-20 2012-06-28 Astrazeneca Ab 2-carboxamide-4-piperazinyl-benzofuran derivative
KR101928505B1 (ko) * 2011-01-28 2018-12-12 에스케이바이오팜 주식회사 피리돈 유도체 및 이를 포함하는 약학적 조성물
RU2017136693A (ru) 2012-05-08 2019-02-08 Форум Фармасьютикалз, Инк. Способы поддержания, лечения или улучшения когнитивной функции
CN111205283A (zh) * 2020-01-20 2020-05-29 广州九植医药科技有限公司 一种盐酸帕洛诺司琼有关物质b的合成方法
CN111205284A (zh) * 2020-01-20 2020-05-29 广州九植医药科技有限公司 一种盐酸帕洛诺司琼有关物质a的合成方法
EP4213832A4 (en) * 2020-09-18 2024-10-16 Merck Sharp & Dohme LLC Modified benzofuran-carboxamides as glucosylceramide synthase inhibitors

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0000540D0 (sv) * 2000-02-18 2000-02-18 Astrazeneca Ab New compounds
JP4616971B2 (ja) * 2000-07-18 2011-01-19 田辺三菱製薬株式会社 １−アザビシクロアルカン化合物およびその医薬用途
AR036040A1 (es) * 2001-06-12 2004-08-04 Upjohn Co Compuestos de heteroarilo multiciclicos sustituidos con quinuclidinas y composiciones farmaceuticas que los contienen
CZ2004408A3 (cs) * 2001-10-02 2005-03-16 Pharmacia & Upjohn Company Azabicyklicky substituované kondenzované heteroarylsloučeniny
DE10164139A1 (de) 2001-12-27 2003-07-10 Bayer Ag 2-Heteroarylcarbonsäureamide
ES2276072T3 (es) * 2002-06-10 2007-06-16 Bayer Healthcare Ag Amidas de acidos 2-heteroarilcarboxilicos.
DE10234424A1 (de) 2002-07-29 2004-02-12 Bayer Ag Benzothiophen-, Benzofuran- und Indolharnstoffe

Also Published As

Publication number Publication date
AU2003238450A1 (en) 2003-12-22
NO20050063L (no) 2005-01-06
US20160122337A1 (en) 2016-05-05
US20140350008A1 (en) 2014-11-27
MXPA04012439A (es) 2005-04-19
UY27841A1 (es) 2003-12-31
CA2488761A1 (en) 2003-12-18
CA2488761C (en) 2011-05-31
CN1675204A (zh) 2005-09-28
EP1515967B1 (de) 2006-11-02
JP4542891B2 (ja) 2010-09-15
US10214524B2 (en) 2019-02-26
PL374551A1 (en) 2005-10-31
WO2003104227A1 (de) 2003-12-18
US20110263591A1 (en) 2011-10-27
US9067931B2 (en) 2015-06-30
US7977485B2 (en) 2011-07-12
US20060160877A1 (en) 2006-07-20
IL165505A0 (en) 2006-01-15
ES2276072T3 (es) 2007-06-16
BR0312446A (pt) 2005-04-19
DE50305587D1 (en) 2006-12-14
JP2005533052A (ja) 2005-11-04
US20120258964A1 (en) 2012-10-11
EP1515967A1 (de) 2005-03-23

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