BG110386A - USE OF ANTAGONISTS OF CENTRAL RECEPTORS OF CANNABINOIDS FOR THE RECEIPT OF MEDICINAL PRODUCTS TO FACILITATE THE STOPPING OF TOBACCO CONSUMPTION - Google Patents

USE OF ANTAGONISTS OF CENTRAL RECEPTORS OF CANNABINOIDS FOR THE RECEIPT OF MEDICINAL PRODUCTS TO FACILITATE THE STOPPING OF TOBACCO CONSUMPTION

Info

Publication number
BG110386A
BG110386A BG110386A BG11038601A BG110386A BG 110386 A BG110386 A BG 110386A BG 110386 A BG110386 A BG 110386A BG 11038601 A BG11038601 A BG 11038601A BG 110386 A BG110386 A BG 110386A
Authority
BG
Bulgaria
Prior art keywords
antagonist
central
medicines used
tobacco consumption
facilitate stopping
Prior art date
Application number
BG110386A
Other languages
Bulgarian (bg)
English (en)
Inventor
Jean BLANCHARD
Francois Menard
Original Assignee
Sanofi-Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Aventis filed Critical Sanofi-Aventis
Publication of BG110386A publication Critical patent/BG110386A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Addiction (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
BG110386A 2000-02-09 2001-02-07 USE OF ANTAGONISTS OF CENTRAL RECEPTORS OF CANNABINOIDS FOR THE RECEIPT OF MEDICINAL PRODUCTS TO FACILITATE THE STOPPING OF TOBACCO CONSUMPTION BG110386A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0001682A FR2804604B1 (fr) 2000-02-09 2000-02-09 Utilisation d'un antagoniste des recepteurs aux cannabinoides centraux pour la preparation de medicaments utiles pour faciliter l'arret de la consommation de tabac

Publications (1)

Publication Number Publication Date
BG110386A true BG110386A (en) 2009-09-30

Family

ID=8846875

Family Applications (2)

Application Number Title Priority Date Filing Date
BG110386A BG110386A (en) 2000-02-09 2001-02-07 USE OF ANTAGONISTS OF CENTRAL RECEPTORS OF CANNABINOIDS FOR THE RECEIPT OF MEDICINAL PRODUCTS TO FACILITATE THE STOPPING OF TOBACCO CONSUMPTION
BG106946A BG65856B1 (bg) 2000-02-09 2002-07-23 Използване на антагонисти на централни канабиноидни рецептори за получаване на лекарствени средства за улесняване спирането на консумацията на тютюн

Family Applications After (1)

Application Number Title Priority Date Filing Date
BG106946A BG65856B1 (bg) 2000-02-09 2002-07-23 Използване на антагонисти на централни канабиноидни рецептори за получаване на лекарствени средства за улесняване спирането на консумацията на тютюн

Country Status (32)

Country Link
US (2) US6930122B2 (cg-RX-API-DMAC7.html)
EP (1) EP1257275B1 (cg-RX-API-DMAC7.html)
JP (2) JP2003522145A (cg-RX-API-DMAC7.html)
CN (1) CN1250220C (cg-RX-API-DMAC7.html)
AR (1) AR028505A1 (cg-RX-API-DMAC7.html)
AT (1) ATE292467T1 (cg-RX-API-DMAC7.html)
AU (1) AU781827B2 (cg-RX-API-DMAC7.html)
BG (2) BG110386A (cg-RX-API-DMAC7.html)
BR (1) BR0108126A (cg-RX-API-DMAC7.html)
CA (1) CA2397262C (cg-RX-API-DMAC7.html)
CZ (1) CZ296685B6 (cg-RX-API-DMAC7.html)
DE (1) DE60109903T2 (cg-RX-API-DMAC7.html)
DK (1) DK1257275T3 (cg-RX-API-DMAC7.html)
EE (1) EE04836B1 (cg-RX-API-DMAC7.html)
ES (1) ES2240416T3 (cg-RX-API-DMAC7.html)
FR (1) FR2804604B1 (cg-RX-API-DMAC7.html)
HU (1) HU225328B1 (cg-RX-API-DMAC7.html)
IL (1) IL150710A0 (cg-RX-API-DMAC7.html)
IS (1) IS6450A (cg-RX-API-DMAC7.html)
MX (1) MXPA02007766A (cg-RX-API-DMAC7.html)
NO (1) NO324521B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ519924A (cg-RX-API-DMAC7.html)
PL (1) PL201685B1 (cg-RX-API-DMAC7.html)
PT (1) PT1257275E (cg-RX-API-DMAC7.html)
RS (1) RS50404B (cg-RX-API-DMAC7.html)
RU (1) RU2257207C2 (cg-RX-API-DMAC7.html)
SI (1) SI1257275T1 (cg-RX-API-DMAC7.html)
SK (1) SK284952B6 (cg-RX-API-DMAC7.html)
TW (1) TWI243677B (cg-RX-API-DMAC7.html)
UA (1) UA72783C2 (cg-RX-API-DMAC7.html)
WO (1) WO2001058450A2 (cg-RX-API-DMAC7.html)
ZA (1) ZA200205317B (cg-RX-API-DMAC7.html)

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JP2005528366A (ja) 2002-03-26 2005-09-22 メルク　エンド　カムパニー　インコーポレーテッド カンナビノイド受容体モジュレータとしてのスピロ環式アミド
JP2005531520A (ja) 2002-03-28 2005-10-20 メルク　エンド　カムパニー　インコーポレーテッド 置換２，３−ジフェニルピリジン類
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WO2004058145A2 (en) 2002-12-19 2004-07-15 Merck & Co., Inc. Substituted amides
US7329658B2 (en) 2003-02-06 2008-02-12 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US7176210B2 (en) 2003-02-10 2007-02-13 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
US7145012B2 (en) 2003-04-23 2006-12-05 Pfizer Inc. Cannabinoid receptor ligands and uses thereof
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US20040224962A1 (en) * 2003-05-09 2004-11-11 Pfizer Inc Pharmaceutical composition for the treatment of obesity or to facilitate or promote weight loss
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CA2526103A1 (en) * 2003-05-20 2004-12-29 Bob M. Ii Moore Cannabinoid derivatives, methods of making, and use thereof
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US20060025448A1 (en) 2004-07-22 2006-02-02 Cadila Healthcare Limited Hair growth stimulators
ES2435790T3 (es) 2004-12-03 2013-12-23 Intervet International B.V. Piperazinas sustituidas como antagonistas de CB1
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WO2007121687A1 (en) * 2006-04-26 2007-11-01 Institute Of Pharmacology And Toxicology Academy Of Military Medical Sciences P.L.A. China 4-methyl-1h-diaryl pyrazole derivatives and their uses as medicament
CN101062919B (zh) * 2006-04-26 2012-08-15 中国人民解放军军事医学科学院毒物药物研究所 4-甲基-1h-二芳基吡唑衍生物及其作为药物的用途
US20070287734A1 (en) * 2006-06-09 2007-12-13 Auspex Pharmaceuticals, Inc. Preparation and utility of substituted pyrazole compounds with cannabinoid receptor activity
RU2477634C2 (ru) * 2006-06-16 2013-03-20 Теракос, Инк. Лечение психологических состояний с применением антагонистов m1-мускариновых рецепторов
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RU2533224C2 (ru) * 2010-07-21 2014-11-20 Мапикс Эс.Эй.Ар.Эл. Способ лечения зависимости от психоактивных веществ, алкоголизма и табакокурения и лекарственное средство для лечения зависимости от психоактивных веществ, алкоголизма и табакокурения
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FR2713225B1 (fr) * 1993-12-02 1996-03-01 Sanofi Sa N-pipéridino-3-pyrazolecarboxamide substitué.
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Also Published As

Publication number Publication date
CA2397262A1 (en) 2001-08-16
CA2397262C (en) 2007-09-11
US20030087933A1 (en) 2003-05-08
YU59002A (sh) 2005-07-19
US20050187253A1 (en) 2005-08-25
PL358221A1 (en) 2004-08-09
IS6450A (is) 2002-06-28
BG106946A (bg) 2003-05-30
PT1257275E (pt) 2005-07-29
EP1257275B1 (fr) 2005-04-06
HUP0300237A2 (hu) 2003-07-28
NZ519924A (en) 2005-01-28
HK1051140A1 (en) 2003-07-25
AU3562001A (en) 2001-08-20
RU2002118309A (ru) 2004-02-20
CN1250220C (zh) 2006-04-12
AU781827B2 (en) 2005-06-16
NO20023765D0 (no) 2002-08-08
MXPA02007766A (es) 2002-10-11
EE04836B1 (et) 2007-06-15
BR0108126A (pt) 2003-01-28
ATE292467T1 (de) 2005-04-15
DE60109903D1 (de) 2005-05-12
JP2010018622A (ja) 2010-01-28
FR2804604B1 (fr) 2005-05-27
IL150710A0 (en) 2003-02-12
WO2001058450A3 (fr) 2002-04-25
SK284952B6 (sk) 2006-03-02
US6930122B2 (en) 2005-08-16
CZ296685B6 (cs) 2006-05-17
NO20023765L (no) 2002-10-09
DE60109903T2 (de) 2006-02-09
TWI243677B (en) 2005-11-21
JP2003522145A (ja) 2003-07-22
SI1257275T1 (en) 2005-10-31
NO324521B1 (no) 2007-11-12
ZA200205317B (en) 2003-09-04
EE200200439A (et) 2003-12-15
RS50404B (sr) 2009-12-31
DK1257275T3 (da) 2005-08-08
HUP0300237A3 (en) 2003-09-29
AR028505A1 (es) 2003-05-14
FR2804604A1 (fr) 2001-08-10
PL201685B1 (pl) 2009-04-30
HU225328B1 (en) 2006-09-28
SK11292002A3 (sk) 2003-02-04
WO2001058450A2 (fr) 2001-08-16
RU2257207C2 (ru) 2005-07-27
BG65856B1 (bg) 2010-03-31
UA72783C2 (en) 2005-04-15
CN1406128A (zh) 2003-03-26
EP1257275A2 (fr) 2002-11-20
ES2240416T3 (es) 2005-10-16
CZ20022698A3 (cs) 2002-11-13

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