IL150710A0 - Use of a central cannabinoid receptor antagonist for preparing medicines designed to facilitate smoking cessation - Google Patents

Use of a central cannabinoid receptor antagonist for preparing medicines designed to facilitate smoking cessation

Info

Publication number
IL150710A0
IL150710A0 IL15071001A IL15071001A IL150710A0 IL 150710 A0 IL150710 A0 IL 150710A0 IL 15071001 A IL15071001 A IL 15071001A IL 15071001 A IL15071001 A IL 15071001A IL 150710 A0 IL150710 A0 IL 150710A0
Authority
IL
Israel
Prior art keywords
receptor antagonist
smoking cessation
cannabinoid receptor
preparing medicines
central cannabinoid
Prior art date
Application number
IL15071001A
Other languages
English (en)
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of IL150710A0 publication Critical patent/IL150710A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Addiction (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
IL15071001A 2000-02-09 2001-02-07 Use of a central cannabinoid receptor antagonist for preparing medicines designed to facilitate smoking cessation IL150710A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0001682A FR2804604B1 (fr) 2000-02-09 2000-02-09 Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles pour faciliter l'arret de la consommation de tabac
PCT/FR2001/000356 WO2001058450A2 (fr) 2000-02-09 2001-02-07 Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles pour faciliter l'arret de la consommation de tabac

Publications (1)

Publication Number Publication Date
IL150710A0 true IL150710A0 (en) 2003-02-12

Family

ID=8846875

Family Applications (1)

Application Number Title Priority Date Filing Date
IL15071001A IL150710A0 (en) 2000-02-09 2001-02-07 Use of a central cannabinoid receptor antagonist for preparing medicines designed to facilitate smoking cessation

Country Status (32)

Country Link
US (2) US6930122B2 (cg-RX-API-DMAC7.html)
EP (1) EP1257275B1 (cg-RX-API-DMAC7.html)
JP (2) JP2003522145A (cg-RX-API-DMAC7.html)
CN (1) CN1250220C (cg-RX-API-DMAC7.html)
AR (1) AR028505A1 (cg-RX-API-DMAC7.html)
AT (1) ATE292467T1 (cg-RX-API-DMAC7.html)
AU (1) AU781827B2 (cg-RX-API-DMAC7.html)
BG (2) BG110386A (cg-RX-API-DMAC7.html)
BR (1) BR0108126A (cg-RX-API-DMAC7.html)
CA (1) CA2397262C (cg-RX-API-DMAC7.html)
CZ (1) CZ296685B6 (cg-RX-API-DMAC7.html)
DE (1) DE60109903T2 (cg-RX-API-DMAC7.html)
DK (1) DK1257275T3 (cg-RX-API-DMAC7.html)
EE (1) EE04836B1 (cg-RX-API-DMAC7.html)
ES (1) ES2240416T3 (cg-RX-API-DMAC7.html)
FR (1) FR2804604B1 (cg-RX-API-DMAC7.html)
HU (1) HU225328B1 (cg-RX-API-DMAC7.html)
IL (1) IL150710A0 (cg-RX-API-DMAC7.html)
IS (1) IS6450A (cg-RX-API-DMAC7.html)
MX (1) MXPA02007766A (cg-RX-API-DMAC7.html)
NO (1) NO324521B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ519924A (cg-RX-API-DMAC7.html)
PL (1) PL201685B1 (cg-RX-API-DMAC7.html)
PT (1) PT1257275E (cg-RX-API-DMAC7.html)
RS (1) RS50404B (cg-RX-API-DMAC7.html)
RU (1) RU2257207C2 (cg-RX-API-DMAC7.html)
SI (1) SI1257275T1 (cg-RX-API-DMAC7.html)
SK (1) SK284952B6 (cg-RX-API-DMAC7.html)
TW (1) TWI243677B (cg-RX-API-DMAC7.html)
UA (1) UA72783C2 (cg-RX-API-DMAC7.html)
WO (1) WO2001058450A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA200205317B (cg-RX-API-DMAC7.html)

Families Citing this family (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2804604B1 (fr) * 2000-02-09 2005-05-27 Sanofi Synthelabo Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles pour faciliter l'arret de la consommation de tabac
US6462237B1 (en) * 2001-06-14 2002-10-08 Usv Limited Cyclodextrin stabilized pharmaceutical compositions of bupropion hydrochloride
AU2002356039A1 (en) 2001-08-13 2003-03-03 Honeywell International Inc. Methods of conducting wafer level burn-in of electronic devices
JP2005533748A (ja) 2002-03-08 2005-11-10 シグナル ファーマシューティカルズ，インコーポレイテッド 増殖性障害および癌を治療、予防、または管理するための併用療法
WO2003077847A2 (en) 2002-03-12 2003-09-25 Merck & Co., Inc. Substituted amides
JP2005528366A (ja) 2002-03-26 2005-09-22 メルク　エンド　カムパニー　インコーポレーテッド カンナビノイド受容体モジュレータとしてのスピロ環式アミド
JP2005531520A (ja) 2002-03-28 2005-10-20 メルク　エンド　カムパニー　インコーポレーテッド 置換２，３−ジフェニルピリジン類
WO2003086288A2 (en) 2002-04-12 2003-10-23 Merck & Co., Inc. Bicyclic amides
US6825209B2 (en) 2002-04-15 2004-11-30 Research Triangle Institute Compounds having unique CB1 receptor binding selectivity and methods for their production and use
ATE375349T1 (de) 2002-08-02 2007-10-15 Merck & Co Inc Substituierte furo(2,3-b)pyridin derivate
CA2499497A1 (en) 2002-09-27 2004-04-08 Merck & Co., Inc. Substituted pyrimidines
US7129239B2 (en) 2002-10-28 2006-10-31 Pfizer Inc. Purine compounds and uses thereof
US7247628B2 (en) 2002-12-12 2007-07-24 Pfizer, Inc. Cannabinoid receptor ligands and uses thereof
WO2004058145A2 (en) 2002-12-19 2004-07-15 Merck & Co., Inc. Substituted amides
US7329658B2 (en) 2003-02-06 2008-02-12 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US7176210B2 (en) 2003-02-10 2007-02-13 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
US7145012B2 (en) 2003-04-23 2006-12-05 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
US7268133B2 (en) 2003-04-23 2007-09-11 Pfizer, Inc. Patent Department Cannabinoid receptor ligands and uses thereof
US20040224962A1 (en) * 2003-05-09 2004-11-11 Pfizer Inc Pharmaceutical composition for the treatment of obesity or to facilitate or promote weight loss
US20040224963A1 (en) * 2003-05-09 2004-11-11 Pfizer Inc Pharmaceutical composition for the prevention and treatment of nicotine addiction in a mammal
CA2526103A1 (en) * 2003-05-20 2004-12-29 Bob M. Ii Moore Cannabinoid derivatives, methods of making, and use thereof
US7232823B2 (en) 2003-06-09 2007-06-19 Pfizer, Inc. Cannabinoid receptor ligands and uses thereof
CA2543882A1 (en) * 2003-10-30 2005-05-19 Merck & Co., Inc. Aralkyl amines as cannabinoid receptor modulators
MX2007000491A (es) 2004-07-12 2007-03-28 Cadila Healthcare Ltd Nuevos compuestos heterociclicos.
US20060025448A1 (en) 2004-07-22 2006-02-02 Cadila Healthcare Limited Hair growth stimulators
ES2435790T3 (es) 2004-12-03 2013-12-23 Intervet International B.V. Piperazinas sustituidas como antagonistas de CB1
NZ569814A (en) * 2006-01-18 2011-10-28 Schering Corp Cannibinoid receptor modulators
WO2007121687A1 (en) * 2006-04-26 2007-11-01 Institute Of Pharmacology And Toxicology Academy Of Military Medical Sciences P.L.A. China 4-methyl-1h-diaryl pyrazole derivatives and their uses as medicament
CN101062919B (zh) * 2006-04-26 2012-08-15 中国人民解放军军事医学科学院毒物药物研究所 4-甲基-1h-二芳基吡唑衍生物及其作为药物的用途
US20070287734A1 (en) * 2006-06-09 2007-12-13 Auspex Pharmaceuticals, Inc. Preparation and utility of substituted pyrazole compounds with cannabinoid receptor activity
RU2477634C2 (ru) * 2006-06-16 2013-03-20 Теракос, Инк. Лечение психологических состояний с применением антагонистов m1-мускариновых рецепторов
WO2008046905A1 (en) * 2006-10-20 2008-04-24 Solvay Pharmaceuticals B.V. Micellar nanoparticles of chemical substances
WO2008130616A2 (en) * 2007-04-19 2008-10-30 Schering Corporation Diaryl morpholines as cb1 modulators
WO2009005671A2 (en) * 2007-06-28 2009-01-08 Schering Corporation Substituted piperazines as cb1 antagonists
EP2170846A2 (en) * 2007-06-28 2010-04-07 Intervet International BV Substituted piperazines as cb1 antagonists
EP2095814A1 (de) * 2008-02-26 2009-09-02 Wolfgang J. Kox Medikamentengestützter Nikotinentzug
WO2010018856A1 (ja) * 2008-08-13 2010-02-18 持田製薬株式会社 カンナビノイド受容体関連疾患の予防／改善または治療剤
RU2533224C2 (ru) * 2010-07-21 2014-11-20 Мапикс Эс.Эй.Ар.Эл. Способ лечения зависимости от психоактивных веществ, алкоголизма и табакокурения и лекарственное средство для лечения зависимости от психоактивных веществ, алкоголизма и табакокурения
WO2013068371A1 (en) 2011-11-08 2013-05-16 Intervet International B.V. Soft chewable dosage form compositions of cannabinoid receptor type 1 (cb-1) antagonists
WO2014181357A1 (en) * 2013-05-09 2014-11-13 Council Of Scientific & Industrial Research Novel pyrazole derivatives with silicon incorporation
US20200035118A1 (en) 2018-07-27 2020-01-30 Joseph Pandolfino Methods and products to facilitate smokers switching to a tobacco heating product or e-cigarettes
US10897925B2 (en) 2018-07-27 2021-01-26 Joseph Pandolfino Articles and formulations for smoking products and vaporizers

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5780051A (en) * 1992-04-02 1998-07-14 Dynagen, Inc. Methods and articles of manufacture for nicotine cessation and monitoring nicotine use
FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
US5596106A (en) * 1994-07-15 1997-01-21 Eli Lilly And Company Cannabinoid receptor antagonists
FR2758723B1 (fr) * 1997-01-28 1999-04-23 Sanofi Sa Utilisation des antagonistes des recepteurs aux cannabinoides centraux pour la preparation de medicaments
FR2765107B1 (fr) * 1997-06-26 2000-03-24 Sanofi Sa Utilisation d'un antagoniste specifique des recepteurs 5ht2 pour la preparation de medicaments utiles dans le traitement du syndrome d'apnee du sommeil
FR2789079B3 (fr) 1999-02-01 2001-03-02 Sanofi Synthelabo Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
FR2804604B1 (fr) * 2000-02-09 2005-05-27 Sanofi Synthelabo Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles pour faciliter l'arret de la consommation de tabac

Also Published As

Publication number Publication date
CA2397262A1 (en) 2001-08-16
CA2397262C (en) 2007-09-11
US20030087933A1 (en) 2003-05-08
YU59002A (sh) 2005-07-19
US20050187253A1 (en) 2005-08-25
PL358221A1 (en) 2004-08-09
IS6450A (is) 2002-06-28
BG106946A (bg) 2003-05-30
PT1257275E (pt) 2005-07-29
EP1257275B1 (fr) 2005-04-06
HUP0300237A2 (hu) 2003-07-28
NZ519924A (en) 2005-01-28
HK1051140A1 (en) 2003-07-25
AU3562001A (en) 2001-08-20
RU2002118309A (ru) 2004-02-20
CN1250220C (zh) 2006-04-12
AU781827B2 (en) 2005-06-16
NO20023765D0 (no) 2002-08-08
MXPA02007766A (es) 2002-10-11
EE04836B1 (et) 2007-06-15
BR0108126A (pt) 2003-01-28
ATE292467T1 (de) 2005-04-15
DE60109903D1 (de) 2005-05-12
JP2010018622A (ja) 2010-01-28
FR2804604B1 (fr) 2005-05-27
WO2001058450A3 (fr) 2002-04-25
SK284952B6 (sk) 2006-03-02
US6930122B2 (en) 2005-08-16
CZ296685B6 (cs) 2006-05-17
NO20023765L (no) 2002-10-09
DE60109903T2 (de) 2006-02-09
TWI243677B (en) 2005-11-21
JP2003522145A (ja) 2003-07-22
BG110386A (en) 2009-09-30
SI1257275T1 (en) 2005-10-31
NO324521B1 (no) 2007-11-12
ZA200205317B (en) 2003-09-04
EE200200439A (et) 2003-12-15
RS50404B (sr) 2009-12-31
DK1257275T3 (da) 2005-08-08
HUP0300237A3 (en) 2003-09-29
AR028505A1 (es) 2003-05-14
FR2804604A1 (fr) 2001-08-10
PL201685B1 (pl) 2009-04-30
HU225328B1 (en) 2006-09-28
SK11292002A3 (sk) 2003-02-04
WO2001058450A2 (fr) 2001-08-16
RU2257207C2 (ru) 2005-07-27
BG65856B1 (bg) 2010-03-31
UA72783C2 (en) 2005-04-15
CN1406128A (zh) 2003-03-26
EP1257275A2 (fr) 2002-11-20
ES2240416T3 (es) 2005-10-16
CZ20022698A3 (cs) 2002-11-13

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Legal Events

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