IL160084A0 - Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity - Google Patents

Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity

Info

Publication number
IL160084A0
IL160084A0 IL16008402A IL16008402A IL160084A0 IL 160084 A0 IL160084 A0 IL 160084A0 IL 16008402 A IL16008402 A IL 16008402A IL 16008402 A IL16008402 A IL 16008402A IL 160084 A0 IL160084 A0 IL 160084A0
Authority
IL
Israel
Prior art keywords
thieno
pyrimidines
combined
agonistic activity
fsh agonistic
Prior art date
Application number
IL16008402A
Other languages
English (en)
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of IL160084A0 publication Critical patent/IL160084A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A61P5/08—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH for decreasing, blocking or antagonising the activity of the anterior pituitary hormones

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL16008402A 2001-09-04 2002-08-29 Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity IL160084A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01203327 2001-09-04
PCT/EP2002/009647 WO2003020726A1 (en) 2001-09-04 2002-08-29 Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity

Publications (1)

Publication Number Publication Date
IL160084A0 true IL160084A0 (en) 2004-06-20

Family

ID=8180876

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16008402A IL160084A0 (en) 2001-09-04 2002-08-29 Thieno [2,3-d] pyrimidines with combined la and fsh agonistic activity

Country Status (28)

Country Link
US (1) US7317006B2 (hu)
EP (1) EP1427733B1 (hu)
JP (1) JP4262092B2 (hu)
KR (1) KR100900018B1 (hu)
CN (1) CN1246324C (hu)
AR (1) AR036407A1 (hu)
AT (1) ATE345345T1 (hu)
AU (1) AU2002337035B2 (hu)
BR (1) BR0211938A (hu)
CA (1) CA2456901C (hu)
CY (1) CY1106012T1 (hu)
DE (1) DE60216128T2 (hu)
DK (1) DK1427733T3 (hu)
ES (1) ES2275005T3 (hu)
HR (1) HRP20040202A2 (hu)
HU (1) HUP0401444A3 (hu)
IL (1) IL160084A0 (hu)
IS (1) IS2424B (hu)
MX (1) MXPA04002045A (hu)
NO (1) NO20040927L (hu)
NZ (1) NZ531340A (hu)
PE (1) PE20030439A1 (hu)
PL (1) PL368502A1 (hu)
PT (1) PT1427733E (hu)
RU (1) RU2298011C2 (hu)
TW (1) TWI228508B (hu)
WO (1) WO2003020726A1 (hu)
ZA (1) ZA200401455B (hu)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6890923B2 (en) * 2002-12-16 2005-05-10 Astrazeneca Ab Compounds
GB0315950D0 (en) * 2003-06-11 2003-08-13 Xention Discovery Ltd Compounds
GB0525164D0 (en) * 2005-12-09 2006-01-18 Xention Discovery Ltd Compounds
CN100430403C (zh) * 2006-10-13 2008-11-05 中国科学院上海有机化学研究所 3-芳基-5,6-取代噻吩并嘧啶-4-羰基-2-巯基乙腈、合成方法和用途
US20090118276A1 (en) * 2007-11-02 2009-05-07 Wyeth Thienopyrimidines, thienopyridines, and pyrrolopyrimidines as b-raf inhibitors
TWI389913B (zh) * 2008-09-08 2013-03-21 Lg Life Sciences Ltd 并合雜環化合物
CA2741030A1 (en) 2008-10-20 2010-04-29 Marvin C. Gershengorn Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
GB0905525D0 (en) 2009-03-31 2009-05-13 Univ Leiden Compounds and uses
BR112012018108A2 (pt) 2010-01-22 2015-10-20 Bayer Ip Gmbh combinações acaricidas e/ou inseticidas de ingredientes ativos
JP5965387B2 (ja) 2010-04-08 2016-08-03 アメリカ合衆国 Ｔｓｈ受容体用のインバースアゴニストおよびニュートラルアンタゴニスト
RU2619091C2 (ru) * 2015-10-13 2017-05-11 Министерство Промышленности И Торговли Рф Цилиндрический термоэмиссионный катод
WO2023239854A2 (en) * 2022-06-08 2023-12-14 Icahn School Of Medicine At Mount Sinai Method of treating obesity with a luteinizing hormone receptor agonist

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2054784T3 (es) 1987-08-08 1994-08-16 Akzo Nv Un metodo para la fabricacion de un implante.
TW564247B (en) 1999-04-08 2003-12-01 Akzo Nobel Nv Bicyclic heteraromatic compound

Also Published As

Publication number Publication date
ZA200401455B (en) 2004-11-19
ATE345345T1 (de) 2006-12-15
ES2275005T3 (es) 2007-06-01
BR0211938A (pt) 2004-09-21
PL368502A1 (en) 2005-04-04
KR20040029134A (ko) 2004-04-03
EP1427733B1 (en) 2006-11-15
HUP0401444A3 (en) 2008-05-28
AR036407A1 (es) 2004-09-08
CA2456901C (en) 2011-01-04
CY1106012T1 (el) 2011-04-06
EP1427733A1 (en) 2004-06-16
JP2005505555A (ja) 2005-02-24
HRP20040202A2 (en) 2004-08-31
IS2424B (is) 2008-10-15
US7317006B2 (en) 2008-01-08
DK1427733T3 (da) 2007-03-19
RU2298011C2 (ru) 2007-04-27
PE20030439A1 (es) 2003-05-17
AU2002337035B2 (en) 2008-04-24
CN1551884A (zh) 2004-12-01
DE60216128T2 (de) 2007-09-27
WO2003020726A1 (en) 2003-03-13
CN1246324C (zh) 2006-03-22
MXPA04002045A (es) 2004-07-08
KR100900018B1 (ko) 2009-06-01
DE60216128D1 (de) 2006-12-28
PT1427733E (pt) 2007-02-28
JP4262092B2 (ja) 2009-05-13
RU2004110042A (ru) 2005-08-20
HUP0401444A2 (hu) 2004-11-29
NO20040927L (no) 2004-03-03
US20040180873A1 (en) 2004-09-16
TWI228508B (en) 2005-03-01
NZ531340A (en) 2005-08-26
IS7130A (is) 2004-01-29
CA2456901A1 (en) 2003-03-13

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