IL130293A0 - Preparation of thiazoles - Google Patents
Preparation of thiazolesInfo
- Publication number
- IL130293A0 IL130293A0 IL13029397A IL13029397A IL130293A0 IL 130293 A0 IL130293 A0 IL 130293A0 IL 13029397 A IL13029397 A IL 13029397A IL 13029397 A IL13029397 A IL 13029397A IL 130293 A0 IL130293 A0 IL 130293A0
- Authority
- IL
- Israel
- Prior art keywords
- alkyl
- halogen
- formula
- phenyl
- compound
- Prior art date
Links
- 150000003557 thiazoles Chemical class 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 7
- 150000001875 compounds Chemical class 0.000 abstract 3
- 125000001997 phenyl group Chemical class [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 3
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000001797 benzyl group Chemical class [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
- 229910052799 carbon Inorganic materials 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical group [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- AFVFQIVMOAPDHO-UHFFFAOYSA-M Methanesulfonate Chemical group CS([O-])(=O)=O AFVFQIVMOAPDHO-UHFFFAOYSA-M 0.000 abstract 1
- 125000000304 alkynyl group Chemical group 0.000 abstract 1
- -1 benzothilzolyl Chemical class 0.000 abstract 1
- 125000000113 cyclohexyl group Chemical class [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 125000004076 pyridyl group Chemical class 0.000 abstract 1
- 125000000714 pyrimidinyl group Chemical class 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 125000000335 thiazolyl group Chemical class 0.000 abstract 1
- JOXIMZWYDAKGHI-UHFFFAOYSA-N toluene-4-sulfonic acid Chemical compound CC1=CC=C(S(O)(=O)=O)C=C1 JOXIMZWYDAKGHI-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/16—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/36—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/70—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/70—Sulfur atoms
- C07D277/74—Sulfur atoms substituted by carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH312596 | 1996-12-19 | ||
| PCT/EP1997/007088 WO1998027075A1 (en) | 1996-12-19 | 1997-12-17 | Preparation of thiazoles |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL130293A0 true IL130293A0 (en) | 2000-06-01 |
Family
ID=4249152
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL13029397A IL130293A0 (en) | 1996-12-19 | 1997-12-17 | Preparation of thiazoles |
Country Status (11)
| Country | Link |
|---|---|
| US (5) | US6548676B1 (de) |
| EP (3) | EP1577307A3 (de) |
| JP (1) | JP4354533B2 (de) |
| KR (1) | KR100521067B1 (de) |
| AT (2) | ATE307807T1 (de) |
| AU (1) | AU6205698A (de) |
| DE (2) | DE69714076T2 (de) |
| DK (2) | DK0946532T3 (de) |
| ES (2) | ES2181059T3 (de) |
| IL (1) | IL130293A0 (de) |
| WO (1) | WO1998027075A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI359810B (en) * | 2004-11-04 | 2012-03-11 | Mitsubishi Tanabe Pharma Corp | Carboxylic acid derivative containing thiazole rin |
| WO2016057931A1 (en) | 2014-10-10 | 2016-04-14 | The Research Foundation For The State University Of New York | Trifluoromethoxylation of arenes via intramolecular trifluoromethoxy group migration |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US546167A (en) * | 1895-09-10 | Mills | ||
| EP0192060B1 (de) | 1985-02-04 | 1991-09-18 | Nihon Bayer Agrochem K.K. | Heterocyclische Verbindungen |
| US5180833A (en) * | 1990-03-16 | 1993-01-19 | Takeda Chemical Industries, Ltd. | Process for the preparation of chlorothiazole derivatives |
| AU640239B2 (en) | 1990-06-18 | 1993-08-19 | Mitsubishi Chemical Corporation | Pyrazolecarboxamide, insecticidal and miticidal composition, and fungicidal composition for use in agriculture and horticulture |
| ZA9610046B (en) * | 1995-12-01 | 1997-07-10 | Ciba Geigy | Process for preparing 2-chlorothiazole compounds |
-
1997
- 1997-12-17 ES ES97954817T patent/ES2181059T3/es not_active Expired - Lifetime
- 1997-12-17 DK DK97954817T patent/DK0946532T3/da active
- 1997-12-17 JP JP52732398A patent/JP4354533B2/ja not_active Expired - Fee Related
- 1997-12-17 ES ES01129478T patent/ES2246985T3/es not_active Expired - Lifetime
- 1997-12-17 DE DE69714076T patent/DE69714076T2/de not_active Expired - Lifetime
- 1997-12-17 IL IL13029397A patent/IL130293A0/xx not_active IP Right Cessation
- 1997-12-17 DK DK01129478T patent/DK1201662T3/da active
- 1997-12-17 EP EP05013434A patent/EP1577307A3/de not_active Withdrawn
- 1997-12-17 EP EP97954817A patent/EP0946532B1/de not_active Expired - Lifetime
- 1997-12-17 US US09/331,433 patent/US6548676B1/en not_active Expired - Fee Related
- 1997-12-17 AT AT01129478T patent/ATE307807T1/de active
- 1997-12-17 AT AT97954817T patent/ATE220670T1/de active
- 1997-12-17 WO PCT/EP1997/007088 patent/WO1998027075A1/en not_active Ceased
- 1997-12-17 KR KR10-1999-7005612A patent/KR100521067B1/ko not_active Expired - Fee Related
- 1997-12-17 EP EP01129478A patent/EP1201662B1/de not_active Expired - Lifetime
- 1997-12-17 DE DE69734479T patent/DE69734479T2/de not_active Expired - Lifetime
- 1997-12-17 AU AU62056/98A patent/AU6205698A/en not_active Abandoned
-
2003
- 2003-03-27 US US10/400,826 patent/US7161011B2/en not_active Expired - Fee Related
-
2006
- 2006-10-24 US US11/552,255 patent/US7323564B2/en not_active Expired - Fee Related
-
2007
- 2007-11-30 US US11/947,891 patent/US7538229B2/en not_active Expired - Fee Related
-
2009
- 2009-04-16 US US12/424,594 patent/US7795442B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US7538229B2 (en) | 2009-05-26 |
| DK1201662T3 (da) | 2006-02-13 |
| EP0946532A1 (de) | 1999-10-06 |
| EP1577307A2 (de) | 2005-09-21 |
| ATE307807T1 (de) | 2005-11-15 |
| US7323564B2 (en) | 2008-01-29 |
| DE69714076T2 (de) | 2003-03-06 |
| US20070055063A1 (en) | 2007-03-08 |
| WO1998027075A1 (en) | 1998-06-25 |
| KR20000069614A (ko) | 2000-11-25 |
| DE69734479D1 (de) | 2005-12-01 |
| EP1201662B1 (de) | 2005-10-26 |
| ES2181059T3 (es) | 2003-02-16 |
| US20030216579A1 (en) | 2003-11-20 |
| US20090198054A1 (en) | 2009-08-06 |
| ES2246985T3 (es) | 2006-03-01 |
| KR100521067B1 (ko) | 2005-10-14 |
| DE69734479T2 (de) | 2006-06-29 |
| EP0946532B1 (de) | 2002-07-17 |
| US7795442B2 (en) | 2010-09-14 |
| EP1201662A1 (de) | 2002-05-02 |
| US20080076920A1 (en) | 2008-03-27 |
| JP4354533B2 (ja) | 2009-10-28 |
| DK0946532T3 (da) | 2002-11-11 |
| US7161011B2 (en) | 2007-01-09 |
| US6548676B1 (en) | 2003-04-15 |
| AU6205698A (en) | 1998-07-15 |
| DE69714076D1 (de) | 2002-08-22 |
| JP2001506255A (ja) | 2001-05-15 |
| EP1577307A3 (de) | 2009-04-29 |
| ATE220670T1 (de) | 2002-08-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| HP | Change in proprietorship | ||
| FF | Patent granted | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| KB | Patent renewed | ||
| MM9K | Patent not in force due to non-payment of renewal fees |