IS7130A - Þénó[2,3-d]pýrimidín með sameinaðri LH og FSH gerandefnisvirkni - Google Patents

Þénó[2,3-d]pýrimidín með sameinaðri LH og FSH gerandefnisvirkni

Info

Publication number
IS7130A
IS7130A IS7130A IS7130A IS7130A IS 7130 A IS7130 A IS 7130A IS 7130 A IS7130 A IS 7130A IS 7130 A IS7130 A IS 7130A IS 7130 A IS7130 A IS 7130A
Authority
IS
Iceland
Prior art keywords
pyrimidine
theno
combined
agonist activity
fsh agonist
Prior art date
Application number
IS7130A
Other languages
English (en)
Other versions
IS2424B (is
Inventor
Gerard Jules Marie Hanssen Robert
Marius Timmers Cornelis
Original Assignee
Akzo Nobel N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel N.V. filed Critical Akzo Nobel N.V.
Publication of IS7130A publication Critical patent/IS7130A/is
Publication of IS2424B publication Critical patent/IS2424B/is

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/06Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/06Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A61P5/08Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH for decreasing, blocking or antagonising the activity of the anterior pituitary hormones

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IS7130A 2001-09-04 2004-01-29 Þíenó[2,3-d]pýrimidín með sameinaðri LH og FSH gerandefnisvirkni IS2424B (is)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP01203327 2001-09-04
PCT/EP2002/009647 WO2003020726A1 (en) 2001-09-04 2002-08-29 Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity

Publications (2)

Publication Number Publication Date
IS7130A true IS7130A (is) 2004-01-29
IS2424B IS2424B (is) 2008-10-15

Family

ID=8180876

Family Applications (1)

Application Number Title Priority Date Filing Date
IS7130A IS2424B (is) 2001-09-04 2004-01-29 Þíenó[2,3-d]pýrimidín með sameinaðri LH og FSH gerandefnisvirkni

Country Status (28)

Country Link
US (1) US7317006B2 (is)
EP (1) EP1427733B1 (is)
JP (1) JP4262092B2 (is)
KR (1) KR100900018B1 (is)
CN (1) CN1246324C (is)
AR (1) AR036407A1 (is)
AT (1) ATE345345T1 (is)
AU (1) AU2002337035B2 (is)
BR (1) BR0211938A (is)
CA (1) CA2456901C (is)
CY (1) CY1106012T1 (is)
DE (1) DE60216128T2 (is)
DK (1) DK1427733T3 (is)
ES (1) ES2275005T3 (is)
HR (1) HRP20040202A2 (is)
HU (1) HUP0401444A3 (is)
IL (1) IL160084A0 (is)
IS (1) IS2424B (is)
MX (1) MXPA04002045A (is)
NO (1) NO20040927L (is)
NZ (1) NZ531340A (is)
PE (1) PE20030439A1 (is)
PL (1) PL368502A1 (is)
PT (1) PT1427733E (is)
RU (1) RU2298011C2 (is)
TW (1) TWI228508B (is)
WO (1) WO2003020726A1 (is)
ZA (1) ZA200401455B (is)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6890923B2 (en) * 2002-12-16 2005-05-10 Astrazeneca Ab Compounds
GB0315950D0 (en) * 2003-06-11 2003-08-13 Xention Discovery Ltd Compounds
GB0525164D0 (en) * 2005-12-09 2006-01-18 Xention Discovery Ltd Compounds
CN100430403C (zh) * 2006-10-13 2008-11-05 中国科学院上海有机化学研究所 3-芳基-5,6-取代噻吩并嘧啶-4-羰基-2-巯基乙腈、合成方法和用途
US20090118276A1 (en) * 2007-11-02 2009-05-07 Wyeth Thienopyrimidines, thienopyridines, and pyrrolopyrimidines as b-raf inhibitors
TWI389913B (zh) * 2008-09-08 2013-03-21 Lg Life Sciences Ltd 并合雜環化合物
WO2010047674A1 (en) 2008-10-20 2010-04-29 The Government Of The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Low molecular weight thyroid stimulating hormone receptor (tshr) agonists
GB0905525D0 (en) 2009-03-31 2009-05-13 Univ Leiden Compounds and uses
PE20121693A1 (es) 2010-01-22 2012-12-01 Bayer Ip Gmbh Combinacion de espiromesifeno y abamectina como insecticidas
AU2011237421B2 (en) 2010-04-08 2016-10-13 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Inverse agonists and neutral antagonists for the TSH receptor
WO2016029375A1 (en) 2014-08-27 2016-03-03 The Procter & Gamble Company Wearable article having elastic belt
WO2016029372A1 (en) 2014-08-27 2016-03-03 The Procter & Gamble Company Wearable article having elastic belt
RU2619091C2 (ru) * 2015-10-13 2017-05-11 Министерство Промышленности И Торговли Рф Цилиндрический термоэмиссионный катод
EP3439600B1 (en) 2016-04-08 2022-06-22 The Procter & Gamble Company Wearable article having artwork
WO2023239854A2 (en) * 2022-06-08 2023-12-14 Icahn School Of Medicine At Mount Sinai Method of treating obesity with a luteinizing hormone receptor agonist

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2054784T3 (es) 1987-08-08 1994-08-16 Akzo Nv Un metodo para la fabricacion de un implante.
TW564247B (en) * 1999-04-08 2003-12-01 Akzo Nobel Nv Bicyclic heteraromatic compound

Also Published As

Publication number Publication date
IL160084A0 (en) 2004-06-20
DE60216128T2 (de) 2007-09-27
JP2005505555A (ja) 2005-02-24
NO20040927L (no) 2004-03-03
NZ531340A (en) 2005-08-26
HUP0401444A3 (en) 2008-05-28
HUP0401444A2 (hu) 2004-11-29
RU2298011C2 (ru) 2007-04-27
KR20040029134A (ko) 2004-04-03
US20040180873A1 (en) 2004-09-16
KR100900018B1 (ko) 2009-06-01
PE20030439A1 (es) 2003-05-17
ZA200401455B (en) 2004-11-19
BR0211938A (pt) 2004-09-21
CY1106012T1 (el) 2011-04-06
PL368502A1 (en) 2005-04-04
ES2275005T3 (es) 2007-06-01
AU2002337035B2 (en) 2008-04-24
RU2004110042A (ru) 2005-08-20
DE60216128D1 (de) 2006-12-28
US7317006B2 (en) 2008-01-08
HRP20040202A2 (en) 2004-08-31
CA2456901A1 (en) 2003-03-13
IS2424B (is) 2008-10-15
CN1551884A (zh) 2004-12-01
DK1427733T3 (da) 2007-03-19
EP1427733B1 (en) 2006-11-15
JP4262092B2 (ja) 2009-05-13
AR036407A1 (es) 2004-09-08
CN1246324C (zh) 2006-03-22
EP1427733A1 (en) 2004-06-16
ATE345345T1 (de) 2006-12-15
CA2456901C (en) 2011-01-04
MXPA04002045A (es) 2004-07-08
WO2003020726A1 (en) 2003-03-13
PT1427733E (pt) 2007-02-28
TWI228508B (en) 2005-03-01

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