IL146731A0 - Factor viia inhibitors - Google Patents

Factor viia inhibitors

Info

Publication number
IL146731A0
IL146731A0 IL14673100A IL14673100A IL146731A0 IL 146731 A0 IL146731 A0 IL 146731A0 IL 14673100 A IL14673100 A IL 14673100A IL 14673100 A IL14673100 A IL 14673100A IL 146731 A0 IL146731 A0 IL 146731A0
Authority
IL
Israel
Prior art keywords
factor viia
viia inhibitors
inhibitors
factor
viia
Prior art date
Application number
IL14673100A
Other languages
English (en)
Original Assignee
Aventis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh
Publication of IL146731A0 publication Critical patent/IL146731A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06086Dipeptides with the first amino acid being basic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pyridine Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
IL14673100A 1999-06-08 2000-05-27 Factor viia inhibitors IL146731A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99111109A EP1059302A1 (en) 1999-06-08 1999-06-08 Factor VIIa inhibitors
PCT/EP2000/004846 WO2000075172A2 (en) 1999-06-08 2000-05-27 FACTOR VIIa INHIBITORS

Publications (1)

Publication Number Publication Date
IL146731A0 true IL146731A0 (en) 2002-07-25

Family

ID=8238315

Family Applications (2)

Application Number Title Priority Date Filing Date
IL14673100A IL146731A0 (en) 1999-06-08 2000-05-27 Factor viia inhibitors
IL146731A IL146731A (en) 1999-06-08 2001-11-25 Factor VIIa inhibitors

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL146731A IL146731A (en) 1999-06-08 2001-11-25 Factor VIIa inhibitors

Country Status (32)

Country Link
US (1) US6500803B1 (cs)
EP (2) EP1059302A1 (cs)
JP (1) JP4546683B2 (cs)
KR (1) KR100979069B1 (cs)
CN (1) CN1359390B (cs)
AR (1) AR024292A1 (cs)
AT (1) ATE246707T1 (cs)
AU (1) AU774037B2 (cs)
BR (1) BR0011461A (cs)
CA (1) CA2376064C (cs)
CZ (1) CZ300365B6 (cs)
DE (1) DE60004363T2 (cs)
DK (1) DK1189929T3 (cs)
EE (1) EE04855B1 (cs)
ES (1) ES2202137T3 (cs)
HK (1) HK1047289B (cs)
HR (1) HRP20010912B1 (cs)
HU (1) HUP0201451A3 (cs)
IL (2) IL146731A0 (cs)
ME (1) MEP57708A (cs)
MX (1) MXPA01012568A (cs)
NO (1) NO328249B1 (cs)
NZ (1) NZ515966A (cs)
PL (1) PL202879B1 (cs)
PT (1) PT1189929E (cs)
RS (1) RS50415B (cs)
RU (1) RU2248359C2 (cs)
SI (1) SI1189929T1 (cs)
SK (1) SK286902B6 (cs)
TR (1) TR200103550T2 (cs)
WO (1) WO2000075172A2 (cs)
ZA (1) ZA200110053B (cs)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1059302A1 (en) * 1999-06-08 2000-12-13 Aventis Pharma Deutschland GmbH Factor VIIa inhibitors
DE10005631A1 (de) * 2000-02-09 2001-08-23 Max Planck Gesellschaft Arginin-Mimetika als Faktor X¶a¶-Inhibitoren
GB0014134D0 (en) * 2000-06-10 2000-08-02 Astrazeneca Ab Combination therapy
EP1364960A4 (en) * 2001-02-02 2005-05-18 Chugai Pharmaceutical Co Ltd PEPTIDE DERIVATIVES
GB0127615D0 (en) * 2001-07-09 2002-01-09 Aventis Pharm Prod Inc Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
JP5043429B2 (ja) * 2003-08-18 2012-10-10 ハー・ルンドベック・アクチエゼルスカベット トランス−4−((1r,3s)−6−クロロ−3−フェニルインダン−1−イル)−1,2,2−トリメチルピペラジンのコハク酸塩およびマロン酸塩、および薬剤としての使用方法
TWI453198B (zh) 2005-02-16 2014-09-21 Lundbeck & Co As H 製造反式-1-((1r,3s)-6-氯基-3-苯基茚滿-1-基) -3 , 3 -二甲基六氫吡與其鹽類之方法及製造4-((1r , 3s)-6 -氯基-3-苯基茚滿-1-基 )-1,2,2-三甲基六氫吡與其鹽類之方法
TWI376373B (en) 2005-02-16 2012-11-11 Lundbeck & Co As H Crystalline base of a pharmaceutical compound
ES2337831T3 (es) * 2005-06-24 2010-04-29 Bristol-Myers Squibb Company Derivados de fenilglicinamida y piridilclicinamida utiles como agentes anticoagulantes.
WO2007131996A1 (en) * 2006-05-12 2007-11-22 Genmedica Therapeutics Sl Meta-xylylenediamine vanadate salts
US11021514B2 (en) 2016-06-01 2021-06-01 Athira Pharma, Inc. Compounds
DK3993876T3 (en) 2019-07-01 2024-12-02 Tonix Pharma Ltd Anti-cd154 antibodies and uses thereof
EP4274587A1 (en) 2021-01-06 2023-11-15 Tonix Pharma Limited Methods of inducing immune tolerance with modified anti-cd154 antibodies

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5023236A (en) * 1988-04-07 1991-06-11 Corvas, Inc. Factor VII/VIIA active site inhibitors
US5506134A (en) 1990-10-22 1996-04-09 Corvas International, Inc. Hypridoma and monoclonal antibody which inhibits blood coagulation tissue factor/factor VIIa complex
US5788965A (en) 1991-02-28 1998-08-04 Novo Nordisk A/S Modified factor VII
US5833982A (en) 1991-02-28 1998-11-10 Zymogenetics, Inc. Modified factor VII
DE4115468A1 (de) * 1991-05-11 1992-11-12 Behringwerke Ag Amidinophenylalaninderivate, verfahren zu deren herstellung, deren verwendung und diese enthaltende mittel als antikoagulantien
SE9301916D0 (sv) * 1993-06-03 1993-06-03 Ab Astra New peptides derivatives
SI9520044B (sl) * 1994-04-26 2004-08-31 Aventis Pharmaceuticals Inc. Inhibitorji Xa faktorja
PT892780E (pt) * 1996-02-22 2003-02-28 Bristol Myers Squibb Pharma Co Analogos de m-amidino fenilo como inibidores do factor xa
AR013084A1 (es) * 1997-06-19 2000-12-13 Astrazeneca Ab Derivados de amidino utiles como inhibidores de la trombina, composicion farmaceutica, utilizacion de dichos compuestos para la preparacion demedicamentos y proceso para la preparacion de los compuestos mencionados
EP0987274A1 (en) * 1998-09-15 2000-03-22 Hoechst Marion Roussel Deutschland GmbH Factor VIIa Inhibitors
EP1059302A1 (en) * 1999-06-08 2000-12-13 Aventis Pharma Deutschland GmbH Factor VIIa inhibitors

Also Published As

Publication number Publication date
HK1047289A1 (zh) 2003-02-14
ATE246707T1 (de) 2003-08-15
HUP0201451A3 (en) 2003-08-28
WO2000075172A2 (en) 2000-12-14
DK1189929T3 (da) 2003-11-24
HRP20010912A2 (en) 2003-04-30
YU86101A (sh) 2004-07-15
EE200100662A (et) 2003-04-15
KR20020020728A (ko) 2002-03-15
WO2000075172A3 (en) 2001-05-31
NZ515966A (en) 2003-09-26
HRP20010912B1 (en) 2010-10-31
PL352200A1 (en) 2003-08-11
AU5397600A (en) 2000-12-28
TR200103550T2 (tr) 2002-05-21
HK1047289B (zh) 2010-10-22
DE60004363D1 (de) 2003-09-11
BR0011461A (pt) 2002-03-19
EE04855B1 (et) 2007-06-15
CA2376064A1 (en) 2000-12-14
EP1189929A2 (en) 2002-03-27
CZ300365B6 (cs) 2009-04-29
SK286902B6 (sk) 2009-07-06
JP2003502294A (ja) 2003-01-21
CN1359390A (zh) 2002-07-17
AU774037B2 (en) 2004-06-17
AR024292A1 (es) 2002-09-25
US6500803B1 (en) 2002-12-31
ES2202137T3 (es) 2004-04-01
SK17592001A3 (sk) 2002-05-09
NO20016005D0 (no) 2001-12-07
CA2376064C (en) 2011-04-26
PT1189929E (pt) 2003-12-31
CZ20014357A3 (cs) 2002-03-13
DE60004363T2 (de) 2004-06-24
PL202879B1 (pl) 2009-07-31
NO20016005L (no) 2002-02-06
SI1189929T1 (en) 2004-02-29
JP4546683B2 (ja) 2010-09-15
EP1059302A1 (en) 2000-12-13
RU2248359C2 (ru) 2005-03-20
ZA200110053B (en) 2002-07-03
EP1189929B1 (en) 2003-08-06
MEP57708A (en) 2011-05-10
MXPA01012568A (es) 2002-04-10
KR100979069B1 (ko) 2010-08-31
HUP0201451A2 (en) 2002-08-28
RS50415B (sr) 2009-12-31
CN1359390B (zh) 2010-05-26
NO328249B1 (no) 2010-01-18
IL146731A (en) 2007-07-24

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