HUP0401444A3 - Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity, use of the compounds and pharmaceutical compositions containing the same - Google Patents
Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity, use of the compounds and pharmaceutical compositions containing the sameInfo
- Publication number
- HUP0401444A3 HUP0401444A3 HU0401444A HUP0401444A HUP0401444A3 HU P0401444 A3 HUP0401444 A3 HU P0401444A3 HU 0401444 A HU0401444 A HU 0401444A HU P0401444 A HUP0401444 A HU P0401444A HU P0401444 A3 HUP0401444 A3 HU P0401444A3
- Authority
- HU
- Hungary
- Prior art keywords
- thieno
- pyrimidines
- compounds
- combined
- pharmaceutical compositions
- Prior art date
Links
- 230000001270 agonistic effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- DDWBRNXDKNIQDY-UHFFFAOYSA-N thieno[2,3-d]pyrimidine Chemical class N1=CN=C2SC=CC2=C1 DDWBRNXDKNIQDY-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
- A61P5/08—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH for decreasing, blocking or antagonising the activity of the anterior pituitary hormones
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Reproductive Health (AREA)
- Diabetes (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP01203327 | 2001-09-04 | ||
| PCT/EP2002/009647 WO2003020726A1 (en) | 2001-09-04 | 2002-08-29 | Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUP0401444A2 HUP0401444A2 (hu) | 2004-11-29 |
| HUP0401444A3 true HUP0401444A3 (en) | 2008-05-28 |
Family
ID=8180876
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0401444A HUP0401444A3 (en) | 2001-09-04 | 2002-08-29 | Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity, use of the compounds and pharmaceutical compositions containing the same |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US7317006B2 (hu) |
| EP (1) | EP1427733B1 (hu) |
| JP (1) | JP4262092B2 (hu) |
| KR (1) | KR100900018B1 (hu) |
| CN (1) | CN1246324C (hu) |
| AR (1) | AR036407A1 (hu) |
| AT (1) | ATE345345T1 (hu) |
| AU (1) | AU2002337035B2 (hu) |
| BR (1) | BR0211938A (hu) |
| CA (1) | CA2456901C (hu) |
| CY (1) | CY1106012T1 (hu) |
| DE (1) | DE60216128T2 (hu) |
| DK (1) | DK1427733T3 (hu) |
| ES (1) | ES2275005T3 (hu) |
| HR (1) | HRP20040202A2 (hu) |
| HU (1) | HUP0401444A3 (hu) |
| IL (1) | IL160084A0 (hu) |
| IS (1) | IS2424B (hu) |
| MX (1) | MXPA04002045A (hu) |
| NO (1) | NO20040927L (hu) |
| NZ (1) | NZ531340A (hu) |
| PE (1) | PE20030439A1 (hu) |
| PL (1) | PL368502A1 (hu) |
| PT (1) | PT1427733E (hu) |
| RU (1) | RU2298011C2 (hu) |
| TW (1) | TWI228508B (hu) |
| WO (1) | WO2003020726A1 (hu) |
| ZA (1) | ZA200401455B (hu) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6890923B2 (en) * | 2002-12-16 | 2005-05-10 | Astrazeneca Ab | Compounds |
| GB0315950D0 (en) * | 2003-06-11 | 2003-08-13 | Xention Discovery Ltd | Compounds |
| GB0525164D0 (en) * | 2005-12-09 | 2006-01-18 | Xention Discovery Ltd | Compounds |
| CN100430403C (zh) * | 2006-10-13 | 2008-11-05 | 中国科学院上海有机化学研究所 | 3-芳基-5,6-取代噻吩并嘧啶-4-羰基-2-巯基乙腈、合成方法和用途 |
| US20090118276A1 (en) * | 2007-11-02 | 2009-05-07 | Wyeth | Thienopyrimidines, thienopyridines, and pyrrolopyrimidines as b-raf inhibitors |
| TWI389913B (zh) * | 2008-09-08 | 2013-03-21 | Lg Life Sciences Ltd | 并合雜環化合物 |
| EP2358684B8 (en) | 2008-10-20 | 2014-10-22 | The Government of the United States of America as represented by the Secretary of the Department of Health and Human Services | Low molecular weight thyroid stimulating hormone receptor (tshr) agonists |
| GB0905525D0 (en) | 2009-03-31 | 2009-05-13 | Univ Leiden | Compounds and uses |
| RS55986B1 (sr) | 2010-01-22 | 2017-09-29 | Bayer Ip Gmbh | Akaricidne i/ili insekticidne kombinacije aktivnih supstanci |
| EP2563777A4 (en) | 2010-04-08 | 2013-09-04 | Us Health | INVERSE AGONISTS AND NEUTRAL AGONISTS FOR THE TSH RECEPTOR |
| RU2619091C2 (ru) * | 2015-10-13 | 2017-05-11 | Министерство Промышленности И Торговли Рф | Цилиндрический термоэмиссионный катод |
| WO2023239854A2 (en) * | 2022-06-08 | 2023-12-14 | Icahn School Of Medicine At Mount Sinai | Method of treating obesity with a luteinizing hormone receptor agonist |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE86484T1 (de) | 1987-08-08 | 1993-03-15 | Akzo Nv | Kontrazeptives implantat. |
| TW564247B (en) * | 1999-04-08 | 2003-12-01 | Akzo Nobel Nv | Bicyclic heteraromatic compound |
-
2002
- 2002-07-22 TW TW091116284A patent/TWI228508B/zh not_active IP Right Cessation
- 2002-08-29 IL IL16008402A patent/IL160084A0/xx not_active IP Right Cessation
- 2002-08-29 WO PCT/EP2002/009647 patent/WO2003020726A1/en active IP Right Grant
- 2002-08-29 DE DE60216128T patent/DE60216128T2/de not_active Expired - Lifetime
- 2002-08-29 NZ NZ531340A patent/NZ531340A/en unknown
- 2002-08-29 AU AU2002337035A patent/AU2002337035B2/en not_active Ceased
- 2002-08-29 DK DK02772230T patent/DK1427733T3/da active
- 2002-08-29 PT PT02772230T patent/PT1427733E/pt unknown
- 2002-08-29 BR BR0211938-2A patent/BR0211938A/pt not_active IP Right Cessation
- 2002-08-29 AT AT02772230T patent/ATE345345T1/de not_active IP Right Cessation
- 2002-08-29 RU RU2004110042/04A patent/RU2298011C2/ru not_active IP Right Cessation
- 2002-08-29 KR KR1020047003095A patent/KR100900018B1/ko not_active IP Right Cessation
- 2002-08-29 CA CA2456901A patent/CA2456901C/en not_active Expired - Fee Related
- 2002-08-29 MX MXPA04002045A patent/MXPA04002045A/es active IP Right Grant
- 2002-08-29 CN CNB028172604A patent/CN1246324C/zh not_active Expired - Fee Related
- 2002-08-29 EP EP02772230A patent/EP1427733B1/en not_active Expired - Lifetime
- 2002-08-29 JP JP2003524996A patent/JP4262092B2/ja not_active Expired - Fee Related
- 2002-08-29 ES ES02772230T patent/ES2275005T3/es not_active Expired - Lifetime
- 2002-08-29 HU HU0401444A patent/HUP0401444A3/hu unknown
- 2002-08-29 US US10/488,482 patent/US7317006B2/en not_active Expired - Lifetime
- 2002-08-29 PL PL02368502A patent/PL368502A1/xx not_active Application Discontinuation
- 2002-09-02 AR ARP020103309A patent/AR036407A1/es unknown
- 2002-09-03 PE PE2002000840A patent/PE20030439A1/es not_active Application Discontinuation
-
2004
- 2004-01-29 IS IS7130A patent/IS2424B/is unknown
- 2004-02-23 ZA ZA200401455A patent/ZA200401455B/en unknown
- 2004-03-01 HR HR20040202A patent/HRP20040202A2/hr not_active Application Discontinuation
- 2004-03-03 NO NO20040927A patent/NO20040927L/no not_active Application Discontinuation
-
2007
- 2007-02-13 CY CY20071100189T patent/CY1106012T1/el unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| GB9A | Succession in title |
Owner name: N.V. ORGANON, NL Free format text: FORMER OWNER(S): AKZO NOBEL N.V., NL |
|
| FD9A | Lapse of provisional protection due to non-payment of fees |