IL160707A0 - 1, 8-naphthyridine derivatives as antidiabetics - Google Patents

1, 8-naphthyridine derivatives as antidiabetics

Info

Publication number
IL160707A0
IL160707A0 IL16070702A IL16070702A IL160707A0 IL 160707 A0 IL160707 A0 IL 160707A0 IL 16070702 A IL16070702 A IL 16070702A IL 16070702 A IL16070702 A IL 16070702A IL 160707 A0 IL160707 A0 IL 160707A0
Authority
IL
Israel
Prior art keywords
antidiabetics
naphthyridine derivatives
naphthyridine
derivatives
Prior art date
Application number
IL16070702A
Other languages
English (en)
Original Assignee
Bayer Pharmaceuticals Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharmaceuticals Corp filed Critical Bayer Pharmaceuticals Corp
Publication of IL160707A0 publication Critical patent/IL160707A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/10—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH
    • A61P5/12—Drugs for disorders of the endocrine system of the posterior pituitary hormones, e.g. oxytocin, ADH for decreasing, blocking or antagonising the activity of the posterior pituitary hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/42—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of mineralocorticosteroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
IL16070702A 2001-09-26 2002-09-23 1, 8-naphthyridine derivatives as antidiabetics IL160707A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US32451101P 2001-09-26 2001-09-26
PCT/US2002/030176 WO2003027112A1 (en) 2001-09-26 2002-09-23 1, 8-naphthyridine derivatives as antidiabetics

Publications (1)

Publication Number Publication Date
IL160707A0 true IL160707A0 (en) 2004-08-31

Family

ID=23263913

Family Applications (2)

Application Number Title Priority Date Filing Date
IL16070702A IL160707A0 (en) 2001-09-26 2002-09-23 1, 8-naphthyridine derivatives as antidiabetics
IL16070802A IL160708A0 (en) 2001-09-26 2002-09-23 1, 6-naphthyridine derivatives as antidiabetics

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL16070802A IL160708A0 (en) 2001-09-26 2002-09-23 1, 6-naphthyridine derivatives as antidiabetics

Country Status (24)

Country Link
US (5) US6900205B2 (xx)
EP (2) EP1432711A1 (xx)
JP (2) JP2005504807A (xx)
KR (2) KR20040041178A (xx)
CN (2) CN1578781A (xx)
AR (2) AR037503A1 (xx)
BR (2) BR0212864A (xx)
CA (2) CA2463039A1 (xx)
CO (2) CO5560542A2 (xx)
EC (2) ECSP045084A (xx)
GT (2) GT200200191A (xx)
HN (1) HN2002000275A (xx)
HR (2) HRP20040309A2 (xx)
HU (2) HUP0402310A2 (xx)
IL (2) IL160707A0 (xx)
MA (2) MA27079A1 (xx)
MX (2) MXPA04002136A (xx)
NO (2) NO20041560L (xx)
PE (2) PE20030601A1 (xx)
PL (2) PL369567A1 (xx)
RU (2) RU2004112787A (xx)
UY (2) UY27457A1 (xx)
WO (2) WO2003027113A1 (xx)
ZA (2) ZA200403064B (xx)

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IL160708A0 (en) 2004-08-31
GT200200194A (es) 2003-07-03
US20040014751A1 (en) 2004-01-22
EP1432710A1 (en) 2004-06-30
HRP20040317A2 (en) 2006-06-30
AR037503A1 (es) 2004-11-17
JP2005504807A (ja) 2005-02-17
JP2005504808A (ja) 2005-02-17
RU2004112787A (ru) 2005-10-10
NO20041560L (no) 2004-05-11
US20040157875A1 (en) 2004-08-12
US7109196B2 (en) 2006-09-19
MA26344A1 (fr) 2004-10-01
HN2002000275A (es) 2005-02-22
BR0212829A (pt) 2004-08-03
MXPA04002035A (es) 2004-06-07
CA2463039A1 (en) 2003-04-03
CO5560542A2 (es) 2005-09-30
ECSP045084A (es) 2004-06-28
CA2461132A1 (en) 2003-04-03
HUP0401889A2 (hu) 2005-01-28
US6677352B1 (en) 2004-01-13
US6964971B2 (en) 2005-11-15
WO2003027112A1 (en) 2003-04-03
EP1432711A1 (en) 2004-06-30
CO5560611A2 (es) 2005-09-30
KR20040041177A (ko) 2004-05-14
MA27079A1 (fr) 2004-12-20
BR0212864A (pt) 2004-08-17
PE20030549A1 (es) 2003-08-18
AR037504A1 (es) 2004-11-17
PL369567A1 (en) 2005-05-02
ZA200403064B (en) 2005-06-29
UY27457A1 (es) 2003-04-30
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PL369531A1 (en) 2005-05-02
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NO20041567L (no) 2004-05-11
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CN1578781A (zh) 2005-02-09
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US20060189609A1 (en) 2006-08-24
US20040209866A1 (en) 2004-10-21
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